Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0136 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Echinococcus multilocularis | beta tubulin | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0099 | 0.5243 | 0.5243 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0099 | 0.5243 | 0.5243 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0099 | 0.5243 | 0.5243 |
Trypanosoma brucei | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Toxoplasma gondii | beta-tubulin, putative | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0136 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0136 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0136 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | tubulin subunit beta | 0.0136 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0099 | 0.5243 | 0.5243 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0068 | 0.122 | 0.122 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Plasmodium falciparum | tubulin beta chain | 0.0136 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0099 | 0.5243 | 0.5243 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0099 | 0.5243 | 0.5243 |
Echinococcus multilocularis | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0068 | 0.122 | 0.122 |
Trypanosoma brucei | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus granulosus | tubulin subunit TubB | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0136 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0099 | 0.5243 | 0.4212 |
Toxoplasma gondii | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0099 | 0.5243 | 0.4212 |
Brugia malayi | alpha-tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | tubulin subunit beta | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0099 | 0.5243 | 0.5243 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0099 | 0.5243 | 0.4212 |
Echinococcus multilocularis | hypothetical protein | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | BEN-1 protein | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0068 | 0.122 | 0.122 |
Echinococcus granulosus | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0099 | 0.5243 | 0.5243 |
Trichomonas vaginalis | tubulin, putative | 0.0136 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | tubulin subunit beta | 0.0136 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0136 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0099 | 0.5243 | 0.4212 |
Plasmodium falciparum | alpha tubulin 1 | 0.0099 | 0.5243 | 0.4212 |
Echinococcus multilocularis | tubulin subunit beta | 0.0136 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0099 | 0.5243 | 0.5243 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0136 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0136 | 1 | 1 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0099 | 0.5243 | 0.4212 |
Giardia lamblia | Alpha-tubulin | 0.0099 | 0.5243 | 0.4212 |
Trypanosoma brucei | beta tubulin | 0.0136 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | tubulin subunit alpha | 0.0099 | 0.5243 | 0.4212 |
Brugia malayi | Tubulin alpha-2 chain | 0.0099 | 0.5243 | 0.4212 |
Trypanosoma brucei | beta tubulin | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0099 | 0.5243 | 0.5243 |
Loa Loa (eye worm) | beta-tubulin | 0.0136 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0136 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0136 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0136 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | tubulin beta chain | 0.0136 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0099 | 0.5243 | 0.5243 |
Schistosoma mansoni | tubulin subunit beta | 0.0136 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0099 | 0.5243 | 0.5243 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0099 | 0.5243 | 0.4212 |
Trypanosoma brucei | beta tubulin | 0.0136 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Loa Loa (eye worm) | hypothetical protein | 0.0099 | 0.5243 | 0.5243 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0136 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0068 | 0.122 | 0.122 |
Loa Loa (eye worm) | alpha-tubulin | 0.0099 | 0.5243 | 0.5243 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | beta tubulin | 0.0136 | 1 | 1 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | tubulin subunit alpha | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0072 | 0.1782 | 0.1782 |
Echinococcus granulosus | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus granulosus | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0099 | 0.5243 | 0.4212 |
Schistosoma mansoni | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Brugia malayi | tubulin alpha chain - mouse | 0.0099 | 0.5243 | 0.4212 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0136 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0099 | 0.5243 | 0.4212 |
Giardia lamblia | Beta tubulin | 0.0136 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0136 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Brugia malayi | beta-tubulin, identical | 0.0136 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0072 | 0.1782 | 0.1782 |
Trypanosoma brucei | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Brugia malayi | tubulin alpha-2 chain | 0.0099 | 0.5243 | 0.4212 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0072 | 0.1782 | 0.1782 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0068 | 0.122 | 0.122 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0099 | 0.5243 | 0.5243 |
Trypanosoma brucei | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0099 | 0.5243 | 0.4212 |
Entamoeba histolytica | tubulin family protein | 0.0136 | 1 | 1 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0099 | 0.5243 | 0.4212 |
Brugia malayi | Tubulin alpha-2 chain | 0.0099 | 0.5243 | 0.4212 |
Giardia lamblia | Beta tubulin | 0.0136 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0099 | 0.5243 | 0.4212 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0136 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0136 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Leishmania major | beta tubulin | 0.0136 | 1 | 1 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0072 | 0.1782 | 0.1782 |
Leishmania major | alpha tubulin | 0.0099 | 0.5243 | 0.4212 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0136 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0136 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0099 | 0.5243 | 0.4212 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (binding) | = 0 % | Inhibition of ovine COX1 at 100 uM | ChEMBL. | 17079150 |
Inhibition (binding) | = 0 % | Inhibition of ovine COX1 at 100 uM | ChEMBL. | 17079150 |
Inhibition (binding) | = 19 % | Inhibition of ovine COX2 at 100 uM | ChEMBL. | 17079150 |
Inhibition (binding) | = 19 % | Inhibition of ovine COX2 at 100 uM | ChEMBL. | 17079150 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.