Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Brugia malayi | beta-tubulin, identical | 0.03 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.02 | 0.4599 | 0.3252 |
Loa Loa (eye worm) | hypothetical protein | 0.02 | 0.4599 | 0.4599 |
Trypanosoma brucei | beta tubulin | 0.03 | 1 | 1 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Plasmodium vivax | tubulin alpha chain, putative | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.02 | 0.4599 | 0.3252 |
Plasmodium falciparum | alpha tubulin 1 | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | tubulin subunit alpha | 0.02 | 0.4599 | 0.3252 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.03 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.03 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.03 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.107 | 0.107 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.03 | 1 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Entamoeba histolytica | tubulin family protein | 0.03 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.03 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.03 | 1 | 1 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.02 | 0.4599 | 0.4599 |
Brugia malayi | alpha-tubulin | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin, putative | 0.03 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.02 | 0.4599 | 0.3252 |
Trypanosoma brucei | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | tubulin subunit beta | 0.03 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | beta tubulin | 0.03 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Trypanosoma cruzi | alpha tubulin, putative | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.02 | 0.4599 | 0.3252 |
Loa Loa (eye worm) | tubulin alpha chain | 0.02 | 0.4599 | 0.4599 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.03 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.02 | 0.4599 | 0.4599 |
Brugia malayi | Tubulin alpha-2 chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.02 | 0.4599 | 0.4599 |
Loa Loa (eye worm) | alpha-tubulin | 0.02 | 0.4599 | 0.4599 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | tubulin subunit alpha | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.02 | 0.4599 | 0.4599 |
Echinococcus multilocularis | tubulin subunit beta | 0.03 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.03 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.03 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0151 | 0.1997 | 0.1997 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Brugia malayi | Tubulin alpha-2 chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.02 | 0.4599 | 0.4599 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.02 | 0.4599 | 0.4599 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0134 | 0.107 | 0.107 |
Echinococcus granulosus | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Giardia lamblia | Alpha-tubulin | 0.02 | 0.4599 | 0.3252 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.03 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | beta tubulin | 0.03 | 1 | 1 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.03 | 1 | 1 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | tubulin subunit beta | 0.03 | 1 | 1 |
Brugia malayi | tubulin alpha-2 chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.03 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Loa Loa (eye worm) | BEN-1 protein | 0.03 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.03 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | beta tubulin | 0.03 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0134 | 0.107 | 0.107 |
Giardia lamblia | Beta tubulin | 0.03 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.03 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.03 | 1 | 1 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.02 | 0.4599 | 0.3252 |
Brugia malayi | Tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0151 | 0.1997 | 0.1997 |
Toxoplasma gondii | beta-tubulin, putative | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0151 | 0.1997 | 0.1997 |
Giardia lamblia | Beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.02 | 0.4599 | 0.3252 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | tubulin subunit beta | 0.03 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.02 | 0.4599 | 0.4599 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.02 | 0.4599 | 0.4599 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.02 | 0.4599 | 0.3252 |
Schistosoma mansoni | tubulin subunit beta | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.02 | 0.4599 | 0.4599 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0134 | 0.107 | 0.107 |
Entamoeba histolytica | tubulin family protein | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.02 | 0.4599 | 0.4599 |
Echinococcus multilocularis | tubulin subunit TubB | 0.02 | 0.4599 | 0.3252 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0151 | 0.1997 | 0.1997 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.02 | 0.4599 | 0.3252 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.02 | 0.4599 | 0.4599 |
Echinococcus granulosus | tubulin subunit TubB | 0.02 | 0.4599 | 0.3252 |
Loa Loa (eye worm) | hypothetical protein | 0.0134 | 0.107 | 0.107 |
Plasmodium vivax | tubulin alpha chain, putative | 0.02 | 0.4599 | 0.3252 |
Loa Loa (eye worm) | tubulin beta chain | 0.03 | 1 | 1 |
Leishmania major | alpha tubulin | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | tubulin alpha chain | 0.02 | 0.4599 | 0.3252 |
Echinococcus granulosus | tubulin beta 1 chain | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Leishmania major | beta tubulin | 0.03 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.03 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.03 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.03 | 1 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.03 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.03 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.03 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.02 | 0.4599 | 0.4599 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 55.41 % | Activity at human carbonic anhydrase 2 assessed as hydrolysis of p- nitrophenyl acetate at 0.3 umol/L at pH 7.6 | ChEMBL. | 21524585 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.