TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 1032.2 | Formula: C53H69N13O9
H donors: 12 H acceptors: 10 LogP: 2.5 Rotable bonds: 35
Rule of 5 violations (Lipinski): 3
SMILES: CC(C[C@@H](C(=O)N[C@H](C(=O)N)CC(C)C)NC(=O)[C@@H](NC(=O)c1cccc(c1)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)N)CCC(=O)N)C)Cc1nc[nH]c1)C
InChi: 1S/C53H69N13O9/c1-29(2)20-41(46(56)68)63-52(74)42(21-30(3)4)65-53(75)44(25-36-27-57-28-59-36)64-48(70)33-14-11-15-35(23-33)61-47(69)31(5)60-51(73)43(24-34-26-58-39-17-10-9-16-37(34)39)66-50(72)40(18-19-45(55)67)62-49(71)38(54)22-32-12-7-6-8-13-32/h6-17,23,26-31,38,40-44,58H,18-22,24-25,54H2,1-5H3,(H2,55,67)(H2,56,68)(H,57,59)(H,60,73)(H,61,69)(H,62,71)(H,63,74)(H,64,70)(H,65,75)(H,66,72)/t31-,38-,40-,41-,42-,43-,44-/m0/s1
InChiKey: ZARTZEIYNBUNPR-USXQZJOHSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

Species	Target name	Source	Bibliographic reference
Rattus norvegicus	Gastrin releasing peptide receptor	Starlite/ChEMBL	References

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

Species	Potential target	Known druggable target	Length	Alignment span	Identity
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	377 aa	22.0 %
Onchocerca volvulus	Mitochondrial inner membrane protein homolog	Gastrin releasing peptide receptor	384 aa	370 aa	21.9 %
Schistosoma mansoni	biogenic amine (octopamine/dopamine) receptor	Gastrin releasing peptide receptor	384 aa	358 aa	22.9 %
Echinococcus granulosus	pyroglutamylated rfamide peptide receptor	Gastrin releasing peptide receptor	384 aa	385 aa	21.0 %
Schistosoma japonicum	ko:K04209 neuropeptide Y receptor, invertebrate, putative	Gastrin releasing peptide receptor	384 aa	327 aa	27.8 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	333 aa	25.2 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	330 aa	26.4 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	324 aa	24.4 %
Echinococcus multilocularis	allatostatin A receptor	Gastrin releasing peptide receptor	384 aa	375 aa	27.2 %
Echinococcus multilocularis	pyroglutamylated rfamide peptide receptor	Gastrin releasing peptide receptor	384 aa	386 aa	19.9 %
Echinococcus multilocularis	neuropeptide receptor	Gastrin releasing peptide receptor	384 aa	316 aa	26.3 %
Schistosoma japonicum	ko:K04135 adrenergic receptor, alpha 1a, putative	Gastrin releasing peptide receptor	384 aa	398 aa	23.6 %
Echinococcus granulosus	neuropeptide receptor	Gastrin releasing peptide receptor	384 aa	316 aa	26.6 %
Schistosoma mansoni	peptide (allatostatin)-like receptor	Gastrin releasing peptide receptor	384 aa	315 aa	27.3 %
Schistosoma mansoni	biogenic amine (5HT) receptor	Gastrin releasing peptide receptor	384 aa	399 aa	23.6 %
Echinococcus granulosus	allatostatin A receptor	Gastrin releasing peptide receptor	384 aa	349 aa	27.2 %
Brugia malayi	ORL1-like opioid receptor	Gastrin releasing peptide receptor	384 aa	354 aa	22.3 %
Echinococcus multilocularis	thyrotropin releasing hormone receptor	Gastrin releasing peptide receptor	384 aa	385 aa	25.2 %
Echinococcus granulosus	thyrotropin releasing hormone receptor	Gastrin releasing peptide receptor	384 aa	385 aa	25.2 %
Schistosoma japonicum	ko:K04134 cholinergic receptor, invertebrate, putative	Gastrin releasing peptide receptor	384 aa	329 aa	23.1 %
Onchocerca volvulus		Gastrin releasing peptide receptor	384 aa	314 aa	22.0 %
Schistosoma japonicum	Rhodopsin, putative	Gastrin releasing peptide receptor	384 aa	327 aa	21.7 %

