TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 317.293 | Formula: C16H15NO6
H donors: 2 H acceptors: 4 LogP: 0.38 Rotable bonds: 6
Rule of 5 violations (Lipinski): 1
SMILES: COC(=O)c1cccc(c1)NC(=O)C1[C@H]2C=C[C@@H](C1C(=O)O)O2
InChi: 1S/C16H15NO6/c1-22-16(21)8-3-2-4-9(7-8)17-14(18)12-10-5-6-11(23-10)13(12)15(19)20/h2-7,10-13H,1H3,(H,17,18)(H,19,20)/t10-,11+,12?,13?/m1/s1
InChiKey: VVTPMAWXBQQILM-IALDZJHCSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

No curated genes were found associated with this compound

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

No druggable targets predicted by sequence similarity

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Loa Loa (eye worm)	hypothetical protein	0.0039	0.2028	0.2917
Schistosoma mansoni	cd36 antigen	0.0039	0.2028	0.2028
Echinococcus granulosus	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Loa Loa (eye worm)	carboxylesterase	0.0013	0.0229	0.0329
Brugia malayi	Pyridine nucleotide-disulphide oxidoreductase, dimerisation domain containing protein	0.0011	0.0133	0.0194
Brugia malayi	Thioredoxin reductase	0.0044	0.2343	0.3414
Echinococcus multilocularis	acetylcholinesterase	0.0074	0.4408	0.4408
Mycobacterium tuberculosis	Probable NADH dehydrogenase Ndh	0.01	0.614	0.8868
Brugia malayi	hypothetical protein	0.0023	0.0959	0.1397
Entamoeba histolytica	hypothetical protein	0.0033	0.1634	0.2836
Leishmania major	acetoin dehydrogenase e3 component-like protein	0.0015	0.0406	0.0436
Echinococcus multilocularis	Basic leucine zipper (bZIP) transcription	0.0033	0.1634	0.1634
Echinococcus multilocularis	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Loa Loa (eye worm)	hypothetical protein	0.0104	0.6392	0.9194
Loa Loa (eye worm)	glutathione reductase	0.0044	0.2343	0.3369
Echinococcus multilocularis	serine:threonine protein kinase PLK1	0.0087	0.53	0.53
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Trypanosoma brucei	dihydrolipoamide dehydrogenase, point mutation	0.0015	0.0406	0.0436
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Trypanosoma cruzi	PAB1-binding protein , putative	0.0023	0.0959	0.1517
Mycobacterium tuberculosis	Probable soluble pyridine nucleotide transhydrogenase SthA (STH) (NAD(P)(+) transhydrogenase [B-specific]) (nicotinamide nucleot	0.0015	0.0406	0.0266
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Mycobacterium ulcerans	dihydrolipoamide dehydrogenase	0.0015	0.0406	1
Trypanosoma brucei	PAB1-binding protein , putative	0.0023	0.0959	0.1517
Plasmodium falciparum	dihydrolipoyl dehydrogenase, mitochondrial	0.0015	0.0406	0.1733
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Echinococcus granulosus	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0013	0.0229	0.0229
Brugia malayi	glutathione reductase	0.0044	0.2343	0.3414
Trypanosoma brucei	dihydrolipoamide dehydrogenase	0.0015	0.0406	0.0436
Loa Loa (eye worm)	thioredoxin reductase	0.0044	0.2343	0.3369
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Schistosoma mansoni	BC026374 protein (S09 family)	0.0013	0.0229	0.0229
Echinococcus multilocularis	Ataxin 2, N terminal,domain containing protein	0.001	0.0087	0.0087
Trichomonas vaginalis	DNA helicase recq, putative	0.0022	0.0884	0.137
Plasmodium vivax	dihydrolipoyl dehydrogenase, apicoplast, putative	0.0015	0.0406	0.005
