Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Toxoplasma gondii | beta-1 tubulin, putative | 0.0231 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.012 | 0.1296 | 0.1296 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0231 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Brugia malayi | tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.012 | 0.1296 | 0.1296 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Plasmodium vivax | tubulin beta chain, putative | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0175 | 0.5571 | 0.4682 |
Giardia lamblia | Beta tubulin | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0125 | 0.1672 | 0.1672 |
Toxoplasma gondii | beta-tubulin, putative | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0125 | 0.1672 | 0.1672 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0175 | 0.5571 | 0.5571 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0175 | 0.5571 | 0.5571 |
Entamoeba histolytica | tubulin family protein | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.012 | 0.1296 | 0.1296 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0125 | 0.1672 | 0.1672 |
Echinococcus multilocularis | hypothetical protein | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin subunit TubB | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.012 | 0.1296 | 0.1296 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin beta chain | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0231 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | beta-tubulin | 0.0231 | 1 | 1 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0231 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Toxoplasma gondii | beta tubulin | 0.0231 | 1 | 1 |
Brugia malayi | beta-tubulin, identical | 0.0231 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | beta tubulin | 0.0231 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | hypothetical protein | 0.0175 | 0.5571 | 0.5571 |
Echinococcus multilocularis | beta tubulin | 0.0231 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0231 | 1 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.012 | 0.1296 | 0.1296 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit alpha | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0231 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma cruzi | beta tubulin, putative | 0.0231 | 1 | 1 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0231 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0175 | 0.5571 | 0.5571 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0175 | 0.5571 | 0.4682 |
Schistosoma mansoni | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | beta tubulin | 0.0231 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0175 | 0.5571 | 0.4682 |
Trichomonas vaginalis | tubulin, putative | 0.0231 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | beta tubulin | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0175 | 0.5571 | 0.4682 |
Plasmodium falciparum | alpha tubulin 2 | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | BEN-1 protein | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin subunit beta | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Echinococcus granulosus | tubulin subunit beta | 0.0231 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0231 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0175 | 0.5571 | 0.5571 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0175 | 0.5571 | 0.5571 |
Loa Loa (eye worm) | alpha-tubulin | 0.0175 | 0.5571 | 0.5571 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0231 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0175 | 0.5571 | 0.4682 |
Brugia malayi | Tubulin alpha-2 chain | 0.0175 | 0.5571 | 0.4682 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0231 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0125 | 0.1672 | 0.1672 |
Schistosoma mansoni | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Leishmania major | alpha tubulin | 0.0175 | 0.5571 | 0.4682 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | 0 uM | In vitro inhibitory concentration of the compound against growth of mouse sarcoma 180 (S-180) cells; Inactive | ChEMBL. | 9046342 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.