Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0173 | 0.2067 | 0.2067 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0224 | 0.439 | 0.2928 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0224 | 0.439 | 0.439 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0149 | 0.1021 | 0.1021 |
Entamoeba histolytica | tubulin family protein | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0224 | 0.439 | 0.439 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0224 | 0.439 | 0.439 |
Trypanosoma brucei | beta tubulin | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0349 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0349 | 1 | 1 |
Echinococcus granulosus | tubulin subunit TubB | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0224 | 0.439 | 0.439 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | tubulin beta chain | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0149 | 0.1021 | 0.1021 |
Schistosoma mansoni | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Brugia malayi | tubulin alpha-2 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0224 | 0.439 | 0.2928 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0349 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Giardia lamblia | Alpha-tubulin | 0.0224 | 0.439 | 0.2928 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Schistosoma mansoni | tubulin subunit beta | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0349 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0224 | 0.439 | 0.439 |
Schistosoma mansoni | tubulin subunit alpha | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0149 | 0.1021 | 0.1021 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0224 | 0.439 | 0.439 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Schistosoma mansoni | tubulin subunit beta | 0.0349 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0224 | 0.439 | 0.2928 |
Giardia lamblia | Beta tubulin | 0.0349 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0224 | 0.439 | 0.2928 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0224 | 0.439 | 0.439 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0224 | 0.439 | 0.439 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0173 | 0.2067 | 0.2067 |
Toxoplasma gondii | beta-tubulin, putative | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0173 | 0.2067 | 0.2067 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Giardia lamblia | Beta tubulin | 0.0349 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0149 | 0.1021 | 0.1021 |
Giardia lamblia | Beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0349 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Trypanosoma brucei | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0224 | 0.439 | 0.439 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0349 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Plasmodium falciparum | alpha tubulin 2 | 0.0224 | 0.439 | 0.2928 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0224 | 0.439 | 0.2928 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0224 | 0.439 | 0.2928 |
Brugia malayi | Tubulin alpha-2 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0173 | 0.2067 | 0.2067 |
Schistosoma mansoni | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | tubulin subunit beta | 0.0349 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0224 | 0.439 | 0.439 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0224 | 0.439 | 0.439 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0349 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | alpha-tubulin | 0.0224 | 0.439 | 0.439 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0224 | 0.439 | 0.2928 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0224 | 0.439 | 0.439 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0224 | 0.439 | 0.2928 |
Brugia malayi | Tubulin alpha-2 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | beta tubulin | 0.0349 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0349 | 1 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0149 | 0.1021 | 0.1021 |
Plasmodium falciparum | tubulin beta chain | 0.0349 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0224 | 0.439 | 0.2928 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0349 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0224 | 0.439 | 0.2928 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0224 | 0.439 | 0.2928 |
Trypanosoma brucei | beta tubulin | 0.0349 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0349 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0349 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Trypanosoma brucei | beta tubulin | 0.0349 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0224 | 0.439 | 0.439 |
Leishmania major | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0224 | 0.439 | 0.2928 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | beta tubulin | 0.0349 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0224 | 0.439 | 0.2928 |
Schistosoma mansoni | tubulin subunit beta | 0.0349 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0224 | 0.439 | 0.2928 |
Trypanosoma brucei | alpha tubulin | 0.0224 | 0.439 | 0.2928 |
Trichomonas vaginalis | tubulin, putative | 0.0349 | 1 | 1 |
Leishmania major | beta tubulin | 0.0349 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0224 | 0.439 | 0.2928 |
Echinococcus multilocularis | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Entamoeba histolytica | tubulin family protein | 0.0349 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0224 | 0.439 | 0.2928 |
Brugia malayi | alpha-tubulin | 0.0224 | 0.439 | 0.2928 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0224 | 0.439 | 0.439 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0224 | 0.439 | 0.2928 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0349 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0349 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (ADMET) | Inhibition of human CYP3A4 at 10 uM | ChEMBL. | 27072905 | |
Inhibition (binding) | Inhibition of human norepinephrine transporter at 10 uM | ChEMBL. | 27072905 | |
Inhibition (binding) | Inhibition of human SERT at 10 uM | ChEMBL. | 27072905 | |
Inhibition (ADMET) | Inhibition of human CYP2C19 at 10 uM | ChEMBL. | 27072905 | |
Inhibition (ADMET) | = 67 % | Inhibition of human CYP2D6 at 10 uM | ChEMBL. | 27072905 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.