Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | chemokine (C-C motif) receptor 1 | Starlite/ChEMBL | References |
Species | Potential target | Known druggable target | Length | Alignment span | Identity |
---|---|---|---|---|---|
Brugia malayi | hypothetical protein | chemokine (C-C motif) receptor 1 | 355 aa | 289 aa | 21.8 % |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0127 | 0.1672 | 0.1672 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0127 | 0.1672 | 0.1672 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0123 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0178 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | hypothetical protein | 0.0178 | 0.5571 | 0.5571 |
Schistosoma mansoni | tubulin subunit alpha | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0127 | 0.1672 | 0.1672 |
Echinococcus multilocularis | hypothetical protein | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0178 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0123 | 0.1296 | 0.1296 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0123 | 0.1296 | 0.1296 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0178 | 0.5571 | 0.4682 |
Giardia lamblia | Alpha-tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0123 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0123 | 0.1296 | 0.1296 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0127 | 0.1672 | 0.1672 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0178 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0178 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0178 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0178 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0178 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0178 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0178 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0178 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | alpha-tubulin | 0.0178 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | alpha-tubulin | 0.0178 | 0.5571 | 0.5571 |
Brugia malayi | alpha-tubulin | 0.0178 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0178 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0178 | 0.5571 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 12 nM | Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cells | ChEMBL. | 23374868 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.