Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Mycobacterium tuberculosis | Probable lipase LipE | 0.0522 | 0.1537 | 0.1357 |
Brugia malayi | ribosomal protein S6 kinase alpha 3 | 0.0527 | 0.1551 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Echinococcus multilocularis | epidermal growth factor receptor | 0.0133 | 0.0368 | 0.203 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.0089 | 0.0236 | 0.13 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Loa Loa (eye worm) | hypothetical protein | 0.0522 | 0.1537 | 0.8473 |
Entamoeba histolytica | protein kinase, putative | 0.0092 | 0.0245 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0522 | 0.1537 | 0.8473 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | beta LACTamase domain containing family member | 0.0522 | 0.1537 | 0.8473 |
Mycobacterium tuberculosis | Probable conserved lipoprotein | 0.0522 | 0.1537 | 0.1357 |
Schistosoma mansoni | proto-oncogene tyrosine-protein kinase src | 0.0015 | 0.0012 | 0.0065 |
Schistosoma mansoni | tyrosine kinase | 0.0133 | 0.0368 | 0.203 |
Treponema pallidum | penicillin-binding protein (pbp-1) | 0.008 | 0.0209 | 0.5 |
Brugia malayi | Protein kinase domain containing protein | 0.0089 | 0.0236 | 0.1521 |
Loa Loa (eye worm) | hypothetical protein | 0.0522 | 0.1537 | 0.8473 |
Echinococcus granulosus | melanoma receptor tyrosine protein kinase | 0.0133 | 0.0368 | 0.203 |
Echinococcus granulosus | tyrosine protein kinase Lyn | 0.0017 | 0.0018 | 0.0097 |
Brugia malayi | Tyrosine-protein kinase abl-1 | 0.0015 | 0.0012 | 0.0076 |
Brugia malayi | beta-lactamase | 0.0522 | 0.1537 | 0.991 |
Schistosoma mansoni | tyrosine kinase | 0.013 | 0.0357 | 0.1965 |
Wolbachia endosymbiont of Brugia malayi | cell division protein FtsI | 0.008 | 0.0209 | 0.5 |
Loa Loa (eye worm) | beta-LACTamase domain containing family member | 0.0522 | 0.1537 | 0.8473 |
Echinococcus multilocularis | serine threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Echinococcus granulosus | protein kinase C gamma type | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | tyrosine protein kinase lyn tyrosine protein kinase blk | 0.0015 | 0.0012 | 0.0065 |
Echinococcus granulosus | protein kinase c iota type | 0.0089 | 0.0236 | 0.13 |
Schistosoma mansoni | tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Brugia malayi | Hr1 repeat family protein | 0.0089 | 0.0236 | 0.1521 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.053 | 0.156 | 1 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.0089 | 0.0236 | 0.13 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Loa Loa (eye worm) | hypothetical protein | 0.0522 | 0.1537 | 0.8473 |
Echinococcus multilocularis | proto oncogene tyrosine protein kinase LCK | 0.0015 | 0.0012 | 0.0065 |
Giardia lamblia | Kinase, AGC AKT | 0.0527 | 0.1551 | 0.5 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Schistosoma mansoni | tyrosine kinase | 0.013 | 0.0357 | 0.1965 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.0089 | 0.0236 | 0.13 |
Toxoplasma gondii | ABC1 family protein | 0.0522 | 0.1537 | 1 |
Trypanosoma brucei | hypothetical protein, conserved | 0.0522 | 0.1537 | 0.5169 |
Brugia malayi | Protein kinase domain containing protein | 0.0291 | 0.0843 | 0.5437 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.0089 | 0.0236 | 0.13 |
Trichomonas vaginalis | AGC family protein kinase | 0.0089 | 0.0236 | 0.0202 |
Loa Loa (eye worm) | TK/EGFR protein kinase | 0.0133 | 0.0368 | 0.203 |
Mycobacterium ulcerans | hypothetical protein | 0.0522 | 0.1537 | 0.2395 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0015 | 0.0012 | 0.0065 |
Treponema pallidum | penicillin-binding protein (pbp-3) | 0.008 | 0.0209 | 0.5 |
