TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 1032.2 | Formula: C53H69N13O9
H donors: 12 H acceptors: 10 LogP: 2.5 Rotable bonds: 35
Rule of 5 violations (Lipinski): 3
SMILES: CC(C[C@@H](C(=O)N[C@H](C(=O)N)CC(C)C)NC(=O)[C@@H](NC(=O)c1cccc(c1)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)N)CCC(=O)N)C)Cc1nc[nH]c1)C
InChi: 1S/C53H69N13O9/c1-29(2)20-41(46(56)68)63-52(74)42(21-30(3)4)65-53(75)44(25-36-27-57-28-59-36)64-48(70)33-14-11-15-35(23-33)61-47(69)31(5)60-51(73)43(24-34-26-58-39-17-10-9-16-37(34)39)66-50(72)40(18-19-45(55)67)62-49(71)38(54)22-32-12-7-6-8-13-32/h6-17,23,26-31,38,40-44,58H,18-22,24-25,54H2,1-5H3,(H2,55,67)(H2,56,68)(H,57,59)(H,60,73)(H,61,69)(H,62,71)(H,63,74)(H,64,70)(H,65,75)(H,66,72)/t31-,38-,40-,41-,42-,43-,44-/m0/s1
InChiKey: ZARTZEIYNBUNPR-USXQZJOHSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

Species	Target name	Source	Bibliographic reference
Rattus norvegicus	Gastrin releasing peptide receptor	Starlite/ChEMBL	References

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

Species	Potential target	Known druggable target	Length	Alignment span	Identity
Schistosoma japonicum	ko:K04134 cholinergic receptor, invertebrate, putative	Gastrin releasing peptide receptor	384 aa	329 aa	23.1 %
Echinococcus granulosus	allatostatin A receptor	Gastrin releasing peptide receptor	384 aa	349 aa	27.2 %
Schistosoma japonicum	ko:K04209 neuropeptide Y receptor, invertebrate, putative	Gastrin releasing peptide receptor	384 aa	327 aa	27.8 %
Echinococcus multilocularis	pyroglutamylated rfamide peptide receptor	Gastrin releasing peptide receptor	384 aa	386 aa	19.9 %
Echinococcus granulosus	pyroglutamylated rfamide peptide receptor	Gastrin releasing peptide receptor	384 aa	385 aa	21.0 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	314 aa	22.0 %
Schistosoma mansoni	peptide (allatostatin)-like receptor	Gastrin releasing peptide receptor	384 aa	315 aa	27.3 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	330 aa	26.4 %
Onchocerca volvulus	Mitochondrial inner membrane protein homolog	Gastrin releasing peptide receptor	384 aa	370 aa	21.9 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	324 aa	24.4 %
Brugia malayi	ORL1-like opioid receptor	Gastrin releasing peptide receptor	384 aa	354 aa	22.3 %
Echinococcus multilocularis	thyrotropin releasing hormone receptor	Gastrin releasing peptide receptor	384 aa	385 aa	25.2 %
Schistosoma mansoni	biogenic amine (octopamine/dopamine) receptor	Gastrin releasing peptide receptor	384 aa	358 aa	22.9 %
Echinococcus granulosus	thyrotropin releasing hormone receptor	Gastrin releasing peptide receptor	384 aa	385 aa	25.2 %
Schistosoma japonicum	ko:K04135 adrenergic receptor, alpha 1a, putative	Gastrin releasing peptide receptor	384 aa	398 aa	23.6 %
Schistosoma japonicum	Rhodopsin, putative	Gastrin releasing peptide receptor	384 aa	327 aa	21.7 %
Schistosoma mansoni	biogenic amine (5HT) receptor	Gastrin releasing peptide receptor	384 aa	399 aa	23.6 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	333 aa	25.2 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	377 aa	22.0 %
Echinococcus multilocularis	allatostatin A receptor	Gastrin releasing peptide receptor	384 aa	375 aa	27.2 %
Echinococcus multilocularis	neuropeptide receptor	Gastrin releasing peptide receptor	384 aa	316 aa	26.3 %
Echinococcus granulosus	neuropeptide receptor	Gastrin releasing peptide receptor	384 aa	316 aa	26.6 %

