Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Echinococcus granulosus | Glutaredoxin protein 5 | 0.4304 | 0.6296 | 0.9473 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.023 | 0.0074 | 0.0111 |
Toxoplasma gondii | protein kinase domain-containing protein | 0.023 | 0.0074 | 0.0076 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.023 | 0.0074 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative,serine/threonine protein kinase, putative | 0.023 | 0.0074 | 1 |
Onchocerca volvulus | Putative zinc finger protein | 0.0181 | 0 | 0.5 |
Trypanosoma cruzi | serine/threonine-protein kinase NRKB, putative | 0.023 | 0.0074 | 0.0111 |
Echinococcus granulosus | nervana 2 | 0.4304 | 0.6296 | 0.9473 |
Loa Loa (eye worm) | AGC/RSK/P70 protein kinase | 0.6547 | 0.9723 | 0.9723 |
Loa Loa (eye worm) | AGC/AKT protein kinase | 0.6728 | 1 | 1 |
Brugia malayi | Protein kinase domain containing protein | 0.2244 | 0.315 | 0.315 |
Plasmodium falciparum | RAC-beta serine/threonine protein kinase | 0.4352 | 0.637 | 1 |
Leishmania major | folate/biopterin transporter, putative | 0.023 | 0.0074 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/PKN protein kinase | 0.2244 | 0.315 | 0.315 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Entamoeba histolytica | hypothetical protein | 0.023 | 0.0074 | 0.0074 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.023 | 0.0074 | 0.0111 |
Echinococcus multilocularis | serine threonine protein kinase nrc serine threonine protein kinase gad | 0.4352 | 0.637 | 0.9584 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Echinococcus granulosus | serine:threonine protein kinase N2 | 0.2244 | 0.315 | 0.4739 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Echinococcus granulosus | serine threonine protein kinase nrc | 0.4352 | 0.637 | 0.9584 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Echinococcus granulosus | protein kinase c epsilon type | 0.2244 | 0.315 | 0.4739 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Entamoeba histolytica | protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Brugia malayi | protein kinase C II. | 0.2244 | 0.315 | 0.315 |
Echinococcus multilocularis | serine:threonine protein kinase 38 | 0.2244 | 0.315 | 0.4739 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Entamoeba histolytica | protein kinase, putative | 0.6728 | 1 | 1 |
Entamoeba histolytica | hypothetical protein | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.2244 | 0.315 | 0.315 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.2425 | 0.3427 | 0.3427 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative | 0.023 | 0.0074 | 1 |
Echinococcus multilocularis | nervana 2 | 0.4304 | 0.6296 | 0.9473 |
Entamoeba histolytica | protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Leishmania major | protein kinase, putative | 0.023 | 0.0074 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.4533 | 0.6647 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Echinococcus multilocularis | protein kinase c epsilon type | 0.2244 | 0.315 | 0.4739 |
Plasmodium vivax | calcium-dependent protein kinase 7, putative | 0.023 | 0.0074 | 0.0116 |
Trypanosoma brucei | serine/threonine-protein kinase NrkA | 0.023 | 0.0074 | 0.0074 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.2244 | 0.315 | 0.4739 |
Echinococcus granulosus | Ribosomal protein S6 kinase beta 2 | 0.2244 | 0.315 | 0.4739 |
Brugia malayi | Protein kinase domain containing protein | 0.2244 | 0.315 | 0.315 |
Toxoplasma gondii | AGC kinase | 0.6547 | 0.9723 | 1 |
Echinococcus granulosus | protein kinase C gamma type | 0.2244 | 0.315 | 0.4739 |
Echinococcus multilocularis | Ribosomal protein S6 kinase beta 2 | 0.2244 | 0.315 | 0.4739 |
Echinococcus granulosus | ribosomal protein s6 kinase beta 1 | 0.2244 | 0.315 | 0.4739 |
Echinococcus multilocularis | ribosomal protein S6 kinase alpha 3 | 0.2244 | 0.315 | 0.4739 |
Trypanosoma cruzi | NIMA-related kinase, putative | 0.023 | 0.0074 | 0.0111 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/DMPK/GEK protein kinase | 0.2244 | 0.315 | 0.315 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Echinococcus multilocularis | Glutaredoxin protein 5 | 0.4304 | 0.6296 | 0.9473 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Entamoeba histolytica | protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Echinococcus granulosus | protein kinase c iota type | 0.2244 | 0.315 | 0.4739 |
Schistosoma mansoni | serine/threonine kinase | 0.2244 | 0.315 | 0.4739 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.4352 | 0.637 | 0.9584 |
Entamoeba histolytica | protein kinase, putative | 0.2244 | 0.315 | 0.315 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.023 | 0.0074 | 0.0111 |
Echinococcus multilocularis | nervana 2 | 0.4304 | 0.6296 | 0.9473 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.2244 | 0.315 | 0.315 |
Onchocerca volvulus | 0.0181 | 0 | 0.5 | |
Onchocerca volvulus | outspread protein homolog | 0.0181 | 0 | 0.5 |
Echinococcus granulosus | nervana 2 | 0.4304 | 0.6296 | 0.9473 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Echinococcus granulosus | calcium:calmodulin dependent protein kinase | 0.4352 | 0.637 | 0.9584 |
Trypanosoma brucei | serine/threonine-protein kinase NRKB, putative | 0.023 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/MSK protein kinase | 0.2244 | 0.315 | 0.315 |
