Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | potassium voltage-gated channel, shaker-related subfamily, member 5 | Starlite/ChEMBL | References |
Species | Potential target | Known druggable target | Length | Alignment span | Identity |
---|---|---|---|---|---|
Echinococcus multilocularis | voltage gated potassium channel | potassium voltage-gated channel, shaker-related subfamily, member 5 | 613 aa | 521 aa | 34.9 % |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Schistosoma mansoni | sodium-dependent neurotransmitter transporter | 0.0025 | 0.0025 | 0.0025 |
Echinococcus multilocularis | vesicular acetylcholine transporter | 0.4843 | 1 | 1 |
Toxoplasma gondii | hypothetical protein | 0.0025 | 0.0025 | 0.5 |
Loa Loa (eye worm) | solute carrier family 6 member 4 | 0.0148 | 0.028 | 0.0255 |
Brugia malayi | Voltage-gated potassium channel, Shaker-family (KCNA, Kv1-like) alpha-subunit | 0.0104 | 0.0188 | 0.0163 |
Trypanosoma cruzi | C-8 sterol isomerase, putative | 0.2284 | 0.4702 | 0.5 |
Loa Loa (eye worm) | serotonin transporter b | 0.0148 | 0.028 | 0.0255 |
Echinococcus granulosus | serotonin transporter | 0.0148 | 0.028 | 0.0255 |
Echinococcus granulosus | potassium voltage gated channel subfamily A | 0.0104 | 0.0188 | 0.0163 |
Schistosoma mansoni | sodium-dependent neurotransmitter transporter | 0.0025 | 0.0025 | 0.0025 |
Loa Loa (eye worm) | hypothetical protein | 0.0148 | 0.028 | 0.0255 |
Chlamydia trachomatis | Ssodium-dependent amino acid transporter | 0.0025 | 0.0025 | 0.5 |
Brugia malayi | ERG2 and Sigma1 receptor like protein | 0.2284 | 0.4702 | 0.4688 |
Schistosoma mansoni | norepinephrine/norepinephrine transporter | 0.0025 | 0.0025 | 0.0025 |
Plasmodium vivax | hypothetical protein, conserved | 0.0025 | 0.0025 | 0.5 |
Loa Loa (eye worm) | vesicular acetylcholine transporter unc-17 | 0.4843 | 1 | 1 |
Brugia malayi | Sodium:neurotransmitter symporter family protein | 0.0148 | 0.028 | 0.0255 |
Toxoplasma gondii | Sodium:neurotransmitter symporter family protein | 0.0025 | 0.0025 | 0.5 |
Onchocerca volvulus | 0.0148 | 0.028 | 0.0255 | |
Echinococcus multilocularis | serotonin transporter | 0.0148 | 0.028 | 0.0255 |
Schistosoma mansoni | vesicular acetylcholine transporter | 0.4843 | 1 | 1 |
Toxoplasma gondii | hypothetical protein | 0.0025 | 0.0025 | 0.5 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0104 | 0.0188 | 0.0188 |
Loa Loa (eye worm) | norepinephrine transporter | 0.0148 | 0.028 | 0.0255 |
Treponema pallidum | sodium- and chloride- dependent transporter | 0.0148 | 0.028 | 0.5 |
Toxoplasma gondii | Sodium:neurotransmitter symporter family protein | 0.0025 | 0.0025 | 0.5 |
Schistosoma mansoni | sodium/chloride dependent neurotransmitter transporter | 0.0025 | 0.0025 | 0.0025 |
Schistosoma mansoni | sodium/chloride dependent transporter | 0.0025 | 0.0025 | 0.0025 |
Plasmodium vivax | amine transporter, putative | 0.0025 | 0.0025 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0148 | 0.028 | 0.0255 |
Schistosoma mansoni | sodium-dependent amino acid transporter | 0.0025 | 0.0025 | 0.0025 |
Plasmodium falciparum | amino acid transporter, putative | 0.0025 | 0.0025 | 0.5 |
Schistosoma mansoni | sodium/chloride dependent transporter | 0.0148 | 0.028 | 0.028 |
Plasmodium falciparum | transporter, putative | 0.0025 | 0.0025 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.1167 | 0.239 | 0.2371 |
Schistosoma mansoni | sodium-dependent neurotransmitter transporter | 0.0025 | 0.0025 | 0.0025 |
Schistosoma mansoni | voltage-gated potassium channel | 0.0104 | 0.0188 | 0.0188 |
Toxoplasma gondii | Sodium:neurotransmitter symporter family protein | 0.0025 | 0.0025 | 0.5 |
Schistosoma mansoni | sodium/chloride dependent transporter | 0.0025 | 0.0025 | 0.0025 |
Echinococcus granulosus | vesicular acetylcholine transporter | 0.4843 | 1 | 1 |
Onchocerca volvulus | Vesicular acetylcholine transporter homolog | 0.4843 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.2284 | 0.4702 | 0.4688 |
Echinococcus multilocularis | potassium voltage gated channel protein | 0.0104 | 0.0188 | 0.0163 |
Schistosoma mansoni | sodium/chloride dependent neurotransmitter transporter | 0.0025 | 0.0025 | 0.0025 |
Leishmania major | C-8 sterol isomerase-like protein | 0.2284 | 0.4702 | 0.5 |
Schistosoma mansoni | norepinephrine/norepinephrine transporter | 0.0025 | 0.0025 | 0.0025 |
Schistosoma mansoni | sodium/chloride dependent neurotransmitter transporter | 0.0025 | 0.0025 | 0.0025 |
Schistosoma mansoni | norepinephrine/norepinephrine transporter | 0.0148 | 0.028 | 0.028 |
Loa Loa (eye worm) | hypothetical protein | 0.0148 | 0.028 | 0.0255 |
Trypanosoma brucei | C-8 sterol isomerase, putative | 0.2284 | 0.4702 | 0.5 |
Echinococcus multilocularis | potassium voltage gated channel subfamily A | 0.0099 | 0.0179 | 0.0154 |
Loa Loa (eye worm) | hypothetical protein | 0.0104 | 0.0188 | 0.0163 |
Echinococcus granulosus | potassium voltage gated channel protein | 0.0104 | 0.0188 | 0.0163 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.