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Brugia malayi	p70 ribosomal S6 kinase beta	0.0207	0.4247	0.3821
Echinococcus granulosus	serine/threonine protein kinase	0.0146	0.2712	1
Brugia malayi	Hr1 repeat family protein	0.0071	0.0833	0.0154
Trichomonas vaginalis	AGC family protein kinase	0.0071	0.0833	0.0883
Chlamydia trachomatis	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Echinococcus multilocularis	peptidase Clp (S14 family)	0.006	0.0557	0.2053
Echinococcus multilocularis	Ataxin 2, N terminal,domain containing protein	0.0073	0.0889	0.3278
Loa Loa (eye worm)	AGC/PKN protein kinase	0.0071	0.0833	0.0154
Trichomonas vaginalis	AGC family protein kinase	0.0071	0.0833	0.0883
Echinococcus granulosus	ATP dependent Clp protease proteolytic subunit	0.0092	0.1347	0.4969
Loa Loa (eye worm)	AGC/AKT protein kinase	0.0216	0.4453	0.4042
Entamoeba histolytica	PH domain containing protein kinase, putative	0.0146	0.2712	0.5373
Echinococcus multilocularis	sodium:potassium dependent atpase beta subunit	0.0136	0.2467	0.9097
Echinococcus multilocularis	protein kinase c epsilon type	0.0071	0.0833	0.3071
Trichomonas vaginalis	low molecular weight protein tyrosine phosphatase, putative	0.0185	0.3689	0.8077
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Schistosoma mansoni	atypical protein kinase C	0.0071	0.0833	0.0246
Echinococcus multilocularis	tyrosyl DNA phosphodiesterase 1	0.0065	0.0689	0.2541
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Mycobacterium leprae	PROBABLE ATP-DEPENDENT CLP PROTEASE PROTEOLYTIC SUBUNIT 2 CLPP2 (ENDOPEPTIDASE CLP 2)	0.0092	0.1347	1
Schistosoma mansoni	hypothetical protein	0.0299	0.6536	1
Plasmodium falciparum	ataxin-2 like protein, putative	0.0163	0.3146	1
Trichomonas vaginalis	low molecular weight protein-tyrosine-phosphatase, putative	0.0185	0.3689	0.8077
Echinococcus multilocularis	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Echinococcus multilocularis	GPCR, family 2	0.0138	0.2517	0.9281
Leishmania major	tyrosyl-DNA phosphodiesterase 1	0.0065	0.0689	0.0777
Trichomonas vaginalis	low molecular weight protein-tyrosine-phosphatase, putative	0.0185	0.3689	0.8077
Brugia malayi	hypothetical protein	0.0105	0.1695	0.1081
Brugia malayi	calcium-independent alpha-latrotoxin receptor 2, putative	0.0138	0.2517	0.1963
Brugia malayi	Protein kinase domain containing protein	0.0071	0.0833	0.0154
Plasmodium falciparum	ataxin-2 like protein, putative	0.0163	0.3146	1
Brugia malayi	Calcitonin receptor-like protein seb-1	0.0437	1	1
Loa Loa (eye worm)	AGC/RSK/P70 protein kinase	0.0207	0.4247	0.3821
Mycobacterium ulcerans	phosphotyrosine protein phosphatase PtpA	0.0185	0.3689	1
Loa Loa (eye worm)	hypothetical protein	0.0092	0.1347	0.0707
Brugia malayi	latrophilin 2 splice variant baaae	0.0299	0.6536	0.628
Echinococcus granulosus	serine threonine protein kinase nrc	0.0138	0.2505	0.9239
Trypanosoma cruzi	tyrosyl-DNA Phosphodiesterase (Tdp1), putative	0.0065	0.0689	0.0777
Brugia malayi	Pax transcription factor protein 2	0.0259	0.553	0.5199
Loa Loa (eye worm)	hypothetical protein	0.0437	1	1
Trichomonas vaginalis	AGC family protein kinase	0.0079	0.1039	0.1403
Entamoeba histolytica	protein kinase, putative	0.0071	0.0833	0.0381
Trypanosoma cruzi	isocitrate dehydrogenase, putative	0.0085	0.1193	0.267
Onchocerca volvulus		0.0259	0.553	1
Schistosoma mansoni	hypothetical protein	0.0073	0.0889	0.0341
