Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0034 | 0.1378 | 0.7844 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0205 | 1 | 1 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0041 | 0.1734 | 0.9868 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trypanosoma brucei | phosphatidylinositol 3-kinase, putative | 0.0019 | 0.0595 | 0.4987 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0041 | 0.1734 | 1 |
Toxoplasma gondii | FATC domain-containing protein | 0.0026 | 0.0952 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Btk29A | 0.0011 | 0.0194 | 0.1118 |
Brugia malayi | SRC-1 | 0.0041 | 0.1734 | 0.1734 |
Echinococcus multilocularis | growth factor receptor bound protein 2 | 0.0008 | 0.0032 | 0.0185 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Echinococcus multilocularis | PIK kinase, FAT and Armadillo domain containing protein | 0.0008 | 0.0056 | 0.0322 |
Schistosoma mansoni | tyrosine kinase | 0.0011 | 0.0194 | 0.0194 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0026 | 0.0952 | 1 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm)-related | 0.0019 | 0.0595 | 0.0595 |
Entamoeba histolytica | FKBP-rapamycin associated protein (FRAP), putative | 0.0019 | 0.0595 | 0.4433 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0011 | 0.0178 | 0.0178 |
Onchocerca volvulus | 0.0007 | 0 | 0.5 | |
Echinococcus multilocularis | tyrosine protein kinase Src64B | 0.0041 | 0.1734 | 1 |
Loa Loa (eye worm) | TK protein kinase | 0.0034 | 0.1341 | 0.1341 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Schistosoma mansoni | tyrosine kinase | 0.0041 | 0.1734 | 0.1734 |
Schistosoma mansoni | proto-oncogene tyrosine-protein kinase abl1 | 0.0008 | 0.0032 | 0.0032 |
Echinococcus granulosus | 3'partial|tyrosine protein kinase Fgr | 0.0041 | 0.1734 | 0.9868 |
Schistosoma mansoni | hypothetical protein | 0.0008 | 0.0056 | 0.0056 |
Echinococcus granulosus | PIK kinase FAT and Armadillo domain containing protein | 0.0008 | 0.0056 | 0.0318 |
Onchocerca volvulus | 0.0007 | 0 | 0.5 | |
Chlamydia trachomatis | serine/threonine protein kinase | 0.0205 | 1 | 0.5 |
Schistosoma mansoni | proto-oncogene tyrosine-protein kinase src | 0.0011 | 0.0194 | 0.0194 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0041 | 0.1734 | 0.9868 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus multilocularis | FKBP12 rapamycin complex associated protein | 0.0019 | 0.0595 | 0.3429 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0041 | 0.1734 | 0.9868 |
Brugia malayi | protein-tyrosine kinase | 0.0038 | 0.154 | 0.154 |
Schistosoma mansoni | nck2/grb4 | 0.0008 | 0.0032 | 0.0032 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0026 | 0.0952 | 0.0952 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus granulosus | serine:threonine protein kinase SMG1 | 0.0011 | 0.0178 | 0.1014 |
Echinococcus granulosus | tyrosine protein kinase Src64B | 0.0041 | 0.1734 | 0.9868 |
Echinococcus granulosus | tyrosine kinase|tyrosine protein kinase Fyn | 0.0038 | 0.154 | 0.8765 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0041 | 0.1734 | 1 |
Echinococcus granulosus | tyrosine protein kinase Blk | 0.0038 | 0.154 | 0.8765 |
Echinococcus multilocularis | serine:threonine protein kinase SMG1 | 0.0011 | 0.0178 | 0.1027 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0041 | 0.1734 | 1 |
Entamoeba histolytica | phosphatidylinositol3-kinaseTor2, putative | 0.0019 | 0.0595 | 0.4433 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Loa Loa (eye worm) | hypothetical protein | 0.0008 | 0.0056 | 0.0056 |
Echinococcus granulosus | proto oncogene tyrosine protein kinase LCK | 0.0041 | 0.1734 | 0.9868 |
Trypanosoma brucei | phosphatidylinositol 3-related kinase, putative | 0.0019 | 0.0595 | 0.4987 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0019 | 0.0595 | 0.0595 |
Entamoeba histolytica | hypothetical protein | 0.0026 | 0.0952 | 0.7093 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus granulosus | FKBP12 rapamycin complex associated protein | 0.0019 | 0.0595 | 0.3384 |
Trypanosoma cruzi | phosphatidylinositol 3-related kinase, putative | 0.0019 | 0.0595 | 0.5386 |
Echinococcus multilocularis | phosphatidylinositol 3 and 4 kinase | 0.0019 | 0.0595 | 0.3429 |
Entamoeba histolytica | protein kinase rad3, putative | 0.0011 | 0.0178 | 0.1328 |
Brugia malayi | FAT domain containing protein | 0.0008 | 0.0056 | 0.0056 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Onchocerca volvulus | 0.0007 | 0 | 0.5 | |
Trypanosoma cruzi | target of rapamycin kinase 3 | 0.0019 | 0.0595 | 0.5386 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0012 | 0.024 | 0.2052 |
Echinococcus multilocularis | tyrosine protein kinase Blk | 0.0038 | 0.154 | 0.8882 |
Echinococcus multilocularis | tyrosine protein kinase Srms | 0.0038 | 0.154 | 0.8882 |
Echinococcus multilocularis | tyrosine protein kinase Fgr | 0.0041 | 0.1734 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0034 | 0.1378 | 0.7949 |
Trypanosoma brucei | phosphatidylinositol kinase related protein, putative | 0.0026 | 0.0952 | 1 |
Echinococcus granulosus | growth factor receptor bound protein 2 | 0.0008 | 0.0032 | 0.0183 |