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Trichomonas vaginalis	AGC family protein kinase	0.0079	0.1039	0.1403
Echinococcus multilocularis	diuretic hormone 44 receptor GPRdih2	0.0138	0.2517	0.9281
Echinococcus multilocularis	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Trichomonas vaginalis	low molecular weight protein-tyrosine-phosphatase, putative	0.0185	0.3689	0.8077
Trypanosoma cruzi	rac serine-threonine kinase, putative	0.0138	0.2505	0.7594
Toxoplasma gondii	AGC kinase	0.0207	0.4247	1
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Echinococcus granulosus	nervana 2	0.0136	0.2467	0.9097
Loa Loa (eye worm)	hypothetical protein	0.0437	1	1
Schistosoma mansoni	serine/threonine-protein kinase	0.0146	0.2712	0.3459
Echinococcus multilocularis	serine threonine protein kinase	0.0071	0.0833	0.3071
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Mycobacterium ulcerans	phosphotyrosine protein phosphatase PtpA	0.0185	0.3689	1
Schistosoma mansoni	serine/threonine-protein kinase	0.0146	0.2712	0.3459
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Echinococcus granulosus	nervana 2	0.0136	0.2467	0.9097
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Echinococcus multilocularis	rac serine:threonine kinase	0.0146	0.2712	1
Schistosoma mansoni	hypothetical protein	0.0073	0.0889	0.0341
Brugia malayi	Protein kinase domain containing protein	0.0216	0.4453	0.4042
Mycobacterium tuberculosis	Phosphotyrosine protein phosphatase PtpA (protein-tyrosine-phosphatase) (PTPase) (LMW phosphatase)	0.0128	0.226	1
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Echinococcus multilocularis	peptidase Clp (S14 family)	0.006	0.0557	0.2053
Echinococcus granulosus	Glutaredoxin protein 5	0.0136	0.2467	0.9097
Brugia malayi	hypothetical protein	0.0163	0.3146	0.2639
Loa Loa (eye worm)	pax transcription factor protein 2	0.0259	0.553	0.5199
Echinococcus multilocularis	nervana 2	0.0136	0.2467	0.9097
Plasmodium vivax	ATP-dependent Clp protease proteolytic subunit, putative	0.0092	0.1347	0.0788
Echinococcus granulosus	Ataxin 2 N terminaldomain containing protein	0.0073	0.0889	0.3278
Echinococcus granulosus	protein kinase c iota type	0.0071	0.0833	0.3071
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Trypanosoma cruzi	PAB1-binding protein , putative	0.0163	0.3146	1
Trypanosoma cruzi	isocitrate dehydrogenase, putative	0.0085	0.1193	0.267
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Mycobacterium tuberculosis	Probable isocitrate dehydrogenase [NADP] Icd1 (oxalosuccinate decarboxylase) (IDH) (NADP+-specific ICDH) (IDP)	0.0085	0.1193	0.3737
Loa Loa (eye worm)	isocitrate dehydrogenase	0.0085	0.1193	0.0541
Trichomonas vaginalis	AGC family protein kinase	0.0071	0.0833	0.0883
Echinococcus granulosus	GPCR family 2	0.0138	0.2517	0.9281
Trypanosoma cruzi	rac serine-threonine kinase, putative	0.0146	0.2712	0.8369
Plasmodium vivax	rac-beta serine/threonine protein kinase, putative	0.0138	0.2505	0.6718
Echinococcus multilocularis	Glutaredoxin protein 5	0.0136	0.2467	0.9097
Leishmania major	tyrosyl-DNA phosphodiesterase 1	0.0065	0.0689	0.0777
Trichomonas vaginalis	serine/threonine-protein kinase sgk, putative	0.007	0.0794	0.0786
Brugia malayi	Hr1 repeat family protein	0.0071	0.0833	0.0154
Echinococcus granulosus	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Loa Loa (eye worm)	AGC/DMPK/GEK protein kinase	0.0071	0.0833	0.0154
