Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.002 | 0.0595 | 0.0595 |
Schistosoma mansoni | adapter molecule crk | 0.0008 | 0.0032 | 0.0032 |
Echinococcus multilocularis | PIK kinase, FAT and Armadillo domain containing protein | 0.0009 | 0.0056 | 0.0322 |
Schistosoma mansoni | growth factor receptor-bound protein | 0.0008 | 0.0032 | 0.0032 |
Echinococcus multilocularis | serine:threonine protein kinase SMG1 | 0.0011 | 0.0178 | 0.1027 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus multilocularis | NCK adaptor protein | 0.0008 | 0.0032 | 0.0185 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.002 | 0.0595 | 0.0595 |
Onchocerca volvulus | 0.0008 | 0 | 0.5 | |
Loa Loa (eye worm) | TK protein kinase | 0.004 | 0.1541 | 0.1541 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.002 | 0.0597 | 0.541 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0044 | 0.1735 | 0.9868 |
Toxoplasma gondii | target of rapamycin (TOR), putative | 0.002 | 0.0595 | 0.4987 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0011 | 0.0178 | 0.0178 |
Entamoeba histolytica | protein kinase, putative | 0.0036 | 0.1342 | 1 |
Trypanosoma brucei | Phosphatidylinositol 3-kinase tor1 | 0.002 | 0.0595 | 0.4987 |
Schistosoma mansoni | growth factor receptor-bound protein | 0.0008 | 0.0032 | 0.0032 |
Brugia malayi | Variant SH3 domain containing protein | 0.0008 | 0.0032 | 0.0032 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Leishmania major | phosphatidylinositol kinase related protein, putative | 0.002 | 0.0597 | 1 |
Echinococcus granulosus | tyrosine protein kinase Lyn | 0.0045 | 0.1758 | 1 |
Schistosoma mansoni | tyrosine kinase | 0.0044 | 0.1735 | 0.1735 |
Onchocerca volvulus | 0.0008 | 0 | 0.5 | |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Loa Loa (eye worm) | TK protein kinase | 0.0036 | 0.1342 | 0.1342 |
Echinococcus granulosus | NCK adaptor protein | 0.0008 | 0.0032 | 0.0183 |
Onchocerca volvulus | 0.0008 | 0 | 0.5 | |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0013 | 0.024 | 0.2052 |
Trypanosoma cruzi | phosphatidylinositol 3-related kinase, putative | 0.002 | 0.0595 | 0.5386 |
Toxoplasma gondii | FATC domain-containing protein | 0.0028 | 0.0952 | 1 |
Schistosoma mansoni | proto-oncogene tyrosine-protein kinase abl1 | 0.0008 | 0.0032 | 0.0032 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor2 | 0.002 | 0.0595 | 0.5386 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Onchocerca volvulus | 0.0008 | 0 | 0.5 | |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Brugia malayi | Phosphatidylinositol 3- and 4-kinase family protein | 0.0028 | 0.0952 | 0.0952 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus multilocularis | FKBP12 rapamycin complex associated protein | 0.002 | 0.0595 | 0.3429 |
Echinococcus multilocularis | proto oncogene tyrosine protein kinase LCK | 0.0044 | 0.1735 | 1 |
Echinococcus multilocularis | c src tyrosine kinase | 0.0012 | 0.0194 | 0.1118 |
Schistosoma mansoni | tyrosine kinase | 0.0012 | 0.0194 | 0.0194 |
Trypanosoma brucei | target of rapamycin kinase 3, putative | 0.002 | 0.0595 | 0.4987 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0037 | 0.1379 | 0.7949 |
Echinococcus granulosus | serine protein kinase ATM | 0.0028 | 0.0952 | 0.5415 |
Onchocerca volvulus | 0.0008 | 0 | 0.5 | |
Echinococcus multilocularis | tyrosine protein kinase Srms | 0.004 | 0.1541 | 0.8882 |
Echinococcus granulosus | tyrosine kinase | 0.004 | 0.1541 | 0.8765 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0044 | 0.1735 | 0.9868 |
Loa Loa (eye worm) | hypothetical protein | 0.0024 | 0.0768 | 0.0768 |