Schistosoma mansoni	blooms syndrome DNA helicase	0.0018	0.0567	0.0567
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Loa Loa (eye worm)	MH2 domain-containing protein	0.011	0.6862	0.9869
Plasmodium falciparum	ataxin-2 like protein, putative	0.0023	0.0959	0.4093
Echinococcus multilocularis	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Trichomonas vaginalis	glutathione reductase, putative	0.0015	0.0406	0.0436
Echinococcus multilocularis	para nitrobenzyl esterase	0.0013	0.0229	0.0229
Brugia malayi	Carboxylesterase family protein	0.0013	0.0229	0.0333
Schistosoma mansoni	serine/threonine protein kinase	0.0087	0.53	0.53
Entamoeba histolytica	hypothetical protein	0.0033	0.1634	0.2836
Trichomonas vaginalis	spcc417.12 protein, putative	0.0013	0.0229	0.009
Plasmodium falciparum	glutathione reductase	0.0044	0.2343	1
Trypanosoma cruzi	PAB1-binding protein , putative	0.0023	0.0959	0.1517
Toxoplasma gondii	ATP-dependent DNA helicase, RecQ family protein	0.0015	0.0384	0.164
Toxoplasma gondii	LsmAD domain-containing protein	0.0023	0.0959	0.4093
Mycobacterium tuberculosis	Probable membrane NADH dehydrogenase NdhA	0.01	0.614	0.8868
Leishmania major	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Trypanosoma cruzi	trypanothione reductase, putative	0.0044	0.2343	0.4221
Trypanosoma cruzi	polo-like protein kinase, putative	0.0087	0.53	1
Schistosoma mansoni	kinase	0.0044	0.2388	0.2388
Onchocerca volvulus	Serine\/threonine kinase homolog	0.0087	0.53	0.8227
Schistosoma mansoni	hypothetical protein	0.001	0.0087	0.0087
Schistosoma mansoni	transcription factor LCR-F1	0.0033	0.1634	0.1634
Mycobacterium tuberculosis	Probable oxidoreductase	0.0111	0.6894	1
Loa Loa (eye worm)	hypothetical protein	0.0104	0.6392	0.9194
Echinococcus granulosus	Basic leucine zipper bZIP transcription	0.0033	0.1634	0.1634
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0013	0.0229	0.0229
Trypanosoma cruzi	polo-like protein kinase, putative	0.0087	0.53	1
Trypanosoma brucei	dihydrolipoyl dehydrogenase	0.0015	0.0406	0.0436
Loa Loa (eye worm)	hypothetical protein	0.0039	0.2028	0.2917
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0013	0.0229	0.0229
Leishmania major	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Plasmodium falciparum	thioredoxin reductase	0.0044	0.2343	1
Leishmania major	hypothetical protein, conserved	0.0023	0.0959	0.1517
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Plasmodium vivax	glutathione reductase, putative	0.0044	0.2343	1
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Trypanosoma cruzi	dihydrolipoyl dehydrogenase, putative	0.0015	0.0406	0.0436
Brugia malayi	hypothetical protein	0.0015	0.0399	0.0581
Plasmodium falciparum	dihydrolipoyl dehydrogenase, apicoplast	0.0015	0.0406	0.1733
Echinococcus granulosus	thioredoxin glutathione reductase	0.0044	0.2343	0.2343
Leishmania major	trypanothione reductase	0.0044	0.2343	0.4221
Toxoplasma gondii	NADPH-glutathione reductase	0.0015	0.0406	0.1733
Brugia malayi	hypothetical protein	0.0013	0.0229	0.0333
Loa Loa (eye worm)	hypothetical protein	0.0023	0.0959	0.1379
Brugia malayi	hypothetical protein	0.0039	0.2028	0.2955
Mycobacterium tuberculosis	Probable reductase	0.01	0.614	0.8868
Echinococcus granulosus	family S9 non peptidase ue S09 family	0.0013	0.0229	0.0229
