TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 291.365 | Formula: C15H17NO3S
H donors: 1 H acceptors: 3 LogP: 3.17 Rotable bonds: 5
Rule of 5 violations (Lipinski): 1
SMILES: CCCN(S(=O)(=O)c1ccc(cc1)O)c1ccccc1
InChi: 1S/C15H17NO3S/c1-2-12-16(13-6-4-3-5-7-13)20(18,19)15-10-8-14(17)9-11-15/h3-11,17H,2,12H2,1H3
InChiKey: VUUWGEGTDFUSTR-UHFFFAOYSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

Species	Target name	Source	Bibliographic reference
Homo sapiens	estrogen receptor 1	Starlite/ChEMBL	References

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

No druggable targets predicted by sequence similarity

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Trichomonas vaginalis	ABC transporter, putative	0.001	0.0062	1
Schistosoma mansoni	notch	0.0165	0.3133	0.3132
Brugia malayi	Peroxidasin	0.0509	1	1
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Echinococcus multilocularis	ATP binding cassette subfamily B (MDR:TAP)	0.001	0.0062	0.0062
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	Notch2	0.0165	0.3133	0.3132
Echinococcus granulosus	hepatocyte nuclear factor 4 alpha	0.0007	0.0002	0.0002
Trichomonas vaginalis	ABC transporter, half transporter, putative	0.001	0.0062	1
Trichomonas vaginalis	ATP-binding cassette transporter, putative	0.001	0.0062	1
Onchocerca volvulus	Peroxidase homolog	0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus granulosus	notch	0.0165	0.3133	0.3133
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Echinococcus multilocularis	neurogenic locus notch protein	0.0165	0.3133	0.3133
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Schistosoma mansoni	Pro-neuregulin-4 membrane-bound isoform (Pro-NRG4) [Contains: Neuregulin-4 (NRG-4)]	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus multilocularis	thyroid hormone receptor alpha	0.0007	0.0002	0.0002
Brugia malayi	Transmembrane cell adhesion receptor mua-3 precursor, putative	0.0165	0.3133	0.3132
Echinococcus multilocularis	neurogenic locus protein delta	0.0165	0.3133	0.3133
Brugia malayi	GCC2 and GCC3 family protein	0.0165	0.3133	0.3132
Schistosoma mansoni	septate junction protein	0.0165	0.3133	0.3132
Onchocerca volvulus		0.0165	0.3133	0.3132
Echinococcus multilocularis	hepatocyte nuclear factor 4 alpha	0.0007	0.0002	0.0002
Brugia malayi	Calcium binding EGF domain containing protein	0.0165	0.3133	0.3132
Giardia lamblia	High cysteine protein	0.0165	0.3133	0.5
Echinococcus granulosus	neurogenic locus notch protein 4	0.0165	0.3133	0.3133
Echinococcus granulosus	COUP TF:Svp nuclear hormone receptor	0.0007	0.0002	0.0002
Loa Loa (eye worm)	blistered cuticle protein 3	0.0509	1	1
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	ATP-binding cassette sub-family B member 2	0.001	0.0062	0.006
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Leishmania major	ATP-binding cassette protein subfamily B, member 2, putative	0.001	0.0062	0.5
Brugia malayi	Animal haem peroxidase family protein	0.0509	1	1
Echinococcus multilocularis	slit 2 protein	0.0165	0.3133	0.3133
Leishmania major	p-glycoprotein	0.001	0.0062	0.5
Trichomonas vaginalis	ABC transporter, putative	0.001	0.0062	1
Trichomonas vaginalis	ABC transporter, half transporter, putative	0.001	0.0062	1
Echinococcus granulosus	multidrug resistance protein 1	0.001	0.0062	0.0062
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Schistosoma mansoni	multidrug resistance protein	0.001	0.0062	0.006
Loa Loa (eye worm)	notch protein	0.0165	0.3133	0.3132
Echinococcus granulosus	multidrug resistance protein 1	0.001	0.0062	0.0062
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Schistosoma mansoni	smdr2	0.001	0.0062	0.006
Schistosoma mansoni	peroxidasin	0.0509	1	1
Brugia malayi	ABC transporter family protein	0.001	0.0062	0.006
Trichomonas vaginalis	ATP-binding cassette transporter, putative	0.001	0.0062	1
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Echinococcus granulosus	ecdysone induced protein 78C	0.0007	0.0002	0.0002
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Schistosoma mansoni	notch	0.0165	0.3133	0.3132
Brugia malayi	Animal haem peroxidase family protein	0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus granulosus	multidrug resistance protein 1	0.001	0.0062	0.0062
Onchocerca volvulus	Peroxidasin homolog	0.0509	1	1
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Brugia malayi	Cadherin domain containing protein	0.0165	0.3133	0.3132
Onchocerca volvulus		0.001	0.0062	0.006
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Schistosoma mansoni	multidrug resistance protein	0.001	0.0062	0.006
