TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 392.372 | Formula: C20H19F3N2O3
H donors: 1 H acceptors: 2 LogP: 4.86 Rotable bonds: 9
Rule of 5 violations (Lipinski): 1
SMILES: N#CC(NC(=O)c1ccc(cc1)OC(F)(F)F)(COc1ccccc1CC)C
InChi: 1S/C20H19F3N2O3/c1-3-14-6-4-5-7-17(14)27-13-19(2,12-24)25-18(26)15-8-10-16(11-9-15)28-20(21,22)23/h4-11H,3,13H2,1-2H3,(H,25,26)
InChiKey: VMRUZVMSSYIVNY-UHFFFAOYSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

No curated genes were found associated with this compound

Predicted pathogen targets for this compound

By orthology

No druggable targets predicted by orthology data

By sequence similarity to non orthologous known druggable targets

No druggable targets predicted by sequence similarity

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Mycobacterium leprae	DIHYDROLIPOAMIDE DEHYDROGENASE LPD (LIPOAMIDE REDUCTASE (NADH)) (LIPOYL DEHYDROGENASE) (DIHYDROLIPOYL DEHYDROGENASE) (DIAPHORASE	0.0127	0.6986	1
Loa Loa (eye worm)	GTP-binding regulatory protein Gs alpha-S chain	0.0049	0.2475	0.3461
Brugia malayi	serine/threonine-protein kinase plk-2	0.01	0.5439	0.7802
Trypanosoma cruzi	dihydrolipoyl dehydrogenase, putative	0.0017	0.0689	0.1175
Trypanosoma cruzi	dihydrolipoyl dehydrogenase, putative	0.0017	0.0689	0.1175
Toxoplasma gondii	ImpB/MucB/SamB family protein	0.0006	0.0057	0.0222
Treponema pallidum	NADH oxidase	0.0017	0.0689	0.5
Plasmodium falciparum	thioredoxin reductase	0.005	0.2569	1
Plasmodium falciparum	glutathione reductase	0.0017	0.0689	0.2517
Toxoplasma gondii	BRCA1 C Terminus (BRCT) domain-containing protein	0.0006	0.0057	0.0222
Brugia malayi	MH1 domain containing protein	0.0009	0.0188	0.0189
Trichomonas vaginalis	DNA helicase recq, putative	0.0026	0.1153	0.137
Echinococcus multilocularis	dna polymerase kappa	0.0021	0.0867	0.0692
Trichomonas vaginalis	CAMK family protein kinase	0.005	0.2537	0.4157
Trypanosoma cruzi	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Brugia malayi	ATP-dependent DNA helicase, RecQ family protein	0.0011	0.0296	0.0346
Entamoeba histolytica	recQ family helicase, putative	0.0014	0.0473	0.0869
Mycobacterium tuberculosis	Probable nitrite reductase [NAD(P)H] large subunit [FAD flavoprotein] NirB	0.0115	0.6254	0.8837
Plasmodium falciparum	glutathione reductase	0.005	0.2569	1
Loa Loa (eye worm)	hypothetical protein	0.0128	0.7043	1
Schistosoma mansoni	kinase	0.0051	0.2613	0.257
Loa Loa (eye worm)	hypothetical protein	0.0048	0.2416	0.3377
Leishmania major	protein kinase, putative,polo-like protein kinase, putative	0.01	0.5439	1
Trypanosoma brucei	DNA polymerase kappa, putative	0.0014	0.0502	0.0827
Entamoeba histolytica	serine/threonine protein kinase, putative	0.01	0.5439	1
Plasmodium vivax	dihydrolipoyl dehydrogenase, mitochondrial, putative	0.0017	0.0689	0.2517
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma brucei	unspecified product	0.0014	0.0502	0.0827
Trypanosoma cruzi	DNA polymerase eta, putative	0.0033	0.1607	0.2879
Trypanosoma cruzi	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma cruzi	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Echinococcus granulosus	guanine nucleotide binding protein Gs subunit	0.0049	0.2475	0.2331
Mycobacterium tuberculosis	Dihydrolipoamide dehydrogenase LpdC (lipoamide reductase (NADH)) (lipoyl dehydrogenase) (dihydrolipoyl dehydrogenase) (diaphoras	0.0127	0.6986	1