Echinococcus granulosus	dihydrolipoamide dehydrogenase	0.0015	0.0406	0.0406
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Loa Loa (eye worm)	RecQ helicase	0.0022	0.0884	0.1271
Schistosoma mansoni	CD36-like class B scavenger receptor	0.0104	0.6392	0.6392
Wolbachia endosymbiont of Brugia malayi	dihydrolipoamide dehydrogenase E3 component	0.0015	0.0406	0.5
Echinococcus multilocularis	neuroligin	0.0013	0.0229	0.0229
Loa Loa (eye worm)	hypothetical protein	0.0104	0.6392	0.9194
Brugia malayi	Carboxylesterase family protein	0.0013	0.0229	0.0333
Plasmodium vivax	ataxin-2 like protein, putative	0.0023	0.0959	0.289
Echinococcus granulosus	serine:threonine protein kinase PLK1	0.0087	0.53	0.53
Trypanosoma brucei	dihydrolipoamide dehydrogenase	0.0015	0.0406	0.0436
Plasmodium vivax	thioredoxin reductase, putative	0.0044	0.2343	1
Schistosoma mansoni	neuroligin 3 (S09 family)	0.0013	0.0229	0.0229
Mycobacterium ulcerans	dihydrolipoamide dehydrogenase, LpdB	0.0015	0.0406	1
Plasmodium falciparum	ataxin-2 like protein, putative	0.0023	0.0959	0.4093
Mycobacterium tuberculosis	Probable dehydrogenase	0.01	0.614	0.8868
Trichomonas vaginalis	mercuric reductase, putative	0.0015	0.0406	0.0436
Schistosoma mansoni	dihydrolipoamide dehydrogenase	0.0015	0.0406	0.0406
Trypanosoma brucei	trypanothione reductase	0.0044	0.2343	0.4221
Loa Loa (eye worm)	acetylcholinesterase 1	0.0074	0.4408	0.634
Trypanosoma cruzi	trypanothione reductase, putative	0.0015	0.0406	0.0436
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Echinococcus multilocularis	thioredoxin glutathione reductase	0.0044	0.2343	0.2343
Brugia malayi	alpha keto acid dehydrogenase complex, E3 component, lipoamide dehydrogenase	0.0011	0.0133	0.0194
Brugia malayi	Carboxylesterase family protein	0.0013	0.0229	0.0333
Entamoeba histolytica	hypothetical protein	0.0033	0.1634	0.2836
Brugia malayi	Bloom's syndrome protein homolog	0.0022	0.0884	0.1288
Toxoplasma gondii	thioredoxin reductase	0.0044	0.2343	1
Trichomonas vaginalis	carboxylesterase domain containing protein, putative	0.0013	0.0229	0.009
Schistosoma mansoni	CD36-like class B scavenger receptor	0.0104	0.6392	0.6392
Trichomonas vaginalis	DNA helicase recq1, putative	0.0022	0.0884	0.137
Leishmania major	2-oxoglutarate dehydrogenase, e3 component, lipoamidedehydrogenase-like protein	0.0015	0.0406	0.0436
Echinococcus multilocularis	geminin	0.0157	1	1
Loa Loa (eye worm)	hypothetical protein	0.0074	0.4408	0.634
Loa Loa (eye worm)	PLK/PLK1 protein kinase	0.0087	0.53	0.7622
Echinococcus granulosus	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Echinococcus multilocularis	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Brugia malayi	serine/threonine-protein kinase plk-2	0.0087	0.53	0.7723
Echinococcus multilocularis	carboxylesterase 5A	0.0074	0.4408	0.4408
Echinococcus multilocularis	acetylcholinesterase	0.0074	0.4408	0.4408
Giardia lamblia	Kinase, PLK	0.0087	0.53	1
Echinococcus multilocularis	family S9 non peptidase ue (S09 family)	0.0013	0.0229	0.0229
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Echinococcus multilocularis	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Entamoeba histolytica	serine/threonine protein kinase, putative	0.0087	0.53	1
