Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0285 | 0.1737 | 0.1737 |
Loa Loa (eye worm) | hypothetical protein | 0.0271 | 0.1251 | 0.1251 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0534 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Brugia malayi | tubulin alpha chain - mouse | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0534 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Schistosoma mansoni | tubulin subunit beta | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0271 | 0.1251 | 0.1251 |
Schistosoma mansoni | tubulin subunit alpha | 0.0395 | 0.5376 | 0.4404 |
Entamoeba histolytica | tubulin family protein | 0.0534 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit beta | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0395 | 0.5376 | 0.5376 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0534 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0395 | 0.5376 | 0.5376 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0395 | 0.5376 | 0.5376 |
Giardia lamblia | Beta tubulin | 0.0534 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0285 | 0.1737 | 0.1737 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0271 | 0.1251 | 0.1251 |
Plasmodium vivax | tubulin beta chain, putative | 0.0534 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Entamoeba histolytica | tubulin family protein | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0395 | 0.5376 | 0.5376 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0395 | 0.5376 | 0.4404 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0395 | 0.5376 | 0.5376 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0285 | 0.1737 | 0.1737 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin subunit TubB | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0395 | 0.5376 | 0.4404 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0395 | 0.5376 | 0.5376 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0534 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0534 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Loa Loa (eye worm) | tubulin beta chain | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0534 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0534 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0534 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0534 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0395 | 0.5376 | 0.4404 |
Schistosoma mansoni | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | beta tubulin | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0395 | 0.5376 | 0.4404 |
Schistosoma mansoni | tubulin subunit beta | 0.0534 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0534 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0534 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0395 | 0.5376 | 0.5376 |
Echinococcus multilocularis | beta tubulin | 0.0534 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Trypanosoma cruzi | beta tubulin, putative | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0534 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0395 | 0.5376 | 0.4404 |
Trypanosoma brucei | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0271 | 0.1251 | 0.1251 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0285 | 0.1737 | 0.1737 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0534 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0395 | 0.5376 | 0.4404 |
Loa Loa (eye worm) | alpha-tubulin | 0.0395 | 0.5376 | 0.5376 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0395 | 0.5376 | 0.4404 |
Brugia malayi | beta-tubulin, identical | 0.0534 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0395 | 0.5376 | 0.5376 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0395 | 0.5376 | 0.5376 |
Echinococcus multilocularis | beta tubulin | 0.0534 | 1 | 1 |
Toxoplasma gondii | beta-tubulin, putative | 0.0534 | 1 | 1 |
Brugia malayi | tubulin alpha-2 chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0395 | 0.5376 | 0.4404 |
Loa Loa (eye worm) | beta-tubulin | 0.0534 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0534 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0395 | 0.5376 | 0.4404 |
Brugia malayi | Tubulin alpha-2 chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0534 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | beta tubulin | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0395 | 0.5376 | 0.5376 |
Echinococcus granulosus | tubulin subunit beta | 0.0534 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0395 | 0.5376 | 0.4404 |
Loa Loa (eye worm) | alpha-tubulin | 0.0395 | 0.5376 | 0.5376 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Brugia malayi | Tubulin alpha-2 chain | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Trypanosoma brucei | beta tubulin | 0.0534 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0395 | 0.5376 | 0.5376 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0395 | 0.5376 | 0.4404 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0395 | 0.5376 | 0.4404 |
Giardia lamblia | Beta tubulin | 0.0534 | 1 | 1 |
Echinococcus granulosus | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0395 | 0.5376 | 0.4404 |
Schistosoma mansoni | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin alpha chain | 0.0395 | 0.5376 | 0.4404 |
Trypanosoma brucei | beta tubulin | 0.0534 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0534 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0395 | 0.5376 | 0.4404 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0271 | 0.1251 | 0.1251 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0395 | 0.5376 | 0.5376 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0395 | 0.5376 | 0.4404 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0395 | 0.5376 | 0.5376 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0534 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0395 | 0.5376 | 0.4404 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0395 | 0.5376 | 0.4404 |
Leishmania major | alpha tubulin | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0395 | 0.5376 | 0.4404 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0395 | 0.5376 | 0.4404 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0534 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0534 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0395 | 0.5376 | 0.4404 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
MIC (functional) | > 100 ug ml-1 | Antimicrobial activity against Escherichia coli ATCC 25922-1 by threefold dilution agar inclusion method | ChEMBL. | 833822 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.