TDR Targets

Basic information

Technical information

TDR Targets ID: 1614849
Name: N-[2-[(2Z)-2-[(2-chlorophenyl)methylidene]hyd razinyl]-4-thiophen-2-yl-1,3-thiazol-5-yl]ace tamide
MW: 376.884 | Formula: C16H13ClN4OS2
H donors: 2 H acceptors: 2 LogP: 4.42 Rotable bonds: 6
Rule of 5 violations (Lipinski): 1
SMILES: CC(=O)Nc1sc(nc1c1cccs1)N/N=C\c1ccccc1Cl
InChi: 1S/C16H13ClN4OS2/c1-10(22)19-15-14(13-7-4-8-23-13)20-16(24-15)21-18-9-11-5-2-3-6-12(11)17/h2-9H,1H3,(H,19,22)(H,20,21)/b18-9-
InChiKey: UGEVKEQAVXQQIO-NVMNQCDNSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

N-[2-[(N'Z)-N'-[(2-chlorophenyl)methylene]hydrazino]-4-(2-thienyl)thiazol-5-yl]acetamide
N-[2-[(N'Z)-N'-[(2-chlorophenyl)methylene]hydrazino]-4-(2-thienyl)-5-thiazolyl]acetamide
N-[2-[(N'Z)-N'-(2-chlorobenzylidene)hydrazino]-4-(2-thienyl)thiazol-5-yl]acetamide
N-[2-[(2Z)-2-[(2-chlorophenyl)methylidene]hydrazinyl]-4-thiophen-2-yl-1,3-thiazol-5-yl]ethanamide
STOCK3S-54759

Targets

Known targets for this compound

Species	Target name	Source	Bibliographic reference
Homo sapiens	apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3D	Starlite/ChEMBL	No references
Homo sapiens	glucagon-like peptide 1 receptor	Starlite/ChEMBL	No references
Homo sapiens	ATPase family, AAA domain containing 5	Starlite/ChEMBL	No references
Homo sapiens	lamin A/C	Starlite/ChEMBL	No references
Homo sapiens	hydroxyprostaglandin dehydrogenase 15-(NAD)	Starlite/ChEMBL	No references
Homo sapiens	nuclear factor, erythroid 2-like 2	Starlite/ChEMBL	No references

Predicted pathogen targets for this compound

By orthology

Species	Potential target	Known druggable target/s	Ortholog Group
Echinococcus multilocularis	musashi	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma japonicum	expressed protein	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus granulosus	lamin	Get druggable targets OG5_128723	All targets in OG5_128723
Loa Loa (eye worm)	hypothetical protein	Get druggable targets OG5_128723	All targets in OG5_128723
Onchocerca volvulus		Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma mansoni	lamin	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus multilocularis	lamin	Get druggable targets OG5_128723	All targets in OG5_128723
Loa Loa (eye worm)	intermediate filament tail domain-containing protein	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma japonicum	Intermediate filament protein ifa-1, putative	Get druggable targets OG5_128723	All targets in OG5_128723
Brugia malayi	intermediate filament protein	Get druggable targets OG5_128723	All targets in OG5_128723
Loa Loa (eye worm)	hypothetical protein	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma japonicum	Lamin-C, putative	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma mansoni	lamin	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma japonicum	ko:K07611 lamin, putative	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma japonicum	expressed protein	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus granulosus	intermediate filament protein	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus granulosus	lamin dm0	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus granulosus	cytoplasmic intermediate filament protein	Get druggable targets OG5_128723	All targets in OG5_128723
Brugia malayi	Intermediate filament tail domain containing protein	Get druggable targets OG5_128723	All targets in OG5_128723
Onchocerca volvulus		Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus multilocularis	cytoplasmic intermediate filament protein	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus multilocularis	lamin dm0	Get druggable targets OG5_128723	All targets in OG5_128723
Loa Loa (eye worm)	hypothetical protein	Get druggable targets OG5_128723	All targets in OG5_128723
Schistosoma mansoni	intermediate filament proteins	Get druggable targets OG5_128723	All targets in OG5_128723
Loa Loa (eye worm)	hypothetical protein	Get druggable targets OG5_128723	All targets in OG5_128723
Echinococcus multilocularis	atpase aaa+ type core atpase aaa type core	Get druggable targets OG5_139225	All targets in OG5_139225
Loa Loa (eye worm)	intermediate filament protein	Get druggable targets OG5_128723	All targets in OG5_128723
Loa Loa (eye worm)	hypothetical protein	Get druggable targets OG5_128723	All targets in OG5_128723

