Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Mycobacterium ulcerans | heat shock protein 90 | 0.003 | 0.0494 | 0.0295 |
Loa Loa (eye worm) | hypothetical protein | 0.0117 | 0.3358 | 0.3358 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.0038 | 0.0749 | 1 |
Echinococcus multilocularis | musashi | 0.0031 | 0.0536 | 0.0624 |
Wolbachia endosymbiont of Brugia malayi | heat shock protein 90 | 0.003 | 0.0494 | 0.5 |
Echinococcus granulosus | family S9 non peptidase ue S09 family | 0.0021 | 0.0205 | 0.0239 |
Trichomonas vaginalis | carboxylesterase domain containing protein, putative | 0.0021 | 0.0205 | 0.0194 |
Echinococcus multilocularis | BC026374 protein (S09 family) | 0.0021 | 0.0205 | 0.0239 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Trichomonas vaginalis | heat shock protein, putative | 0.003 | 0.0494 | 0.0483 |
Loa Loa (eye worm) | heat shock protein 75 | 0.0015 | 0.0012 | 0.0012 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Brugia malayi | hypothetical protein | 0.002 | 0.0151 | 0.014 |
Brugia malayi | Carboxylesterase family protein | 0.0126 | 0.3673 | 0.3666 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Trichomonas vaginalis | set domain proteins, putative | 0.0276 | 0.8599 | 0.8597 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Trichomonas vaginalis | endoplasmin, putative | 0.0023 | 0.0266 | 0.0255 |
Schistosoma mansoni | histone-lysine n-methyltransferase setb1 | 0.0035 | 0.0647 | 0.0636 |
Schistosoma mansoni | histone-lysine n-methyltransferase setb1 | 0.0035 | 0.0647 | 0.0636 |
Trypanosoma cruzi | heat shock protein 90, putative | 0.0038 | 0.0749 | 1 |
Echinococcus granulosus | histone lysine methyltransferase setb | 0.0035 | 0.0647 | 0.0753 |
Brugia malayi | RNA binding protein | 0.0074 | 0.1933 | 0.1924 |
Mycobacterium tuberculosis | Probable chaperone protein HtpG (heat shock protein) (HSP90 family protein) (high temperature protein G) | 0.003 | 0.0494 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0126 | 0.3673 | 0.3673 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Brugia malayi | Pre-SET motif family protein | 0.0242 | 0.7494 | 0.7491 |
Schistosoma mansoni | glutaminase | 0.0318 | 1 | 1 |
Echinococcus multilocularis | tar DNA binding protein | 0.0074 | 0.1933 | 0.2252 |
Echinococcus multilocularis | neuroligin | 0.0021 | 0.0205 | 0.0239 |
Onchocerca volvulus | 0.0021 | 0.0205 | 0.0225 | |
Echinococcus multilocularis | histone lysine methyltransferase setb histone lysine methyltransferase eggless | 0.0035 | 0.0647 | 0.0753 |
Schistosoma mansoni | histone-lysine n-methyltransferase suv9 | 0.0035 | 0.0647 | 0.0636 |
Onchocerca volvulus | 0.0031 | 0.0536 | 0.0611 | |
Brugia malayi | Iron-sulfur cluster assembly accessory protein | 0.0056 | 0.1353 | 0.1343 |
Brugia malayi | Carboxylesterase family protein | 0.0021 | 0.0205 | 0.0194 |
Toxoplasma gondii | LsmAD domain-containing protein | 0.002 | 0.0151 | 0.1892 |
Brugia malayi | cytoplasmic intermediate filament protein | 0.0017 | 0.0055 | 0.0043 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Loa Loa (eye worm) | follicle stimulating hormone receptor | 0.0181 | 0.5482 | 0.5482 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | heat shock protein | 0.0038 | 0.0749 | 0.0738 |
Toxoplasma gondii | heat shock protein HSP90 | 0.0038 | 0.0749 | 1 |
Onchocerca volvulus | 0.0035 | 0.0647 | 0.074 | |
Schistosoma mansoni | lamin | 0.0031 | 0.0536 | 0.0525 |
Loa Loa (eye worm) | hypothetical protein | 0.0031 | 0.0517 | 0.0517 |
Entamoeba histolytica | heat shock protein 90, putative | 0.0038 | 0.0749 | 1 |
Plasmodium falciparum | heat shock protein 90 | 0.0038 | 0.0749 | 1 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | endoplasmin | 0.0038 | 0.0749 | 0.0738 |