Plasmodium vivax | hypothetical protein, conserved | 0.0522 | 0.1537 | 0.5 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.0614 | 0.1814 | 1 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.0089 | 0.0236 | 0.13 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.0089 | 0.0236 | 0.13 |
Loa Loa (eye worm) | beta-lactamase | 0.0522 | 0.1537 | 0.8473 |
Echinococcus multilocularis | tyrosine protein kinase lyn lyn a protein tyrosine kinase lymphocyte specific protein tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Echinococcus multilocularis | c src tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.0089 | 0.0236 | 0.13 |
Schistosoma mansoni | tyrosine kinase | 0.0133 | 0.0368 | 0.203 |
Chlamydia trachomatis | transglycolase/transpeptidase | 0.008 | 0.0209 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0522 | 0.1537 | 0.8473 |
Loa Loa (eye worm) | hypothetical protein | 0.0158 | 0.0442 | 0.2437 |
Chlamydia trachomatis | transglycolase/transpeptidase | 0.008 | 0.0209 | 0.5 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | epidermal growth factor receptor | 0.0133 | 0.0368 | 0.203 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Trichomonas vaginalis | AGC family protein kinase | 0.0089 | 0.0236 | 0.0202 |
Echinococcus granulosus | insulin receptor | 0.0291 | 0.0843 | 0.4649 |
Mycobacterium ulcerans | esterase/lipase LipP | 0.0522 | 0.1537 | 0.2395 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0015 | 0.0012 | 0.0065 |
Echinococcus granulosus | c src tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium tuberculosis | Probable esterase LipL | 0.0522 | 0.1537 | 0.1357 |
Loa Loa (eye worm) | hypothetical protein | 0.0089 | 0.0236 | 0.13 |
Trichomonas vaginalis | AGC family protein kinase | 0.0089 | 0.0236 | 0.0202 |
Loa Loa (eye worm) | hypothetical protein | 0.0522 | 0.1537 | 0.8473 |
Brugia malayi | Protein kinase domain containing protein | 0.0089 | 0.0236 | 0.1521 |
Schistosoma mansoni | family S12 unassigned peptidase (S12 family) | 0.0522 | 0.1537 | 0.8473 |
Brugia malayi | Protein kinase domain containing protein | 0.0162 | 0.0454 | 0.2926 |
Schistosoma mansoni | tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Echinococcus multilocularis | 0.0038 | 0.0081 | 0.0446 | |
Mycobacterium tuberculosis | Conserved protein | 0.0522 | 0.1537 | 0.1357 |
Mycobacterium ulcerans | beta-lactamase | 0.0522 | 0.1537 | 0.2395 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | protein kinase c iota type | 0.0089 | 0.0236 | 0.13 |
Echinococcus granulosus | NDR protein kinase | 0.0089 | 0.0236 | 0.13 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0015 | 0.0012 | 0.0065 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | insulin receptor | 0.0291 | 0.0843 | 0.4649 |
Brugia malayi | Furin-like cysteine rich region family protein | 0.0133 | 0.0368 | 0.2374 |
Schistosoma mansoni | tyrosine kinase | 0.0133 | 0.0368 | 0.203 |
Entamoeba histolytica | protein kinase, putative | 0.0092 | 0.0245 | 1 |
Brugia malayi | beta-lactamase family protein | 0.0522 | 0.1537 | 0.991 |
Echinococcus granulosus | epidermal growth factor receptor | 0.0133 | 0.0368 | 0.203 |
Mycobacterium tuberculosis | Conserved protein | 0.0522 | 0.1537 | 0.1357 |
Brugia malayi | protein kinase C II. | 0.0089 | 0.0236 | 0.1521 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.0089 | 0.0236 | 0.13 |
Onchocerca volvulus | 0.0522 | 0.1537 | 0.5 | |
Treponema pallidum | penicillin-binding protein (pbp-2) | 0.008 | 0.0209 | 0.5 |
Trichomonas vaginalis | D-aminoacylase, putative | 0.0522 | 0.1537 | 1 |
Onchocerca volvulus | 0.0522 | 0.1537 | 0.5 | |
Schistosoma mansoni | tyrosine kinase | 0.0291 | 0.0843 | 0.4649 |
Mycobacterium tuberculosis | Probable hydrolase | 0.0522 | 0.1537 | 0.1357 |