Echinococcus multilocularis	serine:threonine protein kinase N2	0.0071	0.0833	0.3071
Entamoeba histolytica	protein kinase, putative	0.0216	0.4453	1
Echinococcus granulosus	tyrosyl DNA phosphodiesterase 1	0.0065	0.0689	0.2541
Loa Loa (eye worm)	AGC/RSK/RSK protein kinase	0.0071	0.0833	0.0154
Trichomonas vaginalis	AGC family protein kinase	0.0071	0.0833	0.0883
Echinococcus granulosus	nervana 2	0.0136	0.2467	0.9097
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Echinococcus multilocularis	protein kinase c iota type	0.0071	0.0833	0.3071
Loa Loa (eye worm)	AGC/DMPK/GEK protein kinase	0.0071	0.0833	0.0154
Echinococcus multilocularis	isocitrate dehydrogenase 2 (NADP+)	0.0085	0.1193	0.4401
Trichomonas vaginalis	low molecular weight protein tyrosine phosphatase, putative	0.0185	0.3689	0.8077
Brugia malayi	isocitrate dehydrogenase	0.0085	0.1193	0.0541
Echinococcus granulosus	Glutaredoxin protein 5	0.0136	0.2467	0.9097
Loa Loa (eye worm)	isocitrate dehydrogenase	0.0085	0.1193	0.0541
Giardia lamblia	Low molecular weight protein-tyrosine-phosphatase	0.0185	0.3689	1
Brugia malayi	hypothetical protein	0.0163	0.3146	0.2639
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Wolbachia endosymbiont of Brugia malayi	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Brugia malayi	Latrophilin receptor protein 2	0.0138	0.2517	0.1963
Trypanosoma cruzi	PAB1-binding protein , putative	0.0163	0.3146	1
Trypanosoma brucei	tyrosyl-DNA Phosphodiesterase (Tdp1), putative	0.0065	0.0689	0.0521
Trypanosoma brucei	rac serine-threonine kinase, putative	0.0216	0.4453	1
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Toxoplasma gondii	LsmAD domain-containing protein	0.0163	0.3146	0.6395
Toxoplasma gondii	AGC kinase	0.0207	0.4247	1
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Loa Loa (eye worm)	AGC/RSK/MSK protein kinase	0.0071	0.0833	0.0154
Loa Loa (eye worm)	pigment dispersing factor receptor c	0.0437	1	1
Echinococcus granulosus	cadherin EGF LAG seven pass G type receptor	0.0138	0.2517	0.9281
Entamoeba histolytica	protein kinase, putative	0.0207	0.4247	0.9452
Entamoeba histolytica	protein kinase, putative	0.0216	0.4453	1
Trypanosoma cruzi	PAB1-binding protein , putative	0.0163	0.3146	1
Echinococcus granulosus	Ribosomal protein S6 kinase beta 2	0.0071	0.0833	0.3071
Trypanosoma brucei	PAB1-binding protein , putative	0.0163	0.3146	0.6709
Echinococcus granulosus	diuretic hormone 44 receptor GPRdih2	0.0138	0.2517	0.9281
Loa Loa (eye worm)	hypothetical protein	0.0299	0.6536	0.628
Echinococcus multilocularis	Ribosomal protein S6 kinase beta 2	0.0071	0.0833	0.3071
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Schistosoma mansoni	serine/threonine kinase	0.0071	0.0833	0.0246
Loa Loa (eye worm)	AGC/PKC/ETA protein kinase	0.0071	0.0833	0.0154
Echinococcus multilocularis	cadherin EGF LAG seven pass G type receptor	0.0138	0.2517	0.9281
Echinococcus multilocularis	serine:threonine protein kinase 38	0.0071	0.0833	0.3071
Echinococcus granulosus	GPCR family 2	0.0138	0.2517	0.9281
Echinococcus multilocularis	serine threonine protein kinase nrc serine threonine protein kinase gad	0.0138	0.2505	0.9239
Plasmodium vivax	rac-beta serine/threonine protein kinase, putative	0.0138	0.2505	0.6718
Schistosoma mansoni	peptidase Clp (S14 family)	0.0092	0.1347	0.1126
Loa Loa (eye worm)	pax transcription factor protein 2	0.0259	0.553	0.5199
