Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Loa Loa (eye worm) | alpha-tubulin | 0.0231 | 0.5654 | 0.5528 |
Treponema pallidum | cell division protein FtsZ | 0.0079 | 0.1167 | 1 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus multilocularis | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | gamma-tubulin | 0.0182 | 0.4208 | 0.3442 |
Echinococcus granulosus | tubulin epsilon chain | 0.0182 | 0.4208 | 0.3932 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0182 | 0.4208 | 0.3442 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0152 | 0.3321 | 0.3128 |
Trypanosoma brucei | beta tubulin | 0.0378 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Brugia malayi | beta-tubulin, identical | 0.0378 | 1 | 1 |
Schistosoma mansoni | tubulin subunit gamma | 0.0182 | 0.4208 | 0.3442 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0182 | 0.4208 | 0.3442 |
Echinococcus granulosus | tubulin subunit TubB | 0.0231 | 0.5654 | 0.5447 |
Echinococcus multilocularis | tubulin alpha | 0.0182 | 0.4208 | 0.3932 |
Echinococcus granulosus | tubulin delta chain | 0.0079 | 0.1167 | 0.0746 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Echinococcus multilocularis | tubulin delta chain | 0.0079 | 0.1167 | 0.0746 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 0.5654 | 0.5079 |
Onchocerca volvulus | 0.0103 | 0.1874 | 0.5 | |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0103 | 0.1874 | 0.0801 |
Brugia malayi | Tubulin alpha-2 chain | 0.0231 | 0.5654 | 0.5079 |
Toxoplasma gondii | alpha-tubulin I, putative | 0.0231 | 0.5654 | 0.5079 |
Mycobacterium tuberculosis | Cell division protein FtsZ | 0.0079 | 0.1167 | 1 |
Giardia lamblia | Beta tubulin | 0.0378 | 1 | 1 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0103 | 0.1874 | 0.0801 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 0.5654 | 0.5079 |
Brugia malayi | tubulin alpha-2 chain | 0.0231 | 0.5654 | 0.5079 |
Schistosoma mansoni | tubulin subunit epsilon | 0.0182 | 0.4208 | 0.3442 |
Brugia malayi | tubulin alpha chain - mouse | 0.0231 | 0.5654 | 0.5079 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Mycobacterium leprae | cell division protein FtsZ | 0.0079 | 0.1167 | 0.5 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | beta-tubulin | 0.0378 | 1 | 1 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Plasmodium falciparum | tubulin gamma chain | 0.0182 | 0.4208 | 0.3442 |
Entamoeba histolytica | tubulin alpha-1 chain | 0.0231 | 0.5654 | 0.2497 |
Echinococcus granulosus | tubulin gamma 1 chain | 0.0182 | 0.4208 | 0.3932 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Echinococcus granulosus | tubulin subunit beta | 0.0378 | 1 | 1 |
Plasmodium vivax | tubulin epsilon chain, putative | 0.0182 | 0.4208 | 0.3442 |
Echinococcus multilocularis | beta tubulin | 0.0378 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0378 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 1 | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | hypothetical protein | 0.0231 | 0.5654 | 0.5447 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0182 | 0.4208 | 0.3442 |
Trypanosoma brucei | epsilon tubulin | 0.0182 | 0.4208 | 0.3442 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0378 | 1 | 1 |
Echinococcus granulosus | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Schistosoma mansoni | tubulin subunit alpha | 0.0231 | 0.5654 | 0.5079 |
Schistosoma mansoni | tubulin subunit beta | 0.0378 | 1 | 1 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0231 | 0.5654 | 0.5447 |
Entamoeba histolytica | tubulin family protein | 0.0378 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trypanosoma brucei | epsilon tubulin | 0.0182 | 0.4208 | 0.3442 |
Schistosoma mansoni | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0231 | 0.5654 | 0.5528 |
Trypanosoma brucei | tubulin gamma chain | 0.0182 | 0.4208 | 0.3442 |
Loa Loa (eye worm) | hypothetical protein | 0.0128 | 0.2613 | 0.24 |
Trypanosoma cruzi | tubulin gamma chain | 0.0182 | 0.4208 | 0.3442 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0231 | 0.5654 | 0.5447 |