Giardia lamblia	NADH oxidase lateral transfer candidate	0.0017	0.0689	0.1175
Trypanosoma cruzi	ATP-dependent DEAD/H DNA helicase recQ, putative	0.0014	0.0473	0.0773
Schistosoma mansoni	DNA helicase recq5	0.0011	0.0296	0.024
Trypanosoma cruzi	polo-like protein kinase, putative	0.01	0.5439	1
Toxoplasma gondii	ATP-dependent DNA helicase, RecQ family protein	0.0011	0.0296	0.115
Toxoplasma gondii	ATP-dependent DNA helicase, RecQ family protein	0.0011	0.0296	0.115
Plasmodium vivax	glutathione reductase, putative	0.005	0.2569	1
Schistosoma mansoni	Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein)	0.0049	0.2475	0.2432
Schistosoma mansoni	DNA polymerase eta	0.0048	0.2416	0.2373
Trichomonas vaginalis	DNA polymerase eta, putative	0.0021	0.0867	0.0793
Brugia malayi	MH2 domain containing protein	0.0009	0.0188	0.0189
Echinococcus multilocularis	dna polymerase eta	0.0048	0.2416	0.2271
Schistosoma mansoni	smad	0.0009	0.0188	0.0131
Plasmodium falciparum	dihydrolipoyl dehydrogenase, apicoplast	0.0017	0.0689	0.2517
Trypanosoma brucei	dihydrolipoamide dehydrogenase	0.0017	0.0689	0.1175
Schistosoma mansoni	smad1 5 8 and	0.0009	0.0188	0.0131
Mycobacterium tuberculosis	NADPH-dependent mycothiol reductase Mtr	0.005	0.2569	0.2985
Schistosoma mansoni	blooms syndrome DNA helicase	0.002	0.0846	0.0793
Echinococcus granulosus	guanine nucleotide binding protein Gs subunit	0.0049	0.2475	0.2331
Echinococcus granulosus	terminal deoxycytidyl transferase rev1	0.0021	0.0867	0.0692
Brugia malayi	MH1 domain containing protein	0.0009	0.0188	0.0189
Schistosoma mansoni	hypothetical protein	0.018	1	1
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Echinococcus granulosus	dihydrolipoamide dehydrogenase	0.0017	0.0689	0.0512
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Mycobacterium tuberculosis	Probable oxidoreductase	0.0127	0.6986	1
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trichomonas vaginalis	DNA polymerase IV / kappa, putative	0.0021	0.0867	0.0793
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Mycobacterium tuberculosis	Possible DNA-damage-inducible protein P DinP (DNA polymerase V) (pol IV 2) (DNA nucleotidyltransferase (DNA-directed))	0.0021	0.0867	0.0281
Brugia malayi	dihydrolipoyl dehydrogenase, mitochondrial precursor, putative	0.0017	0.0689	0.0917
Echinococcus multilocularis	thioredoxin glutathione reductase	0.005	0.2569	0.2427
Mycobacterium tuberculosis	Probable membrane NADH dehydrogenase NdhA	0.0115	0.6254	0.8837
Trypanosoma brucei	trypanothione reductase	0.005	0.2569	0.4668
Toxoplasma gondii	thioredoxin reductase	0.005	0.2569	1
Plasmodium falciparum	ADP-dependent DNA helicase RecQ	0.0022	0.0976	0.3657
Loa Loa (eye worm)	hypothetical protein	0.0011	0.0296	0.0341
Entamoeba histolytica	hypothetical protein	0.0038	0.1881	0.3459
Loa Loa (eye worm)	ImpB/MucB/SamB family protein	0.0021	0.0867	0.1159
Brugia malayi	Bloom's syndrome protein homolog	0.0026	0.1153	0.1589
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Mycobacterium ulcerans	dihydrolipoamide dehydrogenase, LpdB	0.0017	0.0689	0.7811
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Leishmania major	acetoin dehydrogenase e3 component-like protein	0.0017	0.0689	0.1175
