Species | Target name | Source | Bibliographic reference |
---|---|---|---|
Homo sapiens | ribosomal protein S6 kinase, 70kDa, polypeptide 1 | Starlite/ChEMBL | References |
Homo sapiens | 3-phosphoinositide dependent protein kinase 1 | Starlite/ChEMBL | References |
Homo sapiens | v-akt murine thymoma viral oncogene homolog 1 | Starlite/ChEMBL | References |
Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.0058 | 0.4605 | 0.8803 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0061 | 0.5205 | 0.5109 |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.0059 | 0.4802 | 0.9195 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.0091 | 1 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0061 | 0.5205 | 1 |
Toxoplasma gondii | AGC kinase | 0.0088 | 0.9597 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0031 | 0.0196 | 0.0196 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.0061 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.0059 | 0.4802 | 0.9195 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.0058 | 0.4605 | 0.8803 |
Echinococcus granulosus | nervana 2 | 0.0058 | 0.4605 | 0.8803 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.0059 | 0.4802 | 0.5 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0059 | 0.4884 | 0.936 |
Echinococcus multilocularis | nervana 2 | 0.0058 | 0.4605 | 0.8803 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.0061 | 0.5205 | 1 |
Brugia malayi | phosphoinositide-dependent protein kinase I | 0.0059 | 0.4884 | 0.4782 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.0061 | 0.5205 | 0.5109 |
Trichomonas vaginalis | AGC family protein kinase | 0.0059 | 0.4884 | 0.4884 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0088 | 0.9597 | 0.9589 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0059 | 0.4884 | 0.4782 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.0058 | 0.4605 | 0.8803 |
Loa Loa (eye worm) | AGC/PDK1 protein kinase | 0.0059 | 0.4884 | 0.4782 |
Echinococcus granulosus | nervana 2 | 0.0058 | 0.4605 | 0.8803 |
Echinococcus granulosus | 3-phosphoinositide-dependent protein kinase 1 | 0.0059 | 0.4884 | 0.936 |
Entamoeba histolytica | protein kinase 2, putative | 0.0059 | 0.4802 | 0.4697 |
Trypanosoma cruzi | Protein kinase B | 0.0061 | 0.5205 | 1 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0091 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0059 | 0.4884 | 0.4884 |
Trichomonas vaginalis | AGC family protein kinase | 0.0031 | 0.0196 | 0.0196 |
Trichomonas vaginalis | AGC family protein kinase | 0.0059 | 0.4884 | 0.4884 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0088 | 0.9597 | 0.9589 |
Giardia lamblia | Kinase, AGC PKA | 0.0059 | 0.4802 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.0088 | 0.9597 | 0.9589 |
Trichomonas vaginalis | AGC family protein kinase | 0.0031 | 0.0196 | 0.0196 |
Entamoeba histolytica | protein kinase, putative | 0.0091 | 1 | 1 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.0059 | 0.4802 | 0.9195 |
Echinococcus granulosus | serine/threonine protein kinase | 0.0061 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.0059 | 0.4884 | 0.4782 |
Echinococcus multilocularis | nervana 2 | 0.0058 | 0.4605 | 0.8803 |
Entamoeba histolytica | protein kinase, putative | 0.0091 | 1 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.0058 | 0.4605 | 0.8803 |
Echinococcus multilocularis | 3 phosphoinositide dependent protein kinase 1 | 0.0059 | 0.4884 | 0.936 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.0059 | 0.4884 | 0.4782 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.0059 | 0.4802 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0033 | 0.06 | 0.06 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.0061 | 0.5205 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0091 | 1 | 1 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.