By sequence similarity to non orthologous known druggable targets

Species	Potential target	Known druggable target	Length	Alignment span	Identity
Loa Loa (eye worm)	pigment dispersing factor receptor c	glucagon-like peptide 1 receptor	463 aa	388 aa	25.8 %
Plasmodium falciparum	steroid dehydrogenase, putative	hydroxyprostaglandin dehydrogenase 15-(NAD)	266 aa	216 aa	22.2 %

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Trypanosoma cruzi	zinc carboxypeptidase, putative	0.0124	0.1096	0.5
Leishmania major	zinc carboxypeptidase, putative,metallo-peptidase, Clan MC, Family M14	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Loa Loa (eye worm)	hypothetical protein	0.006	0.0429	0.0709
Echinococcus granulosus	subfamily M14A unassigned peptidase	0.0724	0.7342	1
Echinococcus multilocularis	cytosolic carboxypeptidase protein 5	0.0124	0.1096	0.1096
Entamoeba histolytica	hypothetical protein	0.0043	0.0254	0.5
Echinococcus granulosus	cytosolic carboxypeptidase 1	0.0124	0.1096	0.1493
Schistosoma mansoni	peptidase	0.0124	0.1096	0.1493
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Schistosoma mansoni	intermediate filament proteins	0.0033	0.0141	0.0192
Entamoeba histolytica	hypothetical protein	0.0043	0.0254	0.5
Onchocerca volvulus		0.0724	0.7342	1
Loa Loa (eye worm)	zinc carboxypeptidase	0.0124	0.1096	0.1812
Onchocerca volvulus		0.0124	0.1096	0.1327
Brugia malayi	Corticotropin releasing factor receptor 2 precursor, putative	0.006	0.0429	0.2518
Echinococcus granulosus	lamin dm0	0.0033	0.0141	0.0192
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Echinococcus multilocularis		0.0124	0.1096	0.1096
Echinococcus multilocularis	lamin	0.0033	0.0141	0.0141
Trypanosoma cruzi	metallo-peptidase, Clan MC, Family M14	0.0124	0.1096	0.5
Echinococcus granulosus	intermediate filament protein	0.0033	0.0141	0.0192
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.06	0.6047	1
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Brugia malayi	Intermediate filament tail domain containing protein	0.0033	0.0141	0.0827
Giardia lamblia	Nuclear ATP/GTP-binding protein	0.0124	0.1096	0.5
Toxoplasma gondii	zinc carboxypeptidase superfamily protein	0.0124	0.1096	0.5
Schistosoma mansoni	subfamily M14A unassigned peptidase (M14 family)	0.0724	0.7342	1
Echinococcus multilocularis	subfamily M14A unassigned peptidase	0.0724	0.7342	0.7342
Onchocerca volvulus		0.0724	0.7342	1
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Schistosoma mansoni	protease m14 carboxypeptidase	0.0124	0.1096	0.1493
Onchocerca volvulus	Cytosolic carboxypeptidase 1 homolog	0.0124	0.1096	0.1327
Schistosoma mansoni	metallocarboxypeptidase D peptidase unit 2 (M14 family)	0.0124	0.1096	0.1493
Echinococcus multilocularis	lamin dm0	0.0033	0.0141	0.0141
Trypanosoma brucei	metallo-peptidase, Clan MC, Family M14, putative	0.0124	0.1096	0.5
Toxoplasma gondii	zinc carboxypeptidase superfamily protein	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0041	0.023	0.0381
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0033	0.0141	0.0233
Onchocerca volvulus		0.0724	0.7342	1
Schistosoma mansoni	hypothetical protein	0.0043	0.0254	0.0346
Trypanosoma cruzi	metallo-peptidase, Clan MC, Family M14, putative	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0182	0.1702	0.2815
Giardia lamblia	Nuclear ATP/GTP-binding protein	0.0124	0.1096	0.5
Schistosoma mansoni	lamin	0.0033	0.0141	0.0192
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Leishmania major	zinc carboxypeptidase, putative,metallo-peptidase, Clan MC, Family M14	0.0124	0.1096	0.5
Echinococcus multilocularis	Basic leucine zipper (bZIP) transcription	0.0043	0.0254	0.0254