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Loa Loa (eye worm)	RecQ helicase	0.0026	0.1153	0.1569
Loa Loa (eye worm)	MH1 domain-containing protein	0.0009	0.0188	0.0187
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Mycobacterium tuberculosis	Probable dehydrogenase	0.0115	0.6254	0.8837
Loa Loa (eye worm)	MH2 domain-containing protein	0.0009	0.0188	0.0187
Leishmania major	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Loa Loa (eye worm)	MH2 domain-containing protein	0.0127	0.6955	0.9874
Toxoplasma gondii	ATP-dependent DNA helicase, RecQ family protein	0.0017	0.0668	0.2602
Schistosoma mansoni	hypothetical protein	0.0038	0.1881	0.1835
Brugia malayi	ImpB/MucB/SamB family protein	0.0048	0.2416	0.342
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Brugia malayi	glutathione reductase	0.005	0.2569	0.3642
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Mycobacterium ulcerans	flavoprotein disulfide reductase	0.0017	0.0689	0.7811
Plasmodium vivax	ADP-dependent DNA helicase RecQ, putative	0.0017	0.068	0.248
Brugia malayi	ATP-dependent DNA helicase, RecQ family protein	0.0011	0.0296	0.0346
Trypanosoma brucei	DNA polymerase IV, putative	0.0021	0.0867	0.1504
Echinococcus multilocularis	geminin	0.018	1	1
Brugia malayi	Pyridine nucleotide-disulphide oxidoreductase, dimerisation domain containing protein	0.0013	0.0425	0.0533
Entamoeba histolytica	deoxycytidyl transferase, putative	0.0021	0.0867	0.1594
Trichomonas vaginalis	CAMK family protein kinase	0.005	0.2537	0.4157
Loa Loa (eye worm)	transcription factor SMAD2	0.0127	0.6955	0.9874
Trypanosoma brucei	DNA polymerase eta, putative	0.0048	0.2416	0.4384
Toxoplasma gondii	ImpB/MucB/SamB family protein	0.0033	0.1607	0.6254
Schistosoma mansoni	dihydrolipoamide dehydrogenase	0.0017	0.0689	0.0636
Loa Loa (eye worm)	glutathione reductase	0.005	0.2569	0.3596
Trichomonas vaginalis	glutathione reductase, putative	0.0017	0.0689	0.0436
Brugia malayi	alpha keto acid dehydrogenase complex, E3 component, lipoamide dehydrogenase	0.0013	0.0425	0.0533
Toxoplasma gondii	NADPH-glutathione reductase	0.0017	0.0689	0.2684
Brugia malayi	Smad1	0.0009	0.0188	0.0189
Brugia malayi	MH2 domain containing protein	0.0009	0.0188	0.0189
Trypanosoma brucei	DNA polymerase kappa, putative	0.0014	0.0502	0.0827
Mycobacterium tuberculosis	Probable reductase	0.0115	0.6254	0.8837
Mycobacterium tuberculosis	Conserved hypothetical protein	0.0021	0.0867	0.0281
Schistosoma mansoni	serine/threonine protein kinase	0.01	0.5439	0.5412
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Trypanosoma brucei	dihydrolipoamide dehydrogenase, point mutation	0.0017	0.0689	0.1175
Giardia lamblia	DINP protein human, muc B family	0.0021	0.0867	0.1504
Echinococcus granulosus	dna polymerase eta	0.0048	0.2416	0.2271
Leishmania major	trypanothione reductase	0.005	0.2569	0.4668
Trypanosoma cruzi	trypanothione reductase, putative	0.005	0.2569	0.4668
Echinococcus granulosus	Basic leucine zipper bZIP transcription	0.0038	0.1881	0.1726
Trypanosoma cruzi	polo-like protein kinase, putative	0.01	0.5439	1
Schistosoma mansoni	hypothetical protein	0.018	1	1
Mycobacterium tuberculosis	Probable NADH dehydrogenase Ndh	0.0115	0.6254	0.8837
Mycobacterium ulcerans	DNA polymerase IV	0.0021	0.0867	1