Echinococcus multilocularis | serine:threonine protein kinase N2 | 0.2244 | 0.315 | 0.4739 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.4533 | 0.6647 | 0.6647 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Echinococcus multilocularis | ribosomal protein s6 kinase beta 1 | 0.2244 | 0.315 | 0.4739 |
Leishmania major | serine/threonine-protein kinase a, putative | 0.023 | 0.0074 | 1 |
Trypanosoma cruzi | Protein kinase B | 0.4533 | 0.6647 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Giardia lamblia | Kinase, AGC PKA | 0.4352 | 0.637 | 0.5 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK21, putative | 0.023 | 0.0074 | 0.0111 |
Echinococcus granulosus | Protein kinase C brain isozyme | 0.2244 | 0.315 | 0.4739 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Trichomonas vaginalis | ribosomal protein S6 kinase, 90kD, polypeptide, putative | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Echinococcus granulosus | NDR protein kinase | 0.2244 | 0.315 | 0.4739 |
Echinococcus multilocularis | Protein kinase C, brain isozyme | 0.2244 | 0.315 | 0.4739 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | 3-phosphoinositide dependent protein kinase-1, putative | 0.023 | 0.0074 | 0.0074 |
Trypanosoma brucei | NEK family Serine/threonine-protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | hypothetical protein | 0.2244 | 0.315 | 0.315 |
Echinococcus multilocularis | protein kinase c iota type | 0.2244 | 0.315 | 0.4739 |
Trypanosoma cruzi | Serine/threonine-protein kinase NEK17, putative | 0.023 | 0.0074 | 0.0111 |
Echinococcus multilocularis | serine threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Entamoeba histolytica | PH domain containing protein kinase, putative | 0.4533 | 0.6647 | 0.6647 |
Entamoeba histolytica | p21-activated kinase | 0.023 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/RSK/RSK protein kinase | 0.2244 | 0.315 | 0.315 |
Trypanosoma brucei | protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Trypanosoma brucei | rac serine-threonine kinase, putative | 0.6728 | 1 | 1 |
Schistosoma mansoni | serine/threonine-protein kinase | 0.4533 | 0.6647 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trypanosoma cruzi | rac serine-threonine kinase, putative | 0.4533 | 0.6647 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Plasmodium vivax | rac-beta serine/threonine protein kinase, putative | 0.4352 | 0.637 | 1 |
Entamoeba histolytica | protein kinase, putative | 0.6547 | 0.9723 | 0.9723 |
Schistosoma mansoni | atypical protein kinase C | 0.2244 | 0.315 | 0.4739 |
Onchocerca volvulus | Protein melted homolog | 0.0181 | 0 | 0.5 |
Entamoeba histolytica | protein kinase, putative | 0.6728 | 1 | 1 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Trichomonas vaginalis | serine/threonine-protein kinase sgk, putative | 0.2195 | 0.3076 | 0.3076 |
Brugia malayi | Hr1 repeat family protein | 0.2244 | 0.315 | 0.315 |
Leishmania major | rac serine-threonine kinase, putative,protein kinase, putative | 0.023 | 0.0074 | 1 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Echinococcus granulosus | serine/threonine protein kinase | 0.4533 | 0.6647 | 1 |
Toxoplasma gondii | calcium dependent protein kinase CDPK7 | 0.023 | 0.0074 | 0.0076 |
Entamoeba histolytica | protein kinase 2, putative | 0.4352 | 0.637 | 0.637 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Entamoeba histolytica | protein kinase, putative | 0.023 | 0.0074 | 0.0074 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Echinococcus granulosus | ribosomal protein S6 kinase alpha 3 | 0.2244 | 0.315 | 0.4739 |
Onchocerca volvulus | Putative neuronal RhoA GEF protein | 0.0181 | 0 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Loa Loa (eye worm) | AGC/NDR protein kinase | 0.2244 | 0.315 | 0.315 |
Plasmodium falciparum | calcium-dependent protein kinase 7 | 0.023 | 0.0074 | 0.0116 |
Echinococcus multilocularis | rac serine:threonine kinase | 0.4533 | 0.6647 | 1 |
Echinococcus granulosus | sodium:potassium dependent atpase beta subunit | 0.4304 | 0.6296 | 0.9473 |
Trichomonas vaginalis | AGC family protein kinase | 0.2244 | 0.315 | 0.315 |
Trypanosoma brucei | Serine/threonine-protein kinase NEK21, putative | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Onchocerca volvulus | Abnormal cell migration protein 10 homolog | 0.0181 | 0 | 0.5 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trichomonas vaginalis | AGC family protein kinase | 0.6728 | 1 | 1 |
Echinococcus multilocularis | sodium:potassium dependent atpase beta subunit | 0.4304 | 0.6296 | 0.9473 |
Loa Loa (eye worm) | AGC/PKC/ETA protein kinase | 0.2244 | 0.315 | 0.315 |
Trichomonas vaginalis | AGC family protein kinase | 0.023 | 0.0074 | 0.0074 |
Trypanosoma cruzi | NEK family Serine/threonine-protein kinase, putative | 0.023 | 0.0074 | 0.0111 |
Schistosoma mansoni | serine/threonine protein kinase | 0.2244 | 0.315 | 0.4739 |
Trypanosoma cruzi | serine/threonine protein kinase, putative | 0.023 | 0.0074 | 0.0111 |
Brugia malayi | p70 ribosomal S6 kinase beta | 0.6547 | 0.9723 | 0.9723 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 100 uM | Cytotoxicity against mouse B16 cells after 48 hrs by MTT assay | ChEMBL. | 23314049 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.