Echinococcus multilocularis	serine:threonine protein kinase N2	0.0071	0.0833	0.3071
Echinococcus multilocularis	isocitrate dehydrogenase 2 (NADP+)	0.0085	0.1193	0.4401
Echinococcus multilocularis	ribosomal protein s6 kinase beta 1	0.0071	0.0833	0.3071
Trypanosoma brucei	isocitrate dehydrogenase [NADP], mitochondrial precursor, putative	0.0085	0.1193	0.1791
Echinococcus multilocularis	Ataxin 2, N terminal,domain containing protein	0.0073	0.0889	0.3278
Schistosoma mansoni	hypothetical protein	0.0299	0.6536	1
Echinococcus multilocularis	nervana 2	0.0136	0.2467	0.9097
Echinococcus granulosus	ATP dependent Clp protease proteolytic subunit	0.0092	0.1347	0.4969
Trichomonas vaginalis	AGC family protein kinase	0.0071	0.0833	0.0883
Brugia malayi	protein kinase C II.	0.0071	0.0833	0.0154
Chlamydia trachomatis	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Trichomonas vaginalis	low molecular weight protein-tyrosine-phosphatase, putative	0.0185	0.3689	0.8077
Brugia malayi	Calcitonin receptor-like protein seb-1	0.0437	1	1
Loa Loa (eye worm)	phosphotyrosine protein phosphatase	0.0185	0.3689	0.3222
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Echinococcus granulosus	ribosomal protein S6 kinase alpha 3	0.0071	0.0833	0.3071
Entamoeba histolytica	protein kinase 2, putative	0.0138	0.2505	0.4825
Trichomonas vaginalis	low molecular weight protein-tyrosine-phosphatase, putative	0.0185	0.3689	0.8077
Entamoeba histolytica	PH domain containing protein kinase, putative	0.0146	0.2712	0.5373
Treponema pallidum	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Echinococcus granulosus	serine threonine protein kinase nrc	0.0138	0.2505	0.9239
Brugia malayi	Latrophilin receptor protein 2	0.0138	0.2517	0.1963
Plasmodium falciparum	ataxin-2 like protein, putative	0.0163	0.3146	1
Echinococcus granulosus	Protein kinase C brain isozyme	0.0071	0.0833	0.3071
Echinococcus granulosus	calcium:calmodulin dependent protein kinase	0.0138	0.2505	0.9239
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Trichomonas vaginalis	low molecular weight protein tyrosine phosphatase, putative	0.0185	0.3689	0.8077
Echinococcus multilocularis	ATP dependent Clp protease proteolytic subunit	0.0092	0.1347	0.4969
Echinococcus multilocularis	isocitrate dehydrogenase	0.0085	0.1193	0.4401
Loa Loa (eye worm)	hypothetical protein	0.0092	0.1347	0.0707
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Loa Loa (eye worm)	AGC/PKN protein kinase	0.0071	0.0833	0.0154
Echinococcus multilocularis	tyrosyl DNA phosphodiesterase 1	0.0065	0.0689	0.2541
Entamoeba histolytica	protein tyrosine phosphatase, putative	0.0185	0.3689	0.7971
Trypanosoma cruzi	tyrosyl-DNA Phosphodiesterase (Tdp1), putative	0.0065	0.0689	0.0777
Trypanosoma cruzi	tyrosyl-DNA Phosphodiesterase (Tdp1), putative	0.0065	0.0689	0.0777
Loa Loa (eye worm)	AGC/NDR protein kinase	0.0071	0.0833	0.0154
Echinococcus multilocularis	serine threonine protein kinase nrc serine threonine protein kinase gad	0.0138	0.2505	0.9239
Trichomonas vaginalis	AGC family protein kinase	0.0071	0.0833	0.0883
Loa Loa (eye worm)	hypothetical protein	0.0071	0.0833	0.0154
Wolbachia endosymbiont of Brugia malayi	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Toxoplasma gondii	ATP-dependent Clp endopeptidase, proteolytic subunit ClpP domain-containing protein	0.0092	0.1347	0.0504
Brugia malayi	latrophilin 2 splice variant baaae	0.0299	0.6536	0.628
Loa Loa (eye worm)	hypothetical protein	0.0299	0.6536	0.628