Mycobacterium tuberculosis | Class a beta-lactamase BlaC | 0.1925 | 0.5755 | 0.5665 |
Echinococcus granulosus | proto oncogene tyrosine protein kinase LCK | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium tuberculosis | Probable esterase/lipase LipP | 0.0522 | 0.1537 | 0.1357 |
Trichomonas vaginalis | D-aminoacylase, putative | 0.0522 | 0.1537 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Abl | 0.0015 | 0.0012 | 0.0065 |
Echinococcus granulosus | 3'partial|tyrosine protein kinase Fgr | 0.0015 | 0.0012 | 0.0065 |
Brugia malayi | Hypothetical 52.5 kDa protein ZK945.1 in chromosome II, putative | 0.0522 | 0.1537 | 0.991 |
Trichomonas vaginalis | penicillin-binding protein, putative | 0.0522 | 0.1537 | 1 |
Schistosoma mansoni | tyrosine kinase | 0.0291 | 0.0843 | 0.4649 |
Brugia malayi | beta-lactamase family protein | 0.0522 | 0.1537 | 0.991 |
Echinococcus granulosus | insulin growth factor 1 receptor beta | 0.0291 | 0.0843 | 0.4649 |
Mycobacterium tuberculosis | Conserved protein | 0.0522 | 0.1537 | 0.1357 |
Echinococcus multilocularis | tyrosine protein kinase Btk29A | 0.0309 | 0.0895 | 0.4931 |
Echinococcus multilocularis | insulin growth factor 1 receptor beta | 0.0291 | 0.0843 | 0.4649 |
Loa Loa (eye worm) | TK/INSR protein kinase | 0.0291 | 0.0843 | 0.4649 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.0089 | 0.0236 | 0.13 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.0087 | 0.023 | 0.0158 |
Schistosoma mansoni | tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium ulcerans | lipoprotein LpqF | 0.0924 | 0.2745 | 0.4573 |
Echinococcus granulosus | protein kinase c epsilon type | 0.0089 | 0.0236 | 0.13 |
Schistosoma mansoni | serine/threonine kinase | 0.0089 | 0.0236 | 0.13 |
Schistosoma mansoni | atypical protein kinase C | 0.0089 | 0.0236 | 0.13 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.0089 | 0.0236 | 0.13 |
Echinococcus multilocularis | tyrosine protein kinase Fyn | 0.0015 | 0.0012 | 0.0065 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Trichomonas vaginalis | penicillin-binding protein, putative | 0.0522 | 0.1537 | 1 |
Echinococcus multilocularis | tyrosine protein kinase Src42A | 0.0015 | 0.0012 | 0.0065 |
Echinococcus granulosus | tyrosine protein kinase Fyn | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium leprae | Probable lipase LipE | 0.0522 | 0.1537 | 0.5237 |
Loa Loa (eye worm) | SRC-1 | 0.0015 | 0.0012 | 0.0065 |
Echinococcus granulosus | beta LACTamase domain containing family member | 0.0522 | 0.1537 | 0.8473 |
Onchocerca volvulus | 0.0522 | 0.1537 | 0.5 | |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.0614 | 0.1814 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Mycobacterium leprae | conserved hypothetical protein | 0.0522 | 0.1537 | 0.5237 |
Echinococcus granulosus | epidermal growth factor receptor | 0.0133 | 0.0368 | 0.203 |
Trichomonas vaginalis | esterase, putative | 0.0522 | 0.1537 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.0092 | 0.0245 | 0.1579 |
Schistosoma mansoni | tyrosine kinase | 0.0015 | 0.0012 | 0.0065 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0522 | 0.1537 | 0.5 |
Mycobacterium ulcerans | fusion of enoyl-CoA hydratase, EchA21 and lipase, LipE | 0.0522 | 0.1537 | 0.2395 |
Trichomonas vaginalis | D-aminoacylase, putative | 0.0522 | 0.1537 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.0092 | 0.0245 | 0.0271 |
Trypanosoma brucei | beta lactamase | 0.0924 | 0.2745 | 1 |
Schistosoma mansoni | tyrosine kinase | 0.013 | 0.0357 | 0.1965 |
Echinococcus granulosus | tyrosine protein kinase Src42A | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium tuberculosis | Probable lipase LipD | 0.0522 | 0.1537 | 0.1357 |