Schistosoma mansoni	transcription factor LCR-F1	0.0043	0.0254	0.0346
Trypanosoma brucei	Carboxypeptidase-like protein	0.0124	0.1096	0.5
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Onchocerca volvulus	Carboxypeptidase D homolog	0.0124	0.1096	0.1327
Schistosoma mansoni	peptidase	0.0124	0.1096	0.1493
Trypanosoma cruzi	Carboxypeptidase-like protein	0.0124	0.1096	0.5
Loa Loa (eye worm)	intermediate filament tail domain-containing protein	0.0033	0.0141	0.0233
Loa Loa (eye worm)	zinc carboxypeptidase	0.0124	0.1096	0.1812
Onchocerca volvulus		0.0724	0.7342	1
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Brugia malayi	Carboxypeptidase A2 precursor	0.0124	0.1096	0.6439
Loa Loa (eye worm)	pigment dispersing factor receptor c	0.006	0.0429	0.0709
Toxoplasma gondii	flagellar/basal body protein	0.0124	0.1096	0.5
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Loa Loa (eye worm)	zinc carboxypeptidase	0.0124	0.1096	0.1812
Schistosoma mansoni	peptidase	0.0124	0.1096	0.1493
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0032	0.0135	0.0223
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Brugia malayi	hypothetical protein	0.0182	0.1702	1
Echinococcus granulosus	Zinc carboxypeptidase family protein	0.0124	0.1096	0.1493
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Schistosoma mansoni	lamin	0.0033	0.0141	0.0192
Loa Loa (eye worm)	zinc carboxypeptidase	0.0124	0.1096	0.1812
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Giardia lamblia	Nuclear ATP/GTP-binding protein	0.0124	0.1096	0.5
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Trypanosoma cruzi	metallo-peptidase, Clan MC, Family M14, putative	0.0124	0.1096	0.5
Plasmodium vivax	hypothetical protein, conserved	0.0124	0.1096	0.5
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Entamoeba histolytica	hypothetical protein	0.0043	0.0254	0.5
Loa Loa (eye worm)	intermediate filament protein	0.0033	0.0141	0.0233
Onchocerca volvulus	Subfamily M14A unassigned peptidase homolog	0.0724	0.7342	1
Brugia malayi	Calcitonin receptor-like protein seb-1	0.006	0.0429	0.2518
Echinococcus granulosus	lamin	0.0033	0.0141	0.0192
Schistosoma mansoni	family M14 non-peptidase homologue (M14 family)	0.0124	0.1096	0.1493
Echinococcus granulosus	Basic leucine zipper bZIP transcription	0.0043	0.0254	0.0346
Entamoeba histolytica	hypothetical protein	0.0043	0.0254	0.5
Onchocerca volvulus		0.0182	0.1702	0.2168
Brugia malayi	Zinc carboxypeptidase family protein	0.0124	0.1096	0.6439
Echinococcus multilocularis	Zinc carboxypeptidase family protein	0.0124	0.1096	0.1096
Echinococcus granulosus	cytosolic carboxypeptidase protein 5	0.0124	0.1096	0.1493
Brugia malayi	intermediate filament protein	0.0033	0.0141	0.0827
Schistosoma mansoni	carboxypeptidase N (M14 family)	0.0124	0.1096	0.1493
Onchocerca volvulus		0.0124	0.1096	0.1327
Brugia malayi	hypothetical protein	0.0043	0.0254	0.1493
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Trichomonas vaginalis	Clan MC, family M14, Zinc carboxypeptidase-like metallopeptidase	0.0124	0.1096	0.5
Schistosoma mansoni	hypothetical protein	0.0041	0.023	0.0314
Schistosoma mansoni	hypothetical protein	0.0124	0.1096	0.1493
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Brugia malayi	latrophilin 2 splice variant baaae	0.0041	0.023	0.1353
Toxoplasma gondii	zinc carboxypeptidase, putative	0.0124	0.1096	0.5
Trypanosoma brucei	metallo-peptidase, Clan MC, Family M14, putative	0.0124	0.1096	0.5
Echinococcus multilocularis	musashi	0.0033	0.0141	0.0141
Loa Loa (eye worm)	hypothetical protein	0.0124	0.1096	0.1812
Leishmania major	zinc carboxypeptidase, putative,metallo-peptidase, Clan MC, Family M14	0.0124	0.1096	0.5