Entamoeba histolytica	P-glycoprotein-5	0.001	0.0062	0.5
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Echinococcus multilocularis	ATP binding cassette subfamily B (MDR:TAP)	0.001	0.0062	0.0062
Echinococcus multilocularis	nuclear receptor 2DBD gamma	0.0007	0.0002	0.0002
Echinococcus granulosus	ATP binding cassette subfamily B MDR:TAP	0.001	0.0062	0.0062
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Toxoplasma gondii	EGF family domain-containing protein	0.0165	0.3133	1
Schistosoma mansoni	notch	0.0165	0.3133	0.3132
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Plasmodium vivax	multidrug resistance protein 1, putative	0.001	0.0062	0.5
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus granulosus	5'partial\|ATP binding cassette sub family B	0.001	0.006	0.006
Echinococcus granulosus	protein jagged 2	0.0165	0.3133	0.3133
Echinococcus granulosus	protein jagged 1	0.0165	0.3133	0.3133
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Echinococcus multilocularis	ATP binding cassette subfamily B (MDR:TAP)	0.001	0.0062	0.0062
Echinococcus granulosus	neurogenic locus notch protein	0.0165	0.3133	0.3133
Schistosoma mansoni	notch	0.0165	0.3133	0.3132
Brugia malayi	Animal haem peroxidase family protein	0.0509	1	1
Echinococcus multilocularis	FTZ F1 alpha	0.0007	0.0002	0.0002
Mycobacterium tuberculosis	Probable transmembrane multidrug efflux pump	0.001	0.0062	0.5
Echinococcus granulosus	neurogenic locus protein delta	0.0165	0.3133	0.3133
Echinococcus granulosus	retinoic acid receptor rxr beta a	0.0007	0.0002	0.0002
Onchocerca volvulus	Dual oxidase homolog	0.0509	1	1
Onchocerca volvulus		0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	animal heme peroxidase	0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Brugia malayi	Animal haem peroxidase family protein	0.0509	1	1
Echinococcus granulosus	ATP binding cassette subfamily B MDR:TAP	0.001	0.0062	0.0062
Echinococcus granulosus	Nuclear hormone receptor family member nhr 41	0.0007	0.0002	0.0002
Echinococcus multilocularis	protein jagged 1	0.0165	0.3133	0.3133
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus granulosus	neural cadherin	0.0165	0.3133	0.3133
Echinococcus multilocularis	fibropellin Ia	0.0165	0.3133	0.3133
Echinococcus granulosus	ATP binding cassette subfamily B MDR:TAP	0.001	0.0062	0.0062
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Entamoeba histolytica	P-glycoprotein-2	0.001	0.0062	0.5
Echinococcus granulosus	ATP binding cassette subfamily B MDR:TAP	0.001	0.0062	0.0062
Schistosoma mansoni	slit	0.0165	0.3133	0.3132
Onchocerca volvulus	Neurogenic locus notch homolog	0.0165	0.3133	0.3132
Echinococcus multilocularis	fat cadherin tumor suppressor	0.0165	0.3133	0.3133
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Trichomonas vaginalis	taga, putative	0.001	0.0062	1
Onchocerca volvulus		0.0165	0.3133	0.3132
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Echinococcus multilocularis	multidrug resistance protein 1	0.001	0.0062	0.0062
Onchocerca volvulus	Peroxidase homolog	0.0509	1	1
Brugia malayi	multidrug resistance protein 3	0.001	0.0062	0.006
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Echinococcus multilocularis	ATP binding cassette sub family B	0.001	0.006	0.006
Echinococcus multilocularis	FTZ F1 nuclear receptor protein	0.0007	0.0002	0.0002
Echinococcus granulosus	peroxidasin	0.0509	1	1
Entamoeba histolytica	P-glycoprotein-1	0.001	0.0062	0.5
Echinococcus multilocularis	ATP binding cassette subfamily B (MDR:TAP)	0.001	0.0062	0.0062
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Echinococcus granulosus	delta-like protein 1	0.0165	0.3133	0.3133
Onchocerca volvulus	Slit protein homolog	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Trichomonas vaginalis	ATP-binding cassette transporter, putative	0.001	0.0062	1
Trichomonas vaginalis	ATP-binding cassette transporter, putative	0.001	0.0062	1
Loa Loa (eye worm)	animal heme peroxidase	0.0509	1	1
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Echinococcus multilocularis	ecdysone induced protein 78C	0.0007	0.0002	0.0002
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Onchocerca volvulus		0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.001	0.0062	0.006
Echinococcus multilocularis	neurogenic locus protein delta	0.0165	0.3133	0.3133
Echinococcus granulosus	protein jagged 1	0.0165	0.3133	0.3133
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	multidrug resistance protein 3	0.001	0.0062	0.006
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.001	0.0062	0.006
Echinococcus granulosus	fibropellin Ia	0.0165	0.3133	0.3133
