Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | v-akt murine thymoma viral oncogene homolog 1 | Starlite/ChEMBL | References |
Homo sapiens | v-akt murine thymoma viral oncogene homolog 2 | Starlite/ChEMBL | References |
Homo sapiens | v-akt murine thymoma viral oncogene homolog 3 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | protein kinase, putative | 0.014 | 0.0647 | 0.2296 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0098 | 0.0429 | 0.152 |
Trichomonas vaginalis | AGC family protein kinase | 0.0053 | 0.0193 | 0.298 |
Trypanosoma cruzi | Protein kinase B | 0.0098 | 0.0429 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0053 | 0.0193 | 0.298 |
Brugia malayi | Protein kinase domain containing protein | 0.014 | 0.0647 | 0.0463 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0135 | 0.0622 | 0.0437 |
Echinococcus multilocularis | serine:threonine protein kinase Chk2 | 0.0558 | 0.2819 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0053 | 0.0193 | 0.298 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.0016 | 0 | 0.5 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0083 | 0.0347 | 0.0587 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0093 | 0.0403 | 1 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0098 | 0.0429 | 0.0898 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0098 | 0.0429 | 0.024 |
Echinococcus multilocularis | nervana 2 | 0.0083 | 0.0347 | 0.0587 |
Entamoeba histolytica | protein kinase, putative | 0.014 | 0.0647 | 0.2296 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0093 | 0.0403 | 0.0799 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.014 | 0.0647 | 1 |
Leishmania major | protein kinase, putative | 0.0016 | 0 | 0.5 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0098 | 0.0429 | 0.0898 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0083 | 0.0347 | 0.0587 |
Echinococcus multilocularis | nervana 2 | 0.0083 | 0.0347 | 0.0587 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0135 | 0.0622 | 0.0437 |
Echinococcus granulosus | nervana 2 | 0.0083 | 0.0347 | 0.0587 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.014 | 0.0647 | 0.0463 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0093 | 0.0403 | 0.9399 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0083 | 0.0347 | 0.0587 |
Entamoeba histolytica | protein kinase 2, putative | 0.0093 | 0.0403 | 0.1429 |
Echinococcus granulosus | serine:threonine protein kinase Chk2 | 0.0558 | 0.2819 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0558 | 0.2819 | 0.2678 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0093 | 0.0403 | 0.0799 |
Toxoplasma gondii | AGC kinase | 0.0135 | 0.0622 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0053 | 0.0193 | 0.0684 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0093 | 0.0403 | 0.0799 |
Echinococcus granulosus | nervana 2 | 0.0083 | 0.0347 | 0.0587 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0098 | 0.0429 | 0.152 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0083 | 0.0347 | 0.0587 |
Entamoeba histolytica | protein kinase, putative | 0.0135 | 0.0622 | 0.2205 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Leishmania major | folate/biopterin transporter, putative | 0.0016 | 0 | 0.5 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.0016 | 0 | 0.5 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0098 | 0.0429 | 1 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0093 | 0.0403 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.1941 | 1 | 1 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.0042 | 0.0137 | 0.2119 |
Entamoeba histolytica | protein kinase, putative | 0.0558 | 0.2819 | 1 |
Loa Loa (eye worm) | CAMK/CAMKL/CHK1 protein kinase | 0.1941 | 1 | 1 |
Echinococcus multilocularis | calcium:calmodulin dependent protein kinase I | 0.0558 | 0.2818 | 0.9996 |
Entamoeba histolytica | protein kinase, putative | 0.0558 | 0.2819 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.0016 | 0 | 0.5 |
Leishmania major | protein kinase, putative | 0.0016 | 0 | 0.5 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0098 | 0.0429 | 0.024 |
Giardia lamblia | Kinase, AGC PKA | 0.0093 | 0.0403 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0058 | 0.0219 | 0.3378 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase I | 0.0558 | 0.2818 | 0.9996 |
Trichomonas vaginalis | AGC family protein kinase | 0.014 | 0.0647 | 1 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.