Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0014 | 0 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0014 | 0 | 0.5 |
Trichomonas vaginalis | acetylornithine aminotransferase, putative | 0.0044 | 0.0615 | 1 |
Echinococcus granulosus | ornithine aminotransferase | 0.0044 | 0.0615 | 1 |
Echinococcus multilocularis | ornithine aminotransferase | 0.0044 | 0.0615 | 1 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Plasmodium vivax | ornithine aminotransferase, putative | 0.0044 | 0.0615 | 1 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | beta-tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | alpha tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma cruzi | beta tubulin, putative | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Entamoeba histolytica | tubulin gamma chain | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | tubulin gamma chain | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0014 | 0 | 0.5 |
Mycobacterium leprae | Probable Acetylornithine aminotransferase ArgD | 0.0044 | 0.0615 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | hypothetical protein | 0.0014 | 0 | 0.5 |
Mycobacterium leprae | PROBABLE GLUTAMATE-1-SEMIALDEHYDE 2,1-AMINOMUTASE HEML (GSA) (GLUTAMATE-1-SEMIALDEHYDE AMINOTRANSFERASE) (GSA-AT) | 0.0044 | 0.0615 | 0.5 |
Chlamydia trachomatis | glutamate-1-semialdehyde-2,1-aminomutase | 0.0044 | 0.0615 | 0.5 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | alpha tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0014 | 0 | 0.5 |
Toxoplasma gondii | ornithine aminotransferase, mitochondrial precursor, putative | 0.0044 | 0.0615 | 1 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | alpha-tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | gamma-tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0014 | 0 | 0.5 |
Giardia lamblia | Alpha-tubulin | 0.0014 | 0 | 0.5 |
Mycobacterium tuberculosis | Probable L-lysine-epsilon aminotransferase Lat (L-lysine aminotransferase) (lysine 6-aminotransferase) | 0.049 | 1 | 1 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0014 | 0 | 0.5 |
Giardia lamblia | Gamma tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Echinococcus multilocularis | ornithine aminotransferase | 0.0044 | 0.0615 | 1 |
Mycobacterium leprae | Probable 4-aminobutyrate aminotransferase GabT (GAMMA-AMINO-N-BUTYRATE TRANSAMINASE) (GABA TRANSAMINASE) (GLUTAMATE:SUCCINIC SEM | 0.0044 | 0.0615 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | epsilon tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin beta chain | 0.0014 | 0 | 0.5 |
Trypanosoma cruzi | tubulin gamma chain | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Echinococcus multilocularis | Aminotransferase class III | 0.0044 | 0.0615 | 1 |
Leishmania major | epsilon tubulin, putative | 0.0014 | 0 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | alpha tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Giardia lamblia | Alpha-tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | BEN-1 protein | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | epsilon tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | alpha tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Wolbachia endosymbiont of Brugia malayi | acetylornithine transaminase protein | 0.0044 | 0.0615 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | epsilon tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | alpha-tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Mycobacterium leprae | PROBABLE ADENOSYLMETHIONINE-8-AMINO-7-OXONONANOATE AMINOTRANSFERASE BIOA | 0.0044 | 0.0615 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma brucei | beta tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Giardia lamblia | Beta tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Schistosoma mansoni | ornithine--oxo-acid transaminase | 0.0044 | 0.0615 | 1 |
Trypanosoma brucei | beta tubulin | 0.0014 | 0 | 0.5 |
Echinococcus granulosus | Aminotransferase class III | 0.0044 | 0.0615 | 1 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Entamoeba histolytica | tubulin family protein | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Mycobacterium ulcerans | L-lysine aminotransferase | 0.049 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0014 | 0 | 0.5 |
Plasmodium falciparum | ornithine aminotransferase | 0.0044 | 0.0615 | 1 |
Leishmania major | beta tubulin | 0.0014 | 0 | 0.5 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0014 | 0 | 0.5 |
Leishmania major | alpha tubulin | 0.0014 | 0 | 0.5 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.