Onchocerca volvulus	Peroxidasin homolog	0.0509	1	1
Onchocerca volvulus	Neurogenic locus notch protein homolog	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Brugia malayi	Calcium binding EGF domain containing protein	0.0165	0.3133	0.3132
Echinococcus granulosus	neurogenic locus notch protein	0.0165	0.3133	0.3133
Trichomonas vaginalis	ATP-binding cassette transporter, putative	0.001	0.0062	1
Schistosoma mansoni	notch	0.0165	0.3133	0.3132
Brugia malayi	Muscle positioning protein 4	0.0165	0.3133	0.3132
Loa Loa (eye worm)	animal heme peroxidase	0.0509	1	1
Onchocerca volvulus		0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Schistosoma mansoni	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Brugia malayi	Delta serrate ligand family protein	0.0165	0.3133	0.3132
Echinococcus multilocularis	notch	0.0165	0.3133	0.3133
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Brugia malayi	notch-like transmembrane receptor	0.0165	0.3133	0.3132
Trichomonas vaginalis	ABC transporter, putative	0.001	0.0062	1
Brugia malayi	Blistered cuticle protein 3	0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.001	0.006	0.0058
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Echinococcus multilocularis	peroxidasin	0.0509	1	1
Brugia malayi	Calcium binding EGF domain containing protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	animal heme peroxidase	0.0509	1	1
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Schistosoma mansoni	notch	0.0165	0.3133	0.3132
Echinococcus multilocularis	neurogenic locus notch protein	0.0165	0.3133	0.3133
Echinococcus multilocularis	nuclear receptor 2DBD gamma	0.0007	0.0002	0.0002
Trichomonas vaginalis	abcb9, putative	0.001	0.0062	1
Echinococcus multilocularis	neural cadherin	0.0165	0.3133	0.3133
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Echinococcus granulosus	FTZ F1 nuclear receptor protein	0.0007	0.0002	0.0002
Schistosoma mansoni	multidrug resistance protein	0.001	0.0062	0.006
Entamoeba histolytica	P-glycoprotein-2, putative	0.001	0.0062	0.5
Trichomonas vaginalis	ABC transporter, putative	0.001	0.0062	1
Echinococcus multilocularis	protein jagged 2	0.0165	0.3133	0.3133
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus granulosus	slit 2 protein	0.0165	0.3133	0.3133
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Trichomonas vaginalis	abcb9, putative	0.001	0.0062	1
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Trichomonas vaginalis	abcb9, putative	0.001	0.0062	1
Echinococcus multilocularis	multidrug resistance protein 1	0.001	0.0062	0.0062
Onchocerca volvulus	Chorion peroxidase homolog	0.0509	1	1
Entamoeba histolytica	P-glycoprotein 5, putative	0.001	0.0062	0.5
Brugia malayi	EGF-like domain containing protein	0.0165	0.3133	0.3132
Onchocerca volvulus		0.0165	0.3133	0.3132
Echinococcus granulosus	protein jagged 2	0.0165	0.3133	0.3133
Echinococcus granulosus	nuclear receptor 2DBD gamma	0.0007	0.0002	0.0002
Schistosoma mansoni	peroxidasin	0.0509	1	1
Onchocerca volvulus		0.0509	1	1
Onchocerca volvulus		0.0509	1	1
Echinococcus multilocularis	neurogenic locus notch protein 4	0.0165	0.3133	0.3133
Echinococcus multilocularis	COUP TF:Svp nuclear hormone receptor	0.0007	0.0002	0.0002
Entamoeba histolytica	P-glycoprotein-2	0.001	0.0062	0.5
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Entamoeba histolytica	P-glyco protein 6, putative	0.001	0.0062	0.5
Schistosoma mansoni	laminin gamma-3 chain	0.0165	0.3133	0.3132
Trichomonas vaginalis	multidrug resistance protein 1, 2, putative	0.001	0.0062	1
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Trichomonas vaginalis	lipid A export ATP-binding/permease protein msba, putative	0.001	0.0062	1
Brugia malayi	Cadherin domain containing protein	0.0165	0.3133	0.3132
Loa Loa (eye worm)	hypothetical protein	0.0165	0.3133	0.3132
Echinococcus granulosus	FTZ F1 alpha	0.0007	0.0002	0.0002
Schistosoma mansoni	cell polarity protein	0.0165	0.3133	0.3132
Chlamydia trachomatis	ABC transporter ATP binding protein/permease	0.001	0.0062	0.5
Onchocerca volvulus	Putative cubilin	0.0165	0.3133	0.3132
Echinococcus multilocularis	protein jagged 1	0.0165	0.3133	0.3133
Loa Loa (eye worm)	hypothetical protein	0.0509	1	1
Brugia malayi	Animal haem peroxidase family protein	0.0509	1	1
Plasmodium falciparum	multidrug resistance protein 1	0.001	0.0062	0.5
Echinococcus multilocularis	Nuclear hormone receptor family member nhr 41	0.0007	0.0002	0.0002
Echinococcus granulosus	nuclear receptor 2DBD gamma	0.0007	0.0002	0.0002
Echinococcus multilocularis	ATP binding cassette subfamily B (MDR:TAP)	0.001	0.0062	0.0062