Brugia malayi | intermediate filament protein | 0.0031 | 0.0536 | 0.0525 |
Plasmodium falciparum | endoplasmin, putative | 0.0023 | 0.0266 | 0.345 |
Plasmodium falciparum | ataxin-2 like protein, putative | 0.002 | 0.0151 | 0.1892 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 0.1933 | 0.1924 |
Plasmodium vivax | SET domain protein, putative | 0.0035 | 0.0647 | 0.8618 |
Echinococcus granulosus | para nitrobenzyl esterase | 0.0021 | 0.0205 | 0.0239 |
Echinococcus multilocularis | muscleblind protein 1 | 0.0117 | 0.3358 | 0.3913 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Loa Loa (eye worm) | RNA recognition domain-containing protein domain-containing protein | 0.0074 | 0.1933 | 0.1933 |
Loa Loa (eye worm) | hypothetical protein | 0.0031 | 0.0536 | 0.0536 |
Brugia malayi | Carboxylesterase family protein | 0.0021 | 0.0205 | 0.0194 |
Brugia malayi | hypothetical protein | 0.0275 | 0.8583 | 0.8581 |
Trypanosoma cruzi | heat shock protein 90, putative | 0.0022 | 0.0237 | 0.3058 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 0.1933 | 0.1924 |
Trichomonas vaginalis | heat shock protein, putative | 0.003 | 0.0494 | 0.0483 |
Echinococcus granulosus | neuroligin | 0.0021 | 0.0205 | 0.0239 |
Echinococcus multilocularis | lamin dm0 | 0.0031 | 0.0536 | 0.0624 |
Echinococcus granulosus | heat shock protein heat shock protein 90 alpha | 0.003 | 0.0494 | 0.0576 |
Echinococcus granulosus | tar DNA binding protein | 0.0074 | 0.1933 | 0.2252 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Plasmodium vivax | heat shock protein 86, putative | 0.0038 | 0.0749 | 1 |
Entamoeba histolytica | heat shock protein 90, putative | 0.0038 | 0.0749 | 1 |
Echinococcus granulosus | lamin dm0 | 0.0031 | 0.0536 | 0.0624 |
Trypanosoma brucei | heat shock protein 90, putative | 0.0038 | 0.0749 | 1 |
Echinococcus granulosus | endoplasmin | 0.003 | 0.0494 | 0.0576 |
Schistosoma mansoni | family S9 non-peptidase homologue (S09 family) | 0.0021 | 0.0205 | 0.0194 |
Trypanosoma cruzi | PAB1-binding protein , putative | 0.002 | 0.0151 | 0.1892 |
Loa Loa (eye worm) | hypothetical protein | 0.0126 | 0.3673 | 0.3673 |
Echinococcus multilocularis | endoplasmin | 0.003 | 0.0494 | 0.0576 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Echinococcus granulosus | muscleblind protein | 0.0117 | 0.3358 | 0.3913 |
Trypanosoma brucei | heat shock protein 90, putative | 0.0038 | 0.0749 | 1 |
Mycobacterium leprae | PROBABLE CHAPERONE PROTEIN HTPG (HEAT SHOCK PROTEIN) (HSP90 FAMILY PROTEIN) (HIGH TEMPERATURE PROTEIN G) | 0.003 | 0.0494 | 0.5 |
Schistosoma mansoni | family S9 non-peptidase homologue (S09 family) | 0.0021 | 0.0205 | 0.0194 |
Loa Loa (eye worm) | carboxylesterase | 0.0021 | 0.0205 | 0.0205 |
Schistosoma mansoni | family S9 non-peptidase homologue (S09 family) | 0.0126 | 0.3673 | 0.3666 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | histone-lysine n-methyltransferase setb1 | 0.0035 | 0.0647 | 0.0636 |
Loa Loa (eye worm) | hypothetical protein | 0.0275 | 0.8583 | 0.8583 |
Onchocerca volvulus | 0.0021 | 0.0205 | 0.0225 | |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Plasmodium vivax | endoplasmin, putative | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | acetylcholinesterase | 0.0021 | 0.0205 | 0.0194 |
Loa Loa (eye worm) | hypothetical protein | 0.0117 | 0.3358 | 0.3358 |
Echinococcus multilocularis | family S9 non peptidase ue (S09 family) | 0.0021 | 0.0205 | 0.0239 |
Echinococcus granulosus | lamin | 0.0031 | 0.0536 | 0.0624 |
Brugia malayi | Carboxylesterase family protein | 0.0021 | 0.0205 | 0.0194 |
Leishmania major | lipophosphoglycan biosynthetic protein, putative,heat shock protein 90, putative,glucose regulated protein 94, putative | 0.003 | 0.0494 | 0.655 |