Schistosoma mansoni | phosphatidylinositol 3-and 4-kinase | 0.002 | 0.0595 | 0.0595 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trypanosoma brucei | phosphatidylinositol 4-kinase, putative | 0.002 | 0.0595 | 0.4987 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Schistosoma mansoni | tyrosine kinase | 0.0012 | 0.0194 | 0.0194 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0024 | 0.0768 | 0.7623 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase lyn tyrosine protein kinase blk | 0.0044 | 0.1735 | 1 |
Echinococcus granulosus | phosphatidylinositol 3 and 4 kinase | 0.002 | 0.0595 | 0.3384 |
Loa Loa (eye worm) | hypothetical protein | 0.0013 | 0.024 | 0.024 |
Loa Loa (eye worm) | variant SH3 domain-containing protein | 0.0008 | 0.0032 | 0.0032 |
Trypanosoma cruzi | Phosphatidylinositol 3-kinase tor1 | 0.002 | 0.0595 | 0.5386 |
Echinococcus multilocularis | tyrosine protein kinase Src64B | 0.0044 | 0.1735 | 1 |
Loa Loa (eye worm) | SRC-1 | 0.0044 | 0.1735 | 0.1735 |
Echinococcus granulosus | serine:threonine protein kinase SMG1 | 0.0011 | 0.0178 | 0.1014 |
Loa Loa (eye worm) | NEK/NEK6 protein kinase | 0.022 | 1 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Abl | 0.0012 | 0.0194 | 0.1118 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase Fgr | 0.0044 | 0.1735 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0009 | 0.0056 | 0.0056 |
Echinococcus granulosus | tyrosine protein kinase Src64B | 0.0044 | 0.1735 | 0.9868 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0037 | 0.1379 | 0.7844 |
Schistosoma mansoni | serine/threonine protein kinase | 0.022 | 1 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Echinococcus multilocularis | tyrosine protein kinase lyn lyn a protein tyrosine kinase lymphocyte specific protein tyrosine kinase | 0.0044 | 0.1735 | 1 |
Echinococcus granulosus | 3'partial|tyrosine protein kinase Fgr | 0.0044 | 0.1735 | 0.9868 |
Brugia malayi | Sex muscle abnormal protein 5 | 0.0008 | 0.0032 | 0.0032 |
Brugia malayi | FAT domain containing protein | 0.0009 | 0.0056 | 0.0056 |
Onchocerca volvulus | 0.0008 | 0 | 0.5 | |
Loa Loa (eye worm) | sex muscle abnormal protein 5 | 0.0008 | 0.0032 | 0.0032 |
Trypanosoma brucei | phosphatidylinositol kinase related protein, putative | 0.0028 | 0.0952 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0044 | 0.1735 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Blk | 0.004 | 0.1541 | 0.8882 |
Echinococcus granulosus | tyrosine protein kinase Blk | 0.004 | 0.1541 | 0.8765 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0044 | 0.1735 | 1 |
Brugia malayi | protein-tyrosine kinase | 0.004 | 0.1541 | 0.1541 |
Echinococcus granulosus | tyrosine protein kinase Btk29A | 0.0012 | 0.0194 | 0.1103 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0044 | 0.1735 | 0.9868 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.002 | 0.0595 | 0.0595 |
Echinococcus granulosus | tyrosine protein kinase HCK | 0.0036 | 0.1342 | 0.7634 |
Chlamydia trachomatis | serine/threonine protein kinase | 0.022 | 1 | 0.5 |
Brugia malayi | SRC-1 | 0.0044 | 0.1735 | 0.1735 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm) | 0.0028 | 0.0952 | 0.0952 |
Echinococcus granulosus | proto oncogene tyrosine protein kinase LCK | 0.0044 | 0.1735 | 0.9868 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Trypanosoma brucei | phosphatidylinositol 3-kinase, putative | 0.002 | 0.0595 | 0.4987 |
Brugia malayi | Variant SH3 domain containing protein | 0.0008 | 0.0032 | 0.0032 |
Loa Loa (eye worm) | hypothetical protein | 0.0011 | 0.0178 | 0.0178 |