Echinococcus granulosus	carboxylesterase 5A	0.0074	0.4408	0.4408
Echinococcus multilocularis	lysosome membrane protein 2	0.0104	0.6392	0.6392
Brugia malayi	Carboxylesterase family protein	0.0074	0.4408	0.6425
Chlamydia trachomatis	dihydrolipoyl dehydrogenase	0.0015	0.0406	0.5
Loa Loa (eye worm)	hypothetical protein	0.0074	0.4408	0.634
Echinococcus granulosus	acetylcholinesterase	0.0074	0.4408	0.4408
Brugia malayi	Carboxylesterase family protein	0.0074	0.4408	0.6425
Mycobacterium tuberculosis	Dihydrolipoamide dehydrogenase LpdC (lipoamide reductase (NADH)) (lipoyl dehydrogenase) (dihydrolipoyl dehydrogenase) (diaphoras	0.0111	0.6894	1
Wolbachia endosymbiont of Brugia malayi	dihydrolipoamide dehydrogenase E3 component	0.0015	0.0406	0.5
Echinococcus multilocularis	dihydrolipoamide dehydrogenase	0.0015	0.0406	0.0406
Loa Loa (eye worm)	carboxylesterase	0.0013	0.0229	0.0329
Toxoplasma gondii	pyruvate dehydrogenase complex subunit PDH-E3II	0.0015	0.0406	0.1733
Plasmodium falciparum	thioredoxin reductase	0.0015	0.0406	0.1733
Echinococcus granulosus	Ataxin 2 N terminaldomain containing protein	0.001	0.0087	0.0087
Schistosoma mansoni	gliotactin	0.0013	0.0229	0.0229
Echinococcus granulosus	para nitrobenzyl esterase	0.0013	0.0229	0.0229
Echinococcus granulosus	bloom syndrome protein	0.0022	0.0884	0.0884
Mycobacterium ulcerans	flavoprotein disulfide reductase	0.0015	0.0406	1
Echinococcus granulosus	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Leishmania major	protein kinase, putative,polo-like protein kinase, putative	0.0087	0.53	1
Plasmodium vivax	dihydrolipoyl dehydrogenase, mitochondrial, putative	0.0015	0.0406	0.005
Plasmodium falciparum	glutathione reductase	0.0015	0.0406	0.1733
Toxoplasma gondii	ATP-dependent DNA helicase, RecQ family protein	0.0009	0.00000000028288	0.0000000012075
Brugia malayi	Carboxylesterase family protein	0.0013	0.0229	0.0333
Entamoeba histolytica	hypothetical protein	0.0033	0.1634	0.2836
Brugia malayi	MH2 domain containing protein	0.011	0.6862	1
Echinococcus granulosus	lysosome membrane protein 2	0.0104	0.6392	0.6392
Brugia malayi	dihydrolipoyl dehydrogenase, mitochondrial precursor, putative	0.0015	0.0406	0.0592
Brugia malayi	CD36 family protein	0.0104	0.6392	0.9316
Echinococcus granulosus	BC026374 protein S09 family	0.0013	0.0229	0.0229
Loa Loa (eye worm)	hypothetical protein	0.0039	0.2028	0.2917
Giardia lamblia	NADH oxidase lateral transfer candidate	0.0015	0.0406	0.0766
Echinococcus multilocularis	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Trypanosoma brucei	polo-like protein kinase	0.0087	0.53	1
Mycobacterium tuberculosis	NADPH-dependent mycothiol reductase Mtr	0.0044	0.2343	0.3172
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Schistosoma mansoni	acetylcholinesterase	0.0013	0.0229	0.0229
Echinococcus granulosus	CD36 class B scavenger receptor	0.0104	0.6392	0.6392
Trichomonas vaginalis	CAMK family protein kinase	0.0043	0.231	0.4157
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0074	0.4408	0.4408
Treponema pallidum	NADH oxidase	0.0015	0.0406	0.5
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Schistosoma mansoni	hypothetical protein	0.0157	1	1
Onchocerca volvulus	Lysosome membrane protein 2 homolog	0.0104	0.6392	1
Brugia malayi	hypothetical protein	0.0039	0.2028	0.2955