Toxoplasma gondii | heat shock protein 90, putative | 0.0038 | 0.0749 | 1 |
Echinococcus multilocularis | heat shock protein | 0.0038 | 0.0749 | 0.0872 |
Trypanosoma cruzi | PAB1-binding protein , putative | 0.002 | 0.0151 | 0.1892 |
Echinococcus multilocularis | heat shock protein 90 | 0.0038 | 0.0749 | 0.0872 |
Echinococcus multilocularis | heat shock protein 75 kDa, mitochondrial | 0.0015 | 0.0012 | 0.0014 |
Giardia lamblia | Heat shock protein HSP 90-alpha | 0.0038 | 0.0749 | 1 |
Loa Loa (eye worm) | TAR-binding protein | 0.0074 | 0.1933 | 0.1933 |
Echinococcus granulosus | BC026374 protein S09 family | 0.0021 | 0.0205 | 0.0239 |
Brugia malayi | heat shock protein 90 | 0.0038 | 0.0749 | 0.0738 |
Loa Loa (eye worm) | hypothetical protein | 0.002 | 0.0151 | 0.0151 |
Echinococcus multilocularis | histone lysine N methyltransferase SETMAR | 0.0035 | 0.0647 | 0.0753 |
Brugia malayi | Carboxylesterase family protein | 0.0021 | 0.0205 | 0.0194 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 0.1933 | 0.1924 |
Onchocerca volvulus | 0.0031 | 0.0536 | 0.0611 | |
Trypanosoma cruzi | heat shock protein 85, putative | 0.003 | 0.0494 | 0.655 |
Echinococcus granulosus | heat shock protein 90 | 0.003 | 0.0494 | 0.0576 |
Loa Loa (eye worm) | heat shock protein 90 | 0.0038 | 0.0749 | 0.0749 |
Brugia malayi | glutaminase DH11.1 | 0.0318 | 1 | 1 |
Echinococcus multilocularis | muscleblind protein | 0.0117 | 0.3358 | 0.3913 |
Echinococcus multilocularis | acetylcholinesterase | 0.0126 | 0.3673 | 0.428 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | neuroligin 3 (S09 family) | 0.0021 | 0.0205 | 0.0194 |
Mycobacterium ulcerans | glutaminase | 0.0318 | 1 | 1 |
Brugia malayi | RNA recognition motif domain containing protein | 0.0074 | 0.1933 | 0.1924 |
Loa Loa (eye worm) | RNA binding protein | 0.0074 | 0.1933 | 0.1933 |
Echinococcus granulosus | carboxylesterase 5A | 0.0126 | 0.3673 | 0.428 |
Schistosoma mansoni | heat shock protein | 0.0038 | 0.0749 | 0.0738 |
Schistosoma mansoni | family S9 non-peptidase homologue (S09 family) | 0.0021 | 0.0205 | 0.0194 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.0038 | 0.0749 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Loa Loa (eye worm) | carboxylesterase | 0.0021 | 0.0205 | 0.0205 |
Loa Loa (eye worm) | intermediate filament protein | 0.0031 | 0.0536 | 0.0536 |
Schistosoma mansoni | hypothetical protein | 0.0056 | 0.1353 | 0.1343 |
Treponema pallidum | heat shock protein 90 | 0.003 | 0.0494 | 0.5 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | BC026374 protein (S09 family) | 0.0021 | 0.0205 | 0.0194 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Trichomonas vaginalis | glutaminase, putative | 0.0318 | 1 | 1 |
Echinococcus granulosus | intermediate filament protein | 0.0031 | 0.0536 | 0.0624 |
Trypanosoma cruzi | heat shock protein 90, putative | 0.003 | 0.0494 | 0.655 |
Trichomonas vaginalis | spcc417.12 protein, putative | 0.0021 | 0.0205 | 0.0194 |
Trypanosoma cruzi | Heat shock protein 83, putative | 0.0038 | 0.0749 | 1 |
Schistosoma mansoni | endoplasmin | 0.0038 | 0.0749 | 0.0738 |
Onchocerca volvulus | 0.0276 | 0.8599 | 1 | |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 0.1933 | 0.1924 |
Onchocerca volvulus | 0.0021 | 0.0205 | 0.0225 | |
Trichomonas vaginalis | heat shock protein, putative | 0.003 | 0.0494 | 0.0483 |
Loa Loa (eye worm) | carboxylesterase | 0.0126 | 0.3673 | 0.3673 |
Trypanosoma cruzi | heat shock protein 85, putative | 0.0038 | 0.0749 | 1 |
Trichomonas vaginalis | heat shock protein, putative | 0.0038 | 0.0749 | 0.0738 |
Schistosoma mansoni | intermediate filament proteins | 0.0031 | 0.0536 | 0.0525 |
Echinococcus granulosus | heat shock protein 90 | 0.0038 | 0.0749 | 0.0872 |