Echinococcus granulosus | tyrosine protein kinase Btk29A | 0.0011 | 0.0194 | 0.1103 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.0019 | 0.0595 | 0.0595 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase Abl | 0.0011 | 0.0194 | 0.1118 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0026 | 0.0952 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Brugia malayi | Tyrosine-protein kinase abl-1 | 0.0011 | 0.0194 | 0.0194 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Entamoeba histolytica | Phosphatidylinositol 3- and 4-kinase family | 0.0011 | 0.0178 | 0.1328 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Schistosoma mansoni | fkbp-rapamycin associated protein | 0.0011 | 0.0178 | 0.0178 |
Toxoplasma gondii | target of rapamycin (TOR), putative | 0.0019 | 0.0595 | 0.4987 |
Schistosoma mansoni | growth factor receptor-bound protein | 0.0008 | 0.0032 | 0.0032 |
Loa Loa (eye worm) | variant SH3 domain-containing protein | 0.0008 | 0.0032 | 0.0032 |
Entamoeba histolytica | protein kinase, putative | 0.0034 | 0.1341 | 1 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.0019 | 0.0595 | 0.4987 |
Loa Loa (eye worm) | hypothetical protein | 0.0008 | 0.0032 | 0.0032 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase HCK | 0.0034 | 0.1341 | 0.7735 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Leishmania major | phosphatidylinositol kinase related protein, putative | 0.0019 | 0.0597 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0041 | 0.1734 | 1 |
Echinococcus granulosus | tyrosine protein kinase Lyn | 0.0042 | 0.1757 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Onchocerca volvulus | 0.0007 | 0 | 0.5 | |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Schistosoma mansoni | growth factor receptor-bound protein | 0.0008 | 0.0032 | 0.0032 |
Schistosoma mansoni | adapter molecule crk | 0.0008 | 0.0032 | 0.0032 |
Brugia malayi | Variant SH3 domain containing protein | 0.0008 | 0.0032 | 0.0032 |
Onchocerca volvulus | 0.0007 | 0 | 0.5 | |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0019 | 0.0595 | 0.0595 |
Echinococcus granulosus | c src tyrosine kinase | 0.0011 | 0.0194 | 0.1103 |
Echinococcus granulosus | NCK adaptor protein | 0.0008 | 0.0032 | 0.0183 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Onchocerca volvulus | 0.0007 | 0 | 0.5 | |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0019 | 0.0595 | 0.0595 |
Schistosoma mansoni | tyrosine kinase | 0.0041 | 0.1734 | 0.1734 |
Echinococcus granulosus | tyrosine kinase | 0.0038 | 0.154 | 0.8765 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0019 | 0.0597 | 0.541 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.0019 | 0.0595 | 0.4987 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0022 | 0.0768 | 0.7623 |
Schistosoma mansoni | phosphatidylinositol 3-and 4-kinase | 0.0019 | 0.0595 | 0.0595 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Loa Loa (eye worm) | hypothetical protein | 0.0022 | 0.0768 | 0.0768 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus multilocularis | proto oncogene tyrosine protein kinase LCK | 0.0041 | 0.1734 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Brugia malayi | Sex muscle abnormal protein 5 | 0.0008 | 0.0032 | 0.0032 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor1 | 0.0019 | 0.0595 | 0.5386 |
Echinococcus granulosus | phosphatidylinositol 3 and 4 kinase | 0.0019 | 0.0595 | 0.3384 |
Loa Loa (eye worm) | hypothetical protein | 0.0012 | 0.024 | 0.024 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0041 | 0.1734 | 0.9868 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Loa Loa (eye worm) | NEK/NEK6 protein kinase | 0.0205 | 1 | 1 |
Echinococcus multilocularis | c src tyrosine kinase | 0.0011 | 0.0194 | 0.1118 |
Loa Loa (eye worm) | SRC-1 | 0.0041 | 0.1734 | 0.1734 |
Brugia malayi | Variant SH3 domain containing protein | 0.0008 | 0.0032 | 0.0032 |
Echinococcus multilocularis | serine protein kinase ATM | 0.0026 | 0.0952 | 0.5487 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor2 | 0.0019 | 0.0595 | 0.5386 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0012 | 0.024 | 0.2052 |
Trypanosoma cruzi | phosphatidylinositol 3-related kinase, putative | 0.0019 | 0.0595 | 0.5386 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm) | 0.0026 | 0.0952 | 0.0952 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Giardia lamblia | GTOR | 0.0019 | 0.0595 | 0.5 |
Echinococcus multilocularis | NCK adaptor protein | 0.0008 | 0.0032 | 0.0185 |
Loa Loa (eye worm) | hypothetical protein | 0.0011 | 0.0178 | 0.0178 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.0019 | 0.0595 | 0.4987 |
Echinococcus granulosus | tyrosine protein kinase HCK | 0.0034 | 0.1341 | 0.7634 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0019 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase lyn lyn a protein tyrosine kinase lymphocyte specific protein tyrosine kinase | 0.0041 | 0.1734 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Echinococcus multilocularis | tyrosine protein kinase lyn tyrosine protein kinase blk | 0.0041 | 0.1734 | 1 |
Schistosoma mansoni | tyrosine kinase | 0.0011 | 0.0194 | 0.0194 |
Echinococcus granulosus | serine protein kinase ATM | 0.0026 | 0.0952 | 0.5415 |
Loa Loa (eye worm) | sex muscle abnormal protein 5 | 0.0008 | 0.0032 | 0.0032 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0038 | 0.154 | 0.8882 |
Loa Loa (eye worm) | TK protein kinase | 0.0038 | 0.154 | 0.154 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | = 125 ug ml-1 | Antifungal activity against Candida albicans RCMB 05035 assessed as growth inhibition after 48 hrs by twofold serial dilution method | ChEMBL. | 23357308 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.