Mycobacterium tuberculosis	Probable nitrite reductase [NAD(P)H] large subunit [FAD flavoprotein] NirB	0.01	0.614	0.8868
Trichomonas vaginalis	CAMK family protein kinase	0.0043	0.231	0.4157
Mycobacterium tuberculosis	Putative ferredoxin reductase	0.01	0.614	0.8868
Mycobacterium leprae	DIHYDROLIPOAMIDE DEHYDROGENASE LPD (LIPOAMIDE REDUCTASE (NADH)) (LIPOYL DEHYDROGENASE) (DIHYDROLIPOYL DEHYDROGENASE) (DIAPHORASE	0.0111	0.6894	1
Trichomonas vaginalis	CAMK family protein kinase	0.0087	0.53	1
Schistosoma mansoni	hypothetical protein	0.0033	0.1634	0.1634
Loa Loa (eye worm)	carboxylesterase	0.0074	0.4408	0.634
Loa Loa (eye worm)	hypothetical protein	0.0013	0.0229	0.0329
Brugia malayi	hypothetical protein	0.0033	0.1634	0.2381
Loa Loa (eye worm)	transcription factor SMAD2	0.011	0.6862	0.9869
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0015	0.0406	0.0436
Plasmodium falciparum	ADP-dependent DNA helicase RecQ	0.002	0.0701	0.2991
Echinococcus granulosus	neuroligin	0.0013	0.0229	0.0229
Schistosoma mansoni	scavenger receptor class B type-2 (sr-B2)	0.0104	0.6392	0.6392
Echinococcus multilocularis	BC026374 protein (S09 family)	0.0013	0.0229	0.0229
Echinococcus granulosus	acetylcholinesterase	0.0074	0.4408	0.4408
Loa Loa (eye worm)	hypothetical protein	0.0112	0.6953	1
Mycobacterium tuberculosis	NAD(P)H quinone reductase LpdA	0.0111	0.6894	1
Schistosoma mansoni	hypothetical protein	0.0157	1	1
Echinococcus multilocularis	bloom syndrome protein	0.0022	0.0884	0.0884
Trypanosoma cruzi	dihydrolipoyl dehydrogenase, putative	0.0015	0.0406	0.0436

Activities

Activity type	Activity value	Assay description	Source	Reference
GI50 (functional)	= 97 uM	50% growth inhibition of A2780 (Human ovarian carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	= 97 uM	50% growth inhibition of A2780 (Human ovarian carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of G401 (human kidney carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of HT-29 (human colorectal carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of H460 (human lung carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of L1210 (murine leukemia) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of G401 (human kidney carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of HT-29 (human colorectal carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of H460 (human lung carcinoma) cell line compared with untreated control cells	ChEMBL.	15050639
GI50 (functional)	> 100 uM	50% growth inhibition of L1210 (murine leukemia) cell line compared with untreated control cells	ChEMBL.	15050639
IC50 (binding)	= 12 uM	Inhibitory activity against protein phosphatase 2A from human red blood cells	ChEMBL.	15050639
IC50 (binding)	= 60 uM	Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscle	ChEMBL.	15050639
IC50 (binding)	= 60 uM	Inhibitory activity against protein phosphatase-1 from rabbit skeletal muscle	ChEMBL.	15050639

Phenotypes

Whole-cell/tissue/organism interactions

We have no records of whole-cell/tissue assays done with this compound What does this mean?

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL175576

Bibliographic References

1 literature reference was collected for this gene.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 311368