Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Schistosoma mansoni | smdr2 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Echinococcus granulosus | ubiquitin conjugating enzyme E2 N | 0.0042 | 0.5414 | 0.5414 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Echinococcus granulosus | multidrug resistance associated protein 1 | 0.0034 | 0.347 | 0.347 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Leishmania major | p-glycoprotein | 0.0059 | 1 | 1 |
Mycobacterium ulcerans | drugs-transport transmembrane ATP-binding protein ABC transporter | 0.0021 | 0.019 | 0.5 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0034 | 0.347 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0034 | 0.347 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | taga, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0039 | 0.4732 | 0.4732 |
Echinococcus multilocularis | multidrug resistance associated protein 1 | 0.0034 | 0.347 | 0.3343 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Trypanosoma brucei | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Plasmodium falciparum | ubiquitin-conjugating enzyme E2 N, putative | 0.0042 | 0.5414 | 0.5325 |
Toxoplasma gondii | ubiquitin-conjugating enzyme subfamily protein | 0.0042 | 0.5414 | 0.5325 |
Entamoeba histolytica | ABC transporter, putative | 0.0034 | 0.347 | 0.347 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Mycobacterium tuberculosis | Probable transmembrane multidrug efflux pump | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Leishmania major | ATP-binding cassette protein subfamily C, member 6, putative | 0.0034 | 0.347 | 0.3343 |
Loa Loa (eye worm) | hypothetical protein | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0034 | 0.347 | 0.347 |
Entamoeba histolytica | P-glycoprotein 5, putative | 0.0059 | 1 | 1 |
Entamoeba histolytica | P-glycoprotein 6, putative | 0.0021 | 0.019 | 0.019 |
Chlamydia trachomatis | ABC transporter ATP binding protein/permease | 0.0059 | 1 | 0.5 |
Mycobacterium leprae | PROBABLE DRUGS-TRANSPORT TRANSMEMBRANE ATP-BINDING PROTEIN ABC TRANSPORTER | 0.0021 | 0.019 | 0.5 |
Echinococcus granulosus | 5'partial|ATP binding cassette sub family B | 0.0059 | 0.981 | 0.981 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Leishmania major | ATP-binding cassette protein subfamily C, member 2, putative | 0.0034 | 0.347 | 0.3343 |
Echinococcus multilocularis | ubiquitin conjugating enzyme E2 N | 0.0042 | 0.5414 | 0.5325 |
Entamoeba histolytica | P-glycoprotein-2, putative | 0.0059 | 1 | 1 |
Brugia malayi | ABC transporter family protein | 0.0059 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | abcb9, putative | 0.0059 | 1 | 1 |
Schistosoma mansoni | ubiquitin conjugating enzyme 13 | 0.0042 | 0.5414 | 0.5414 |
Brugia malayi | multidrug resistance related protein 1 | 0.0034 | 0.347 | 0.347 |
Entamoeba histolytica | multidrug resistance protein, putative | 0.0034 | 0.347 | 0.347 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Leishmania major | ubiquitin-conjugating enzyme e2, putative | 0.0042 | 0.5414 | 0.5325 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0034 | 0.347 | 0.3343 |
Brugia malayi | ABC transporter transmembrane region family protein | 0.0034 | 0.347 | 0.347 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Loa Loa (eye worm) | multidrug resistance protein 3 | 0.0059 | 1 | 1 |
Entamoeba histolytica | P-glycoprotein 6, putative | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Leishmania major | ATP-binding cassette protein subfamily C, member 5, putative | 0.0034 | 0.347 | 0.3343 |
Brugia malayi | P-glycoprotein-like protein | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | ABC transporter | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Brugia malayi | Ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 1 |
Entamoeba histolytica | P-glycoprotein-1 | 0.0059 | 1 | 1 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Trypanosoma brucei | ubiquitin-protein ligase, putative | 0.0042 | 0.5414 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0039 | 0.4732 | 0.4732 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Brugia malayi | ABC transporter transmembrane region family protein | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Brugia malayi | hypothetical protein | 0.0021 | 0.019 | 0.019 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Trypanosoma brucei | multidrug resistance protein E | 0.0034 | 0.347 | 0.6278 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | multidrug resistance associated protein 7 | 0.0034 | 0.347 | 0.347 |
Leishmania major | ATP-binding cassette protein subfamily C, member 1, putative | 0.0034 | 0.347 | 0.3343 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0059 | 1 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0059 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0039 | 0.4732 | 0.463 |
Giardia lamblia | ABC transporter, putative | 0.0034 | 0.347 | 1 |
Leishmania major | pentamidine resistance protein 1 | 0.0034 | 0.347 | 0.3343 |