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Mycobacterium ulcerans	DNA polymerase IV	0.0021	0.0867	1
Trichomonas vaginalis	DNA helicase recq1, putative	0.0026	0.1153	0.137
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Trypanosoma brucei	DNA polymerase IV, putative	0.0021	0.0867	0.1504
Chlamydia trachomatis	dihydrolipoyl dehydrogenase	0.0017	0.0689	0.5
Trichomonas vaginalis	CAMK family protein kinase	0.01	0.5439	1
Echinococcus multilocularis	bloom syndrome protein	0.0026	0.1153	0.0984
Loa Loa (eye worm)	thioredoxin reductase	0.005	0.2569	0.3596
Loa Loa (eye worm)	ATP-dependent DNA helicase	0.0011	0.0296	0.0341
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma brucei	ATP-dependent DEAD/H DNA helicase recQ, putative	0.0014	0.0473	0.0773
Plasmodium vivax	dihydrolipoyl dehydrogenase, apicoplast, putative	0.0017	0.0689	0.2517
Leishmania major	ATP-dependent DEAD/H DNA helicase recQ, putative	0.0014	0.0473	0.0773
Plasmodium falciparum	ATP-dependent DNA helicase Q1	0.0011	0.0296	0.0949
Wolbachia endosymbiont of Brugia malayi	dihydrolipoamide dehydrogenase E3 component	0.0017	0.0689	0.5
Giardia lamblia	Sgs1 DNA helicase, putative	0.0011	0.0296	0.0443
Echinococcus multilocularis	ATP dependent DNA helicase Q5	0.0011	0.0296	0.011
Echinococcus granulosus	bloom syndrome protein	0.0026	0.1153	0.0984
Trypanosoma brucei	polo-like protein kinase	0.01	0.5439	1
Leishmania major	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Entamoeba histolytica	hypothetical protein	0.0038	0.1881	0.3459
Mycobacterium ulcerans	dihydrolipoamide dehydrogenase	0.0017	0.0689	0.7811
Echinococcus granulosus	serine:threonine protein kinase PLK1	0.01	0.5439	0.5351
Brugia malayi	MH2 domain containing protein	0.0127	0.6955	1
Schistosoma mansoni	rab geranylgeranyl transferase alpha subunit	0.0021	0.0867	0.0814
Echinococcus multilocularis	Basic leucine zipper (bZIP) transcription	0.0038	0.1881	0.1726
Schistosoma mansoni	DNA helicase recq1	0.0011	0.0296	0.024
Echinococcus multilocularis	ATP dependent DNA helicase Q1	0.0011	0.0296	0.011
Schistosoma mansoni	smad1 5 8 and	0.0009	0.0188	0.0131
Schistosoma mansoni	transcription factor LCR-F1	0.0038	0.1881	0.1835
Echinococcus granulosus	thioredoxin glutathione reductase	0.005	0.2569	0.2427
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Echinococcus granulosus	ATP dependent DNA helicase Q5	0.0011	0.0296	0.011
Wolbachia endosymbiont of Brugia malayi	dihydrolipoamide dehydrogenase E3 component	0.0017	0.0689	0.5
Plasmodium falciparum	thioredoxin reductase	0.0017	0.0689	0.2517
Echinococcus granulosus	ATP dependent DNA helicase Q1	0.0011	0.0296	0.011
Toxoplasma gondii	pyruvate dehydrogenase complex subunit PDH-E3II	0.0017	0.0689	0.2684
Mycobacterium tuberculosis	NAD(P)H quinone reductase LpdA	0.0127	0.6986	1
Leishmania major	2-oxoglutarate dehydrogenase, e3 component, lipoamidedehydrogenase-like protein	0.0017	0.0689	0.1175
Echinococcus granulosus	dna polymerase kappa	0.0021	0.0867	0.0692
Onchocerca volvulus	Serine\/threonine kinase homolog	0.01	0.5439	0.5
Loa Loa (eye worm)	PLK/PLK1 protein kinase	0.01	0.5439	0.7703
Leishmania major	DNA polymerase kappa, putative,DNA polymerase IV, putative	0.0021	0.0867	0.1504
Trichomonas vaginalis	mercuric reductase, putative	0.0017	0.0689	0.0436