Toxoplasma gondii	LsmAD domain-containing protein	0.0163	0.3146	0.6395
Echinococcus multilocularis	Ribosomal protein S6 kinase beta 2	0.0071	0.0833	0.3071
Echinococcus multilocularis	serine:threonine protein kinase N2	0.0071	0.0833	0.3071
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Echinococcus multilocularis	serine:threonine protein kinase 38	0.0071	0.0833	0.3071
Echinococcus multilocularis	Protein kinase C, brain isozyme	0.0071	0.0833	0.3071
Loa Loa (eye worm)	latrophilin receptor protein 2	0.0138	0.2517	0.1963
Loa Loa (eye worm)	pigment dispersing factor receptor c	0.0437	1	1
Brugia malayi	Protein kinase domain containing protein	0.0071	0.0833	0.0154
Entamoeba histolytica	PH domain containing protein kinase, putative	0.0146	0.2712	0.5373
Entamoeba histolytica	protein kinase, putative	0.0071	0.0833	0.0381
Brugia malayi	isocitrate dehydrogenase	0.0085	0.1193	0.0541
Echinococcus granulosus	ribosomal protein s6 kinase beta 1	0.0071	0.0833	0.3071
Echinococcus granulosus	cadherin EGF LAG seven pass G type receptor	0.0138	0.2517	0.9281
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Echinococcus multilocularis	protein kinase c epsilon type	0.0071	0.0833	0.3071
Loa Loa (eye worm)	AGC/RSK/P70 protein kinase	0.0207	0.4247	0.3821
Echinococcus multilocularis	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Brugia malayi	Isocitrate dehydrogenase	0.0085	0.1193	0.0541
Trichomonas vaginalis	low molecular weight protein tyrosine phosphatase, putative	0.0185	0.3689	0.8077
Schistosoma mansoni	NADP-specific isocitrate dehydrogenase	0.0085	0.1193	0.0862
Brugia malayi	p70 ribosomal S6 kinase beta	0.0207	0.4247	0.3821
Echinococcus granulosus	serine:threonine protein kinase N2	0.0071	0.0833	0.3071
Trypanosoma brucei	isocitrate dehydrogenase, putative	0.0085	0.1193	0.1791
Entamoeba histolytica	protein kinase, putative	0.0207	0.4247	0.9452
Echinococcus multilocularis	NADP dependent isocitrate dehydrogenase	0.0085	0.1193	0.4401
Echinococcus granulosus	diuretic hormone 44 receptor GPRdih2	0.0138	0.2517	0.9281
Trypanosoma brucei	rac serine-threonine kinase, putative	0.0216	0.4453	1
Schistosoma mansoni	peptidase Clp (S14 family)	0.0092	0.1347	0.1126
Echinococcus multilocularis	protein kinase c iota type	0.0071	0.0833	0.3071
Brugia malayi	calcium-independent alpha-latrotoxin receptor 2, putative	0.0138	0.2517	0.1963
Schistosoma mansoni	atypical protein kinase C	0.0071	0.0833	0.0246
Trichomonas vaginalis	low molecular weight protein tyrosine phosphatase, putative	0.0185	0.3689	0.8077
Trypanosoma brucei	PAB1-binding protein , putative	0.0163	0.3146	0.6709
Mycobacterium leprae	PROBABLE ATP-DEPENDENT CLP PROTEASE PROTEOLYTIC SUBUNIT 2 CLPP2 (ENDOPEPTIDASE CLP 2)	0.0092	0.1347	1
Brugia malayi	Pax transcription factor protein 2	0.0259	0.553	0.5199
Loa Loa (eye worm)	AGC/PKC/ETA protein kinase	0.0071	0.0833	0.0154
Trypanosoma cruzi	PAB1-binding protein , putative	0.0163	0.3146	1
Entamoeba histolytica	protein kinase, putative	0.0216	0.4453	1
Loa Loa (eye worm)	AGC/RSK/MSK protein kinase	0.0071	0.0833	0.0154
Leishmania major	isocitrate dehydrogenase [NADP], mitochondrial precursor, putative	0.0085	0.1193	0.267
Echinococcus multilocularis	sodium:potassium dependent atpase beta subunit	0.0136	0.2467	0.9097
Echinococcus granulosus	tyrosyl DNA phosphodiesterase 1	0.0065	0.0689	0.2541
Schistosoma mansoni	serine/threonine kinase	0.0071	0.0833	0.0246
