Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | transient receptor potential cation channel, subfamily V, member 1 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | tubulin family protein | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.004 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | BEN-1 protein | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.004 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0103 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0103 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0103 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.004 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0103 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0103 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0103 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.004 | 0.2166 | 0.2166 |
Trypanosoma brucei | alpha tubulin | 0.004 | 0.2166 | 0.2166 |
Toxoplasma gondii | beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0103 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0103 | 1 | 1 |
Onchocerca volvulus | 0.0023 | 0 | 0.5 | |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.004 | 0.2166 | 0.2166 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.004 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.004 | 0.2166 | 0.2166 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.004 | 0.2166 | 0.2166 |
Brugia malayi | Tubulin alpha-2 chain | 0.004 | 0.2166 | 0.2166 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.004 | 0.2166 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0103 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.004 | 0.2166 | 0.2166 |
Echinococcus multilocularis | tubulin subunit beta | 0.0103 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0103 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0103 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.004 | 0.2166 | 0.2166 |
Brugia malayi | Tubulin alpha-2 chain | 0.004 | 0.2166 | 0.2166 |
Trypanosoma brucei | tubulin gamma chain | 0.004 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | tubulin alpha chain | 0.004 | 0.2166 | 0.2166 |
Plasmodium vivax | tubulin beta chain, putative | 0.0103 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0103 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.004 | 0.2166 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.004 | 0.2166 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0103 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.004 | 0.2166 | 0.2166 |
Trypanosoma brucei | alpha tubulin | 0.004 | 0.2166 | 0.2166 |
Entamoeba histolytica | tubulin family protein | 0.0103 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0103 | 1 | 1 |
Brugia malayi | tubulin alpha-2 chain | 0.004 | 0.2166 | 0.2166 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.004 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | hypothetical protein | 0.004 | 0.2166 | 0.2166 |
Schistosoma mansoni | tubulin subunit beta | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.004 | 0.2166 | 0.2166 |
Echinococcus multilocularis | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0103 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.004 | 0.2166 | 0.2166 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0103 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0103 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0103 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.004 | 0.2166 | 0.2166 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0103 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Brugia malayi | Tubulin gamma chain | 0.004 | 0.2166 | 0.2166 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.004 | 0.2166 | 0.2166 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.004 | 0.2166 | 0.2166 |
Trypanosoma brucei | beta tubulin | 0.004 | 0.2166 | 0.2166 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0103 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0103 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.004 | 0.2166 | 0.2166 |
Giardia lamblia | Beta tubulin | 0.0103 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0103 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.004 | 0.2166 | 0.2166 |
Brugia malayi | tubulin alpha chain - mouse | 0.004 | 0.2166 | 0.2166 |
Echinococcus granulosus | beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Leishmania major | beta tubulin | 0.0103 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.004 | 0.2166 | 0.2166 |
Trypanosoma brucei | alpha tubulin | 0.004 | 0.2166 | 0.2166 |
Loa Loa (eye worm) | BEN-1 protein | 0.0103 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
EC50 (functional) | = 25.5 nM | Agonist activity at human recombinant TRPV1 expressed in human HEK293 cells | ChEMBL. | 17046253 |
EC50 (functional) | = 25.5 nM | Agonist activity at human recombinant TRPV1 expressed in human HEK293 cells | ChEMBL. | 17046253 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.