Brugia malayi | Muscleblind-like protein | 0.0117 | 0.3358 | 0.335 |
Onchocerca volvulus | 0.0021 | 0.0205 | 0.0225 | |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.0205 | 0.0205 |
Loa Loa (eye worm) | pre-SET domain-containing protein family protein | 0.0242 | 0.7494 | 0.7494 |
Leishmania major | hypothetical protein, conserved | 0.002 | 0.0151 | 0.1892 |
Brugia malayi | Pre-SET motif family protein | 0.0035 | 0.0647 | 0.0636 |
Plasmodium vivax | ataxin-2 like protein, putative | 0.002 | 0.0151 | 0.1892 |
Echinococcus granulosus | acetylcholinesterase | 0.0126 | 0.3673 | 0.428 |
Schistosoma mansoni | tar DNA-binding protein | 0.0074 | 0.1933 | 0.1924 |
Brugia malayi | Endoplasmin precursor | 0.0038 | 0.0749 | 0.0738 |
Brugia malayi | TAR-binding protein | 0.0074 | 0.1933 | 0.1924 |
Schistosoma mansoni | survival motor neuron protein | 0.0056 | 0.1353 | 0.1343 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Echinococcus granulosus | 5'partial|histone lysine N methyltransferase SETDB2 | 0.0033 | 0.0605 | 0.0704 |
Schistosoma mansoni | gliotactin | 0.0021 | 0.0205 | 0.0194 |
Toxoplasma gondii | histone lysine methyltransferase SET/SUV39 | 0.0035 | 0.0647 | 0.8618 |
Echinococcus multilocularis | carboxylesterase 5A | 0.0126 | 0.3673 | 0.428 |
Echinococcus multilocularis | para nitrobenzyl esterase | 0.0021 | 0.0205 | 0.0239 |
Loa Loa (eye worm) | glutaminase | 0.0318 | 1 | 1 |
Trypanosoma brucei | PAB1-binding protein , putative | 0.002 | 0.0151 | 0.1892 |
Loa Loa (eye worm) | acetylcholinesterase 1 | 0.0126 | 0.3673 | 0.3673 |
Loa Loa (eye worm) | intermediate filament tail domain-containing protein | 0.0031 | 0.0536 | 0.0536 |
Echinococcus granulosus | acetylcholinesterase | 0.0126 | 0.3673 | 0.428 |
Echinococcus multilocularis | survival motor neuron protein 1 | 0.0275 | 0.8583 | 1 |
Brugia malayi | Intermediate filament tail domain containing protein | 0.0031 | 0.0536 | 0.0525 |
Echinococcus granulosus | heat shock protein | 0.0038 | 0.0749 | 0.0872 |
Onchocerca volvulus | 0.0056 | 0.1353 | 0.1562 | |
Echinococcus multilocularis | lamin | 0.0031 | 0.0536 | 0.0624 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Trichomonas vaginalis | heat shock protein, putative | 0.0023 | 0.0266 | 0.0255 |
Echinococcus granulosus | survival motor neuron protein 1 | 0.0275 | 0.8583 | 1 |
Trypanosoma brucei | heat shock protein, putative | 0.0038 | 0.0749 | 1 |
Echinococcus granulosus | heat shock protein 75 kDa mitochondrial | 0.0015 | 0.0012 | 0.0014 |
Brugia malayi | follicle stimulating hormone receptor | 0.0181 | 0.5482 | 0.5477 |
Onchocerca volvulus | 0.0021 | 0.0205 | 0.0225 | |
Loa Loa (eye worm) | cytoplasmic intermediate filament protein | 0.0017 | 0.0055 | 0.0055 |
Brugia malayi | hypothetical protein | 0.0021 | 0.0205 | 0.0194 |
Echinococcus multilocularis | heat shock protein 90 | 0.003 | 0.0494 | 0.0576 |
Trypanosoma brucei | Heat shock protein 83, putative | 0.0038 | 0.0749 | 1 |
Echinococcus multilocularis | acetylcholinesterase | 0.0126 | 0.3673 | 0.428 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Brugia malayi | Carboxylesterase family protein | 0.0126 | 0.3673 | 0.3666 |
Schistosoma mansoni | lamin | 0.0031 | 0.0536 | 0.0525 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.0647 | 0.0647 |
Loa Loa (eye worm) | endoplasmin | 0.0038 | 0.0749 | 0.0749 |
Plasmodium falciparum | ataxin-2 like protein, putative | 0.002 | 0.0151 | 0.1892 |
Leishmania major | heat shock protein 83-1 | 0.0038 | 0.0749 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Activity (binding) | 0 | Inhibition of Gypsophila oldhamiana alpha-glucosidase at 400 uM | ChEMBL. | 18194870 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.