Echinococcus multilocularis	GPCR, family 2	0.0138	0.2517	0.9281
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Entamoeba histolytica	protein kinase, putative	0.0216	0.4453	1
Echinococcus granulosus	peptidase Clp S14 family	0.006	0.0557	0.2053
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Chlamydia trachomatis	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.5
Echinococcus multilocularis	cadherin EGF LAG seven pass G type receptor	0.0138	0.2517	0.9281
Plasmodium falciparum	RAC-beta serine/threonine protein kinase	0.0138	0.2505	0.6718
Brugia malayi	Low molecular weight phosphotyrosine protein phosphatase containing protein	0.0185	0.3689	0.3222
Entamoeba histolytica	protein tyrosine phosphatase, putative	0.0185	0.3689	0.7971
Plasmodium vivax	ataxin-2 like protein, putative	0.0163	0.3146	1
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125
Echinococcus granulosus	Ribosomal protein S6 kinase beta 2	0.0071	0.0833	0.3071
Loa Loa (eye worm)	hypothetical protein	0.0138	0.2517	0.1963
Trypanosoma brucei	tyrosyl-DNA Phosphodiesterase (Tdp1), putative	0.0065	0.0689	0.0521
Echinococcus granulosus	sodium:potassium dependent atpase beta subunit	0.0136	0.2467	0.9097
Brugia malayi	hypothetical protein	0.0105	0.1695	0.1081
Trypanosoma cruzi	Protein kinase B	0.0146	0.2712	0.8369
Onchocerca volvulus		0.0259	0.553	1
Trichomonas vaginalis	AGC family protein kinase	0.0216	0.4453	1
Echinococcus granulosus	serine/threonine protein kinase	0.0146	0.2712	1
Echinococcus granulosus	NDR protein kinase	0.0071	0.0833	0.3071
Plasmodium falciparum	ATP-dependent Clp protease proteolytic subunit	0.0092	0.1347	0.0788
Giardia lamblia	Low molecular weight protein-tyrosine-phosphatase	0.0185	0.3689	1
Echinococcus granulosus	protein kinase C gamma type	0.0071	0.0833	0.3071
Toxoplasma gondii	ATP-dependent Clp endopeptidase, proteolytic subunit ClpP domain-containing protein	0.0092	0.1347	0.0504
Plasmodium falciparum	ataxin-2 like protein, putative	0.0163	0.3146	1
Brugia malayi	Protein kinase domain containing protein	0.0071	0.0833	0.0154
Brugia malayi	Probable ClpP-like protease	0.0092	0.1347	0.0707
Echinococcus multilocularis	ribosomal protein S6 kinase alpha 3	0.0071	0.0833	0.3071
Loa Loa (eye worm)	hypothetical protein	0.0163	0.3146	0.2639
Loa Loa (eye worm)	AGC/AKT protein kinase	0.0216	0.4453	0.4042
Schistosoma mansoni	serine/threonine protein kinase	0.0071	0.0833	0.0246
Trypanosoma cruzi	isocitrate dehydrogenase [NADP], mitochondrial precursor, putative	0.0085	0.1193	0.267
Echinococcus granulosus	protein kinase c epsilon type	0.0071	0.0833	0.3071
Leishmania major	hypothetical protein, conserved	0.0163	0.3146	1
Loa Loa (eye worm)	AGC/RSK/RSK protein kinase	0.0071	0.0833	0.0154
Schistosoma mansoni	hypothetical protein	0.0138	0.2517	0.3125

Activities

Activity type	Activity value	Assay description	Source	Reference
Ki (binding)	= 300 nM	In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.	ChEMBL.	10882361
Ki (binding)	= 300 nM	In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.	ChEMBL.	10882361

Phenotypes

Whole-cell/tissue/organism interactions

We have no records of whole-cell/tissue assays done with this compound What does this mean?

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

No external resources registered for this compound

Bibliographic References

1 literature reference was collected for this gene.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 379514