Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Brugia malayi | tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.012 | 0.1296 | 0.1296 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0125 | 0.1672 | 0.1672 |
Brugia malayi | Tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0175 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin family protein | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0231 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0231 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0125 | 0.1672 | 0.1672 |
Brugia malayi | Tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit beta | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0125 | 0.1672 | 0.1672 |
Giardia lamblia | Beta tubulin | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Giardia lamblia | Beta tubulin | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin beta chain | 0.0231 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0175 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0175 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin beta chain, putative | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0231 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Brugia malayi | Tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0125 | 0.1672 | 0.1672 |
Schistosoma mansoni | tubulin subunit alpha | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha chain - mouse | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0175 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.012 | 0.1296 | 0.1296 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | alpha-tubulin | 0.0175 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.012 | 0.1296 | 0.1296 |
Loa Loa (eye worm) | BEN-1 protein | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | hypothetical protein | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin, putative | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Brugia malayi | alpha-tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0175 | 0.5571 | 0.5571 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0231 | 1 | 1 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0175 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 1 | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.5571 |
Toxoplasma gondii | beta-tubulin, putative | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma cruzi | beta tubulin, putative | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0231 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.012 | 0.1296 | 0.1296 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0175 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0175 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Schistosoma mansoni | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin subunit TubB | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.012 | 0.1296 | 0.1296 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0231 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
ED50 (functional) | = 6.2 mg kg-1 | Antiinflammatory activity of the perorally administered compound assessed in adjuvant arthritis assay in rat | ChEMBL. | 2527995 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.