Schistosoma mansoni | smdr1 | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | multidrug resistance protein E, putative | 0.0034 | 0.347 | 0.6278 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trypanosoma brucei | trans-sialidase | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0039 | 0.4732 | 0.4732 |
Loa Loa (eye worm) | hypothetical protein | 0.0033 | 0.3279 | 0.3279 |
Plasmodium vivax | ubiquitin-conjugating enzyme E2 N, putative | 0.0042 | 0.5414 | 0.5325 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Trypanosoma brucei | p-glycoprotein | 0.0034 | 0.347 | 0.6278 |
Entamoeba histolytica | ubiquitin-conjugating enzyme family protein | 0.0042 | 0.5414 | 0.5414 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 0.5414 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Plasmodium vivax | multidrug resistance protein 1, putative | 0.0059 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0059 | 1 | 1 |
Mycobacterium ulcerans | transmembrane ABC transporter ATP-binding protein | 0.0021 | 0.019 | 0.5 |
Brugia malayi | ABC transporter family protein | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Mycobacterium ulcerans | transmembrane ABC transporter ATP-binding protein | 0.0021 | 0.019 | 0.5 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | ABC-type protease secretion system, ATPase and permease component, AprD | 0.0021 | 0.019 | 0.5 |
Toxoplasma gondii | ATP-binding cassette transporter ABC.B1 | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0034 | 0.347 | 0.347 |
Onchocerca volvulus | 0.0059 | 1 | 0.5 | |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Schistosoma mansoni | multidrug resistance protein | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Schistosoma mansoni | multidrug resistance protein | 0.0059 | 1 | 1 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0033 | 0.3279 | 0.9452 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Brugia malayi | multidrug Resistance Protein family member (mrp-5), putative | 0.0021 | 0.019 | 0.019 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 0.5414 |
Schistosoma mansoni | multidrug resistance protein | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | ABC transporter | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Leishmania major | ABC-thiol transporter | 0.0034 | 0.347 | 0.3343 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Echinococcus multilocularis | multidrug resistance associated protein 7 | 0.0034 | 0.347 | 0.3343 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0059 | 0.981 | 0.981 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Schistosoma mansoni | ATP-binding cassette sub-family B member 7 mitochondrial precursor (abc7) | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Plasmodium falciparum | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0059 | 1 | 1 |
Brugia malayi | ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Leishmania major | p-glycoprotein e | 0.0034 | 0.347 | 0.3343 |
Echinococcus granulosus | ATP binding cassette sub family B | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0034 | 0.347 | 0.347 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | abcb9, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | ATP-binding cassette sub-family B member 2 | 0.0059 | 1 | 1 |
Brugia malayi | ABC transporter family protein | 0.0021 | 0.019 | 0.019 |
Giardia lamblia | MRP-like ABC transporter | 0.0034 | 0.347 | 1 |
Echinococcus granulosus | ATP binding cassette sub family B | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | abcb9, putative | 0.0059 | 1 | 1 |
Entamoeba histolytica | P-glyco protein 6, putative | 0.0059 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | ABC-type multidrug transport system, ATPase and permease component | 0.0021 | 0.019 | 0.5 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 1 |
Loa Loa (eye worm) | ABC transporter transmembrane region family protein | 0.0034 | 0.347 | 0.347 |
Entamoeba histolytica | P-glycoprotein-5 | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0021 | 0.019 | 0.019 |
Mycobacterium ulcerans | component linked with the assembly of cytochrome transport transmembrane ATP-binding protein ABC transporter CydD | 0.0021 | 0.019 | 0.5 |
Brugia malayi | ABC transporter | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | ABC transporter | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0059 | 1 | 1 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Leishmania major | ATP-binding cassette protein subfamily B, member 2, putative | 0.0059 | 1 | 1 |
Mycobacterium leprae | PROBABLE DRUGS-TRANSPORT TRANSMEMBRANE ATP-BINDING PROTEIN ABC TRANSPORTER | 0.0021 | 0.019 | 0.5 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette sub family B | 0.0059 | 0.981 | 0.9806 |
Mycobacterium ulcerans | transmembrane ABC transporter ATP-binding protein | 0.0021 | 0.019 | 0.5 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Brugia malayi | ABC transporter family protein | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Trypanosoma brucei | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (functional) | = 44 % | Percent inhibition against ethanol-induced gastric lesions in male albino rat was determined at a dose of 25 mg/Kg | ChEMBL. | 2296028 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.