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Treponema pallidum	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Echinococcus multilocularis	rac serine:threonine kinase	0.0146	0.2712	1
Echinococcus granulosus	protein kinase c epsilon type	0.0071	0.0833	0.3071
Echinococcus granulosus	protein kinase c iota type	0.0071	0.0833	0.3071
Trypanosoma cruzi	isocitrate dehydrogenase [NADP], mitochondrial precursor, putative	0.0085	0.1193	0.267
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Loa Loa (eye worm)	phosphotyrosine protein phosphatase	0.0185	0.3689	0.3222
Echinococcus granulosus	nervana 2	0.0136	0.2467	0.9097
Loa Loa (eye worm)	hypothetical protein	0.0138	0.2517	0.1963
Trypanosoma cruzi	rac serine-threonine kinase, putative	0.0146	0.2712	0.8369
Entamoeba histolytica	PH domain containing protein kinase, putative	0.0146	0.2712	0.5373
Leishmania major	hypothetical protein, conserved	0.0163	0.3146	1
Trypanosoma cruzi	rac serine-threonine kinase, putative	0.0138	0.2505	0.7594
Echinococcus granulosus	ribosomal protein S6 kinase alpha 3	0.0071	0.0833	0.3071
Brugia malayi	protein kinase C II.	0.0071	0.0833	0.0154
Plasmodium vivax	ATP-dependent Clp protease proteolytic subunit, putative	0.0092	0.1347	0.0788
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Echinococcus multilocularis	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Echinococcus multilocularis	nervana 2	0.0136	0.2467	0.9097
Echinococcus multilocularis	ATP dependent Clp protease proteolytic subunit	0.0092	0.1347	0.4969
Trichomonas vaginalis	low molecular weight protein-tyrosine-phosphatase, putative	0.0185	0.3689	0.8077
Brugia malayi	Protein kinase domain containing protein	0.0071	0.0833	0.0154
Echinococcus granulosus	ribosomal protein s6 kinase beta 1	0.0071	0.0833	0.3071
Echinococcus multilocularis	Protein kinase C, brain isozyme	0.0071	0.0833	0.3071
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Loa Loa (eye worm)	latrophilin receptor protein 2	0.0138	0.2517	0.1963
Schistosoma mansoni	NADP-specific isocitrate dehydrogenase	0.0085	0.1193	0.0862
Echinococcus granulosus	serine:threonine protein kinase N2	0.0071	0.0833	0.3071
Trypanosoma cruzi	Protein kinase B	0.0146	0.2712	0.8369
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Plasmodium falciparum	RAC-beta serine/threonine protein kinase	0.0138	0.2505	0.6718
Schistosoma mansoni	serine/threonine-protein kinase	0.0146	0.2712	0.3459
Leishmania major	isocitrate dehydrogenase [NADP], mitochondrial precursor, putative	0.0085	0.1193	0.267
Echinococcus multilocularis	ribosomal protein S6 kinase alpha 3	0.0071	0.0833	0.3071
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Entamoeba histolytica	protein tyrosine phosphatase, putative	0.0185	0.3689	0.7971
Echinococcus granulosus	peptidase Clp S14 family	0.006	0.0557	0.2053
Trypanosoma brucei	isocitrate dehydrogenase, putative	0.0085	0.1193	0.1791
Trichomonas vaginalis	low molecular weight protein tyrosine phosphatase, putative	0.0185	0.3689	0.8077
Echinococcus multilocularis	isocitrate dehydrogenase	0.0085	0.1193	0.4401
Toxoplasma gondii	ATP-dependent Clp endopeptidase, proteolytic subunit ClpP domain-containing protein	0.0092	0.1347	0.0504
Loa Loa (eye worm)	hypothetical protein	0.0071	0.0833	0.0154
Brugia malayi	Protein kinase domain containing protein	0.0216	0.4453	0.4042
Toxoplasma gondii	ATP-dependent Clp endopeptidase, proteolytic subunit ClpP domain-containing protein	0.0092	0.1347	0.0504