Activities

Activity type	Activity value	Assay description	Source	Reference
EC50 (functional)	= 1430 nM	Effect on binding to ER in Ad5-wt-ER-infected HAECT1 cells by creatine kinase expression	ChEMBL.	16300947
EC50 (functional)	= 1430 nM	Effect on binding to ER in Ad5-wt-ER-infected HAECT1 cells by creatine kinase expression	ChEMBL.	16300947
Efficacy (functional)	= 0.77 %	Selectivity for NFkappaB expression over creatine kinase expression in Ad5-wt-ER-infected HAECT1 cells	ChEMBL.	16300947
Efficacy (functional)	= 0.77 %	Selectivity for NFkappaB expression over creatine kinase expression in Ad5-wt-ER-infected HAECT1 cells	ChEMBL.	16300947
Efficacy (functional)	= 88 %	Effect on binding to ER in Ad5-wt-ER-infected HAECT1 cells by creatine kinase expression at 10 uM relative to estradiol	ChEMBL.	16300947
Efficacy (functional)	= 88 %	Effect on binding to ER in Ad5-wt-ER-infected HAECT1 cells by creatine kinase expression at 10 uM relative to estradiol	ChEMBL.	16300947
Efficacy (functional)	= 113 %	Effect on binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB luciferase reporter at 10 uM relative to estradiol	ChEMBL.	16300947
Efficacy (functional)	= 113 %	Effect on binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB luciferase reporter at 10 uM relative to estradiol	ChEMBL.	16300947
IC50 (functional)	= 303 nM	Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporter	ChEMBL.	16300947
IC50 (functional)	= 303 nM	Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporter	ChEMBL.	16300947

Phenotypes

Whole-cell/tissue/organism interactions

We have no records of whole-cell/tissue assays done with this compound What does this mean?

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL205070

Bibliographic References

1 literature reference was collected for this gene.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 352856