Schistosoma mansoni | hypothetical protein | 0.0009 | 0.0056 | 0.0056 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0044 | 0.1735 | 1 |
Entamoeba histolytica | Phosphatidylinositol 3- and 4-kinase family | 0.0011 | 0.0178 | 0.1328 |
Schistosoma mansoni | proto-oncogene tyrosine-protein kinase src | 0.0012 | 0.0194 | 0.0194 |
Echinococcus multilocularis | growth factor receptor bound protein 2 | 0.0008 | 0.0032 | 0.0185 |
Entamoeba histolytica | hypothetical protein | 0.0028 | 0.0952 | 0.7093 |
Schistosoma mansoni | ataxia telangiectasia mutated (atm)-related | 0.002 | 0.0595 | 0.0595 |
Entamoeba histolytica | FKBP-rapamycin associated protein (FRAP), putative | 0.002 | 0.0595 | 0.4433 |
Schistosoma mansoni | nck2/grb4 | 0.0008 | 0.0032 | 0.0032 |
Trypanosoma cruzi | target of rapamycin kinase 3 | 0.002 | 0.0595 | 0.5386 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0013 | 0.024 | 0.2052 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0028 | 0.0952 | 1 |
Echinococcus granulosus | growth factor receptor bound protein 2 | 0.0008 | 0.0032 | 0.0183 |
Echinococcus granulosus | tyrosine kinase|tyrosine protein kinase Fyn | 0.004 | 0.1541 | 0.8765 |
Echinococcus multilocularis | tyrosine protein kinase HCK | 0.0036 | 0.1342 | 0.7735 |
Schistosoma mansoni | tyrosine kinase | 0.0044 | 0.1735 | 0.1735 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.004 | 0.1541 | 0.8882 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Brugia malayi | Tyrosine-protein kinase abl-1 | 0.0012 | 0.0194 | 0.0194 |
Echinococcus granulosus | FKBP12 rapamycin complex associated protein | 0.002 | 0.0595 | 0.3384 |
Echinococcus multilocularis | phosphatidylinositol 3 and 4 kinase | 0.002 | 0.0595 | 0.3429 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus granulosus | c src tyrosine kinase | 0.0012 | 0.0194 | 0.1103 |
Echinococcus multilocularis | serine protein kinase ATM | 0.0028 | 0.0952 | 0.5487 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Entamoeba histolytica | protein kinase rad3, putative | 0.0011 | 0.0178 | 0.1328 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0044 | 0.1735 | 0.9868 |
Trypanosoma brucei | phosphatidylinositol 3-related kinase, putative | 0.002 | 0.0595 | 0.4987 |
Giardia lamblia | GTOR | 0.002 | 0.0595 | 0.5 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.0011 | 0.0178 | 0.1365 |
Loa Loa (eye worm) | hypothetical protein | 0.0008 | 0.0032 | 0.0032 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0044 | 0.1735 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trypanosoma cruzi | phosphatidylinositol kinase related protein, putative | 0.0028 | 0.0952 | 1 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Echinococcus granulosus | PIK kinase FAT and Armadillo domain containing protein | 0.0009 | 0.0056 | 0.0318 |
Schistosoma mansoni | fkbp-rapamycin associated protein | 0.0011 | 0.0178 | 0.0178 |
Trichomonas vaginalis | PIKK family atypical protein kinase | 0.002 | 0.0595 | 0.6016 |
Trypanosoma cruzi | phosphatidylinositol 3-related kinase, putative | 0.002 | 0.0595 | 0.5386 |
Loa Loa (eye worm) | phosphatidylinositol 3 | 0.002 | 0.0595 | 0.0595 |
Entamoeba histolytica | phosphatidylinositol3-kinaseTor2, putative | 0.002 | 0.0595 | 0.4433 |
Echinococcus multilocularis | tyrosine protein kinase Btk29A | 0.0012 | 0.0194 | 0.1118 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IZ (functional) | = 10 mm | Antibacterial activity against Escherichia coli assessed as growth inhibition at 1 mg/ml by cup-plate method | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.