Brugia malayi	Low molecular weight phosphotyrosine protein phosphatase containing protein	0.0185	0.3689	0.3222
Brugia malayi	Probable ClpP-like protease	0.0092	0.1347	0.0707
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Plasmodium falciparum	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.0788
Echinococcus multilocularis	Glutaredoxin protein 5	0.0136	0.2467	0.9097
Entamoeba histolytica	protein kinase 2, putative	0.0138	0.2505	0.4825
Echinococcus multilocularis	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Echinococcus granulosus	Protein kinase C brain isozyme	0.0071	0.0833	0.3071
Echinococcus multilocularis	diuretic hormone 44 receptor GPRdih2	0.0138	0.2517	0.9281
Echinococcus granulosus	calcium:calmodulin dependent protein kinase	0.0138	0.2505	0.9239
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Trypanosoma brucei	isocitrate dehydrogenase [NADP], mitochondrial precursor, putative	0.0085	0.1193	0.1791
Loa Loa (eye worm)	AGC/NDR protein kinase	0.0071	0.0833	0.0154
Echinococcus granulosus	Ataxin 2 N terminaldomain containing protein	0.0073	0.0889	0.3278
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Echinococcus multilocularis	serine:threonine protein kinase N2	0.0071	0.0833	0.3071
Echinococcus granulosus	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Echinococcus multilocularis	serine threonine protein kinase	0.0071	0.0833	0.3071
Mycobacterium tuberculosis	Probable isocitrate dehydrogenase [NADP] Icd1 (oxalosuccinate decarboxylase) (IDH) (NADP+-specific ICDH) (IDP)	0.0085	0.1193	0.3737
Echinococcus granulosus	protein kinase C gamma type	0.0071	0.0833	0.3071
Loa Loa (eye worm)	hypothetical protein	0.0163	0.3146	0.2639
Echinococcus granulosus	NDR protein kinase	0.0071	0.0833	0.3071
Echinococcus granulosus	sodium:potassium dependent atpase beta subunit	0.0136	0.2467	0.9097
Trichomonas vaginalis	serine/threonine-protein kinase sgk, putative	0.007	0.0794	0.0786
Entamoeba histolytica	protein tyrosine phosphatase, putative	0.0185	0.3689	0.7971
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Schistosoma mansoni	serine/threonine-protein kinase	0.0146	0.2712	0.3459
Mycobacterium tuberculosis	Phosphotyrosine protein phosphatase PtpA (protein-tyrosine-phosphatase) (PTPase) (LMW phosphatase)	0.0128	0.226	1
Echinococcus multilocularis	nervana 2	0.0136	0.2467	0.9097
Brugia malayi	Isocitrate dehydrogenase	0.0085	0.1193	0.0541
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Echinococcus multilocularis	ribosomal protein s6 kinase beta 1	0.0071	0.0833	0.3071
Plasmodium vivax	ataxin-2 like protein, putative	0.0163	0.3146	1
Chlamydia trachomatis	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Trypanosoma cruzi	tyrosyl-DNA Phosphodiesterase (Tdp1), putative	0.0065	0.0689	0.0777

Activities

Activity type	Activity value	Assay description	Source	Reference
Ki (binding)	= 300 nM	In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.	ChEMBL.	10882361
Ki (binding)	= 300 nM	In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.	ChEMBL.	10882361

Phenotypes

Whole-cell/tissue/organism interactions

We have no records of whole-cell/tissue assays done with this compound What does this mean?

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

No external resources registered for this compound

Bibliographic References

1 literature reference was collected for this gene.

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Detailed information for compound 379514