Activities

Activity type	Activity value	Assay description	Source	Reference
Potency (functional)	= 0.3981 um	PUBCHEM_BIOASSAY: qHTS Assay for Modulators of Lamin A Splicing. (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	2.9093 uM	PUBCHEM_BIOASSAY: qHTS screen for small molecules that inhibit ELG1-dependent DNA repair in human embryonic kidney (HEK293T) cells expressing luciferase-tagged ELG1. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493107, AID493125]	ChEMBL.	No reference
Potency (functional)	5.6234 uM	PubChem BioAssay. qHTS of GLP-1 Receptor Inverse Agonists (Inhibition Mode). (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	10 uM	PUBCHEM_BIOASSAY: qHTS for Inhibitors of Vif-A3F Interactions: qHTS. (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	10.3225 uM	PUBCHEM_BIOASSAY: qHTS screen for small molecules that induce genotoxicity in human embryonic kidney (HEK293T) cells expressing luciferase-tagged ELG1. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493106, AID493143]	ChEMBL.	No reference
Potency (functional)	11.5821 uM	PUBCHEM_BIOASSAY: Nrf2 qHTS screen for inhibitors. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493153, AID493163, AID504648]	ChEMBL.	No reference
Potency (functional)	14.7157 uM	PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488745, AID488752, AID488774, AID504848, AID504850]	ChEMBL.	No reference
Potency (functional)	16.5113 uM	PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488752, AID488774, AID504848, AID504850]	ChEMBL.	No reference
Potency (functional)	= 19.9526 um	PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of HPGD (15-Hydroxyprostaglandin Dehydrogenase). (Class of assay: confirmatory) [Related pubchem assays: 2429 (Confirmation qHTS Assay for Inhibitors of HPGD (15-Hydroxyprostaglandin Dehydrogenase)), 2407 (Probe Development Summary for Inhibitors of HPGD (15-Hydroxyprostaglandin Dehydrogenase)), 2427 (Thermal Shift Assay for Inhibitors of HPGD (15-Hydroxyprostaglandin Dehydrogenase))]	ChEMBL.	No reference
Potency (functional)	22.3872 uM	PubChem BioAssay. qHTS of Nrf2 Activators. (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	= 25.1189 um	PUBCHEM_BIOASSAY: qHTS Fluorescence Polarization Assay for Inhibitors of MLL CXXC domain - DNA interaction. (Class of assay: confirmatory) [Related pubchem assays: 2698 (Summary assay.)]	ChEMBL.	No reference
Potency (functional)	28.1838 uM	PubChem BioAssay. qHTS for Antagonists of gsp, the Etiologic Mutation Responsible for Fibrous Dysplasia/McCune-Albright Syndrome: qHTS. (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	31.6228 uM	PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of JMJD2A-Tudor Domain. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504402]	ChEMBL.	No reference
Potency (functional)	= 39.8107 um	PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1). (Class of assay: confirmatory) [Related pubchem assays: 1030 (qHTS Validation Assay for Inhibitors of aldehyde dehydrogenase 1 (ALDH1A1))]	ChEMBL.	No reference
Potency (functional)	44.6684 uM	PubChem BioAssay. qHTS of PTHR Inhibitors: Primary Screen. (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (binding)	= 50.1187 um	PUBCHEM_BIOASSAY: qHTS Assay for Identification of Novel General Anesthetics. In this assay, a GABAergic mimetic model system, apoferritin and a profluorescent 1-aminoanthracene ligand (1-AMA), was used to construct a competitive binding assay for identification of novel general anesthetics (Class of assay: confirmatory) [Related pubchem assays: 2385 (Probe Development Summary for Identification of Novel General Anesthetics), 2323 (Validation apoferritin assay run on SigmaAldrich LOPAC1280 collection)]	ChEMBL.	No reference
Potency (functional)	70.7946 uM	PUBCHEM_BIOASSAY: Inhibitors of the vitamin D receptor (VDR): qHTS. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504855]	ChEMBL.	No reference
Potency (functional)	100 uM	PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Rango (Ran-regulated importin-beta cargo) - Importin beta complex formation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID540273]	ChEMBL.	No reference

Phenotypes

Whole-cell/tissue/organism interactions

Species name	Source	Reference	Is orphan
Plasmodium falciparum	ChEMBL23

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL1973003

Bibliographic References

No literature references available for this target.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 1614849