Echinococcus multilocularis	dihydrolipoamide dehydrogenase	0.0017	0.0689	0.0512
Schistosoma mansoni	Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein)	0.0049	0.2475	0.2432
Trypanosoma brucei	unspecified product	0.0014	0.0502	0.0827
Schistosoma mansoni	Smad4	0.0009	0.0188	0.0131
Trypanosoma brucei	unspecified product	0.0021	0.0867	0.1504
Schistosoma mansoni	terminal deoxycytidyl transferase	0.0021	0.0867	0.0814
Brugia malayi	GTP-binding regulatory protein Gs alpha-S chain, putative	0.0049	0.2475	0.3506
Brugia malayi	Thioredoxin reductase	0.005	0.2569	0.3642
Trypanosoma brucei	DNA polymerase IV, putative	0.0021	0.0867	0.1504
Schistosoma mansoni	Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein)	0.0049	0.2475	0.2432
Leishmania major	DNA polymerase eta, putative	0.0033	0.1607	0.2879
Entamoeba histolytica	hypothetical protein	0.0038	0.1881	0.3459
Leishmania major	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma brucei	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Trypanosoma brucei	dihydrolipoamide dehydrogenase	0.0017	0.0689	0.1175
Echinococcus multilocularis	guanine nucleotide binding protein G(s) subunit	0.0049	0.2475	0.2331
Entamoeba histolytica	hypothetical protein	0.0038	0.1881	0.3459
Echinococcus multilocularis	guanine nucleotide binding protein G(s) subunit	0.0049	0.2475	0.2331
Trypanosoma cruzi	DNA polymerase kappa, putative	0.0021	0.0867	0.1504
Brugia malayi	ImpB/MucB/SamB family protein	0.0021	0.0867	0.1174
Brugia malayi	hypothetical protein	0.0038	0.1881	0.2645
Loa Loa (eye worm)	Smad1	0.0009	0.0188	0.0187
Schistosoma mansoni	smad1 5 8 and	0.0009	0.0188	0.0131
Leishmania major	DNA polymerase eta, putative	0.0048	0.2416	0.4384
Mycobacterium tuberculosis	Putative ferredoxin reductase	0.0115	0.6254	0.8837
Trypanosoma cruzi	DNA polymerase eta, putative	0.0048	0.2416	0.4384
Trypanosoma cruzi	trypanothione reductase, putative	0.0017	0.0689	0.1175
Plasmodium vivax	thioredoxin reductase, putative	0.005	0.2569	1
Plasmodium falciparum	dihydrolipoyl dehydrogenase, mitochondrial	0.0017	0.0689	0.2517
Giardia lamblia	Kinase, PLK	0.01	0.5439	1
Trypanosoma brucei	DNA polymerase kappa, putative	0.0014	0.0502	0.0827
Schistosoma mansoni	TGF-beta signal transducer Smad2	0.0009	0.0188	0.0131
Echinococcus multilocularis	terminal deoxycytidyl transferase rev1	0.0021	0.0867	0.0692
Echinococcus multilocularis	serine:threonine protein kinase PLK1	0.01	0.5439	0.5351
Trypanosoma cruzi	dihydrolipoamide dehydrogenase, putative	0.0017	0.0689	0.1175
Trypanosoma brucei	dihydrolipoyl dehydrogenase	0.0017	0.0689	0.1175

Activities

Activity type	Activity value	Assay description	Source	Reference
EC100 (functional)	= 0.32 ppm	Anthelmintic activity against benzimidazole-resistant Haemonchus contortus isolate by larva development assay	ChEMBL.	18400497
EC100 (functional)	= 0.32 ppm	Anthelmintic activity against levamisole-resistant Trichostrongylus colubriformis isolate by larva development assay	ChEMBL.	18400497

Phenotypes

Whole-cell/tissue/organism interactions

We have no records of whole-cell/tissue assays done with this compound What does this mean?

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL256758

Bibliographic References

1 literature reference was collected for this gene.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 509385