Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Schistosoma mansoni | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | tubulin alpha chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0426 | 0.3982 | 0.3982 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Brugia malayi | Tubulin gamma chain | 0.0426 | 0.3982 | 0.3982 |
Loa Loa (eye worm) | alpha-tubulin | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0705 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-3 chain | 0.0464 | 0.4811 | 0.4342 |
Plasmodium falciparum | alpha tubulin 2 | 0.0705 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.052 | 0.6018 | 0.5658 |
Toxoplasma gondii | beta-tubulin, putative | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin alpha chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Giardia lamblia | Beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin alpha chain | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0705 | 1 | 1 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0583 | 0.7372 | 0.7372 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Loa Loa (eye worm) | hypothetical protein | 0.052 | 0.6018 | 0.5658 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0705 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0705 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0426 | 0.3982 | 0.3982 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0583 | 0.7372 | 0.7372 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0705 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0705 | 1 | 1 |
Onchocerca volvulus | 0.0241 | 0 | 0.5 | |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | alpha-tubulin | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0583 | 0.7372 | 0.5633 |
Schistosoma mansoni | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0705 | 1 | 1 |
Echinococcus multilocularis | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0705 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0583 | 0.7372 | 0.5633 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0705 | 1 | 1 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0705 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0426 | 0.3982 | 0.3982 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0583 | 0.7372 | 0.7372 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin alpha chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0426 | 0.3982 | 0.3982 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0464 | 0.4811 | 0.4811 |
Echinococcus granulosus | tubulin alpha chain | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0705 | 1 | 1 |
Toxoplasma gondii | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0705 | 1 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0705 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0583 | 0.7372 | 0.7372 |
Trypanosoma brucei | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0583 | 0.7372 | 0.7372 |
Brugia malayi | Tubulin alpha-2 chain | 0.0705 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0705 | 1 | 1 |
Echinococcus granulosus | alpha tubulin | 0.0705 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0426 | 0.3982 | 0.3982 |
Brugia malayi | beta-tubulin, identical | 0.0583 | 0.7372 | 0.7372 |
Trypanosoma cruzi | beta tubulin, putative | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | tubulin subunit TubB | 0.0705 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Loa Loa (eye worm) | beta-tubulin | 0.0583 | 0.7372 | 0.7134 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0705 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0705 | 1 | 1 |
Brugia malayi | Tubulin alpha-2 chain | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.052 | 0.6018 | 0.5658 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.052 | 0.6018 | 0.6018 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0426 | 0.3982 | 0.3439 |
Giardia lamblia | Beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0705 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0583 | 0.7372 | 0.7372 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0583 | 0.7372 | 0.7134 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0705 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0705 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0705 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0705 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0583 | 0.7372 | 0.7372 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0583 | 0.7372 | 0.5633 |
Plasmodium falciparum | tubulin beta chain | 0.0583 | 0.7372 | 0.5633 |
Plasmodium vivax | tubulin beta chain, putative | 0.0583 | 0.7372 | 0.5633 |
Brugia malayi | Tubulin beta-1 chain | 0.0583 | 0.7372 | 0.7372 |
Loa Loa (eye worm) | BEN-1 protein | 0.0583 | 0.7372 | 0.7134 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Trypanosoma brucei | beta tubulin | 0.0583 | 0.7372 | 0.7372 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | tubulin gamma chain | 0.0426 | 0.3982 | 0.3982 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.052 | 0.6018 | 0.5658 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Loa Loa (eye worm) | BEN-1 protein | 0.0583 | 0.7372 | 0.7134 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0583 | 0.7372 | 0.5633 |
Plasmodium falciparum | alpha tubulin 1 | 0.0705 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Brugia malayi | tubulin alpha chain - mouse | 0.0705 | 1 | 1 |
Echinococcus multilocularis | hypothetical protein | 0.0705 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Brugia malayi | alpha-tubulin | 0.0705 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0583 | 0.7372 | 0.7134 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0426 | 0.3982 | 0.3982 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0705 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Loa Loa (eye worm) | hypothetical protein | 0.0464 | 0.4811 | 0.4342 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Entamoeba histolytica | tubulin family protein | 0.0583 | 0.7372 | 0.5633 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Schistosoma mansoni | tubulin subunit alpha | 0.0705 | 1 | 1 |
Entamoeba histolytica | tubulin family protein | 0.0583 | 0.7372 | 0.5633 |
Schistosoma mansoni | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0705 | 1 | 1 |
Trypanosoma brucei | beta tubulin | 0.0583 | 0.7372 | 0.7372 |
Schistosoma mansoni | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Echinococcus multilocularis | tubulin alpha chain | 0.0705 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0426 | 0.3982 | 0.3982 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0583 | 0.7372 | 0.7134 |
Echinococcus granulosus | tubulin subunit beta | 0.0583 | 0.7372 | 0.5633 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0583 | 0.7372 | 0.5633 |
Trichomonas vaginalis | tubulin, putative | 0.0583 | 0.7372 | 0.7372 |
Giardia lamblia | Alpha-tubulin | 0.0705 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0705 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0583 | 0.7372 | 0.7134 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0583 | 0.7372 | 0.5633 |
Leishmania major | alpha tubulin | 0.0705 | 1 | 1 |
Leishmania major | beta tubulin | 0.0583 | 0.7372 | 0.5633 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
ED50 (functional) | 0 mg kg-1 | Antiallergic activity by rat passive cutaneous anaphylaxis (PCA) assay when administered iv; ND means no data | ChEMBL. | 6876084 |
ED50 (functional) | > 10 mg kg-1 | Antiallergic activity by rat passive cutaneous anaphylaxis (PCA) assay when administered per orally | ChEMBL. | 6876084 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.