Echinococcus granulosus | tyrosine protein kinase Src64B | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium tuberculosis | Possible conserved lipoprotein LpqK | 0.0522 | 0.1537 | 0.1357 |
Schistosoma mansoni | tyrosine kinase | 0.0303 | 0.0878 | 0.4841 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.0089 | 0.0236 | 0.13 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.0092 | 0.0245 | 0.135 |
Mycobacterium tuberculosis | Probable conserved lipoprotein LpqF | 0.0924 | 0.2745 | 0.259 |
Mycobacterium ulcerans | lipase LipD | 0.0522 | 0.1537 | 0.2395 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0522 | 0.1537 | 0.5 |
Echinococcus multilocularis | tyrosine protein kinase Fgr | 0.0015 | 0.0012 | 0.0065 |
Schistosoma mansoni | family S12 unassigned peptidase (S12 family) | 0.0522 | 0.1537 | 0.8473 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.0614 | 0.1814 | 1 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.0089 | 0.0236 | 0.13 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.0089 | 0.0236 | 0.13 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.0089 | 0.0236 | 0.1521 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0089 | 0.0236 | 0.13 |
Brugia malayi | SRC-1 | 0.0015 | 0.0012 | 0.0076 |
Echinococcus granulosus | tyrosine protein kinase Btk29A | 0.0309 | 0.0895 | 0.4931 |
Echinococcus multilocularis | tyrosine protein kinase Src64B | 0.0015 | 0.0012 | 0.0065 |
Mycobacterium leprae | PROBABLE CONSERVED LIPOPROTEIN LPQF | 0.0924 | 0.2745 | 1 |
Mycobacterium ulcerans | class a beta-lactamase, BlaC | 0.1925 | 0.5755 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.0614 | 0.1814 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | = 4 ug ml-1 | Minimum inhibitory concentration against Propionibacterium acnes NCTC 737 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. aureus ATCC 2977 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against meticilline resistant S. aureus CJ 232 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against meticilline and rifampicin resistant S. aureus CJ 234 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against meticilline and fus resistant S. aureus CJ 234 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. aureus ATCC 6538P | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. aureus ATCC 29213 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. epidermidis ATCC 12228 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Corynebacterium xerosis NCTC 9755 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. faecium EI 119 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Streptococcus. species EF 6 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. pyogenes EC | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. thermophilus EG 5 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. zooepidermidis ED (gr.C) | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against S. salivarius EG 7 (gr.A) | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Clostridium perfringens KT 13 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Micrococcus luteus ATCC 9341 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Bacillus cereus ATCC 10876 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against E. coli HA 44 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Saccharomyces cerevisiae ZZ 7 | ChEMBL. | 11543681 |
MIC (functional) | > 125 ug ml-1 | Minimum inhibitory concentration against Candida albicans ATCC 10231 | ChEMBL. | 11543681 |
MIC (functional) | = 125 ug ml-1 | Minimum inhibitory concentration against Aspergillus niger ATCC 16404 | ChEMBL. | 11543681 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.