Trichomonas vaginalis | tubulin, putative | 0.0103 | 0.1874 | 0.0801 |
Schistosoma mansoni | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | tubulin, beta 4A class IVa | 0.0378 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Chlamydia trachomatis | arginine ABC transporter substrate-binding protein ArtJ | 0.0039 | 0 | 0.5 |
Giardia lamblia | Gamma tubulin | 0.0182 | 0.4208 | 0.3442 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0103 | 0.1874 | 0.0801 |
Echinococcus multilocularis | tubulin subunit beta | 0.0378 | 1 | 1 |
Echinococcus granulosus | tubulin beta 4A class IVa | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin gamma chain, putative | 0.0182 | 0.4208 | 0.3442 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | BEN-1 protein | 0.0378 | 1 | 1 |
Echinococcus multilocularis | tubulin alpha 1C chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Plasmodium falciparum | tubulin beta chain | 0.0378 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trypanosoma cruzi | beta tubulin, putative | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-2A chain | 0.0378 | 1 | 1 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | peroxisome assembly protein 26 | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Brugia malayi | Tubulin gamma chain | 0.0182 | 0.4208 | 0.3442 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | beta tubulin | 0.0378 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | alpha tubulin | 0.0231 | 0.5654 | 0.5447 |
Schistosoma mansoni | tubulin subunit alpha | 0.0231 | 0.5654 | 0.5079 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0231 | 0.5654 | 0.5079 |
Entamoeba histolytica | tubulin family protein | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0128 | 0.2613 | 0.1637 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 0.5654 | 0.5079 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0231 | 0.5654 | 0.5079 |
Toxoplasma gondii | beta-1 tubulin, putative | 0.0378 | 1 | 1 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0378 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | cell division protein FtsZ | 0.0079 | 0.1167 | 0.5 |
Loa Loa (eye worm) | tubulin gamma chain | 0.0182 | 0.4208 | 0.404 |
Echinococcus multilocularis | tubulin epsilon chain | 0.0182 | 0.4208 | 0.3932 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin, putative | 0.0103 | 0.1874 | 0.0801 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0152 | 0.3321 | 0.3128 |
Plasmodium falciparum | tubulin epsilon chain, putative | 0.0182 | 0.4208 | 0.3442 |
Trypanosoma brucei | epsilon tubulin | 0.0182 | 0.4208 | 0.3442 |
Trypanosoma brucei | beta tubulin | 0.0182 | 0.4208 | 0.3442 |
Echinococcus multilocularis | peroxisome assembly protein 26 | 0.0231 | 0.5654 | 0.5447 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Schistosoma mansoni | tubulin subunit alpha | 0.0231 | 0.5654 | 0.5079 |
Trypanosoma brucei | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | tubulin subunit TubB | 0.0231 | 0.5654 | 0.5447 |
Loa Loa (eye worm) | tubulin alpha-3 chain | 0.0128 | 0.2613 | 0.24 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta chain | 0.0079 | 0.1167 | 0.0912 |
Leishmania major | epsilon tubulin, putative | 0.0182 | 0.4208 | 0.3442 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus granulosus | Tubulin beta 2C chain | 0.0378 | 1 | 1 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Giardia lamblia | Beta tubulin | 0.0378 | 1 | 1 |
Schistosoma mansoni | tubulin subunit beta | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0231 | 0.5654 | 0.5528 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Loa Loa (eye worm) | alpha-tubulin | 0.0231 | 0.5654 | 0.5528 |
Loa Loa (eye worm) | tubulin alpha chain | 0.0231 | 0.5654 | 0.5528 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | tubulin alpha 3 chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus multilocularis | beta tubulin | 0.0378 | 1 | 1 |
Echinococcus multilocularis | Tubulin alpha 1 chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin alpha-1 chain, putative | 0.0152 | 0.3321 | 0.2438 |
Toxoplasma gondii | tubulin/FtsZ family, GTPase domain-containing protein | 0.0182 | 0.4208 | 0.3442 |
Echinococcus multilocularis | tubulin gamma 1 chain | 0.0182 | 0.4208 | 0.3932 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus multilocularis | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Brugia malayi | alpha-tubulin | 0.0231 | 0.5654 | 0.5079 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trypanosoma brucei | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin epsilon chain, putative | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus granulosus | Tubulin alpha 1 chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus granulosus | tubulin alpha 1C chain | 0.0231 | 0.5654 | 0.5447 |
Trypanosoma brucei | alpha tubulin, putative | 0.0103 | 0.1874 | 0.0801 |
Trichomonas vaginalis | tubulin alpha chain, putative | 0.0103 | 0.1874 | 0.0801 |
Loa Loa (eye worm) | tubulin beta-4 chain | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | tubulin beta-1 chain | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha-2 chain | 0.0231 | 0.5654 | 0.5528 |
Loa Loa (eye worm) | tubulin beta chain | 0.0378 | 1 | 1 |
Trypanosoma cruzi | alpha tubulin, putative | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Echinococcus granulosus | tubulin beta 1 chain | 0.0378 | 1 | 1 |
Plasmodium vivax | tubulin gamma chain, putative | 0.0182 | 0.4208 | 0.3442 |
Echinococcus multilocularis | tubulin beta 1 chain | 0.0378 | 1 | 1 |
Trypanosoma cruzi | epsilon tubulin, putative | 0.0182 | 0.4208 | 0.3442 |
Mycobacterium ulcerans | cell division protein FtsZ | 0.0079 | 0.1167 | 1 |
Schistosoma mansoni | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Trypanosoma brucei | beta tubulin | 0.0378 | 1 | 1 |
Toxoplasma gondii | alpha tubulin TUBA1 | 0.0231 | 0.5654 | 0.5079 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Brugia malayi | Tubulin beta chain | 0.0103 | 0.1874 | 0.0801 |
Echinococcus multilocularis | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Schistosoma mansoni | tubulin subunit beta | 0.0378 | 1 | 1 |
Plasmodium vivax | tubulin alpha chain, putative | 0.0231 | 0.5654 | 0.5079 |
Toxoplasma gondii | beta tubulin | 0.0378 | 1 | 1 |
Echinococcus granulosus | beta tubulin | 0.0378 | 1 | 1 |
Brugia malayi | Tubulin alpha chain | 0.0231 | 0.5654 | 0.5079 |
Trypanosoma brucei | beta tubulin | 0.0378 | 1 | 1 |
Loa Loa (eye worm) | tubulin alpha 2 | 0.0152 | 0.3321 | 0.3128 |
Brugia malayi | Tubulin alpha-2 chain | 0.0231 | 0.5654 | 0.5079 |
Loa Loa (eye worm) | alpha-tubulin isotype 2 | 0.0152 | 0.3321 | 0.3128 |
Leishmania major | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0231 | 0.5654 | 0.5447 |
Leishmania major | beta tubulin | 0.0378 | 1 | 1 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0103 | 0.1874 | 0.0801 |
Echinococcus granulosus | tubulin alpha | 0.0182 | 0.4208 | 0.3932 |
Trichomonas vaginalis | tubulin beta chain, putative | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | tubulin alpha chain | 0.0231 | 0.5654 | 0.5447 |
Toxoplasma gondii | beta-tubulin, putative | 0.0378 | 1 | 1 |
Plasmodium vivax | tubulin beta chain, putative | 0.0378 | 1 | 1 |
Plasmodium falciparum | alpha tubulin 2 | 0.0231 | 0.5654 | 0.5079 |
Echinococcus granulosus | tubulin alpha 3 chain | 0.0231 | 0.5654 | 0.5447 |
Schistosoma mansoni | tubulin subunit beta | 0.0378 | 1 | 1 |
Giardia lamblia | Alpha-tubulin | 0.0231 | 0.5654 | 0.5079 |
Chlamydia trachomatis | glutamine binding protein | 0.0039 | 0 | 0.5 |
Entamoeba histolytica | tubulin alpha chain, putative | 0.0231 | 0.5654 | 0.2497 |
Trypanosoma brucei | alpha tubulin | 0.0231 | 0.5654 | 0.5079 |
Trypanosoma brucei | beta tubulin | 0.0378 | 1 | 1 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (binding) | = 0.6 nM | Homogenous Time-Resolved Fluorescence Assay (HTRF2 